BR0016737A - 14,15-ciclopropano-androstanos insaturados, processos para a sua preparação e composições farmacêuticas contendo estes compostos - Google Patents

14,15-ciclopropano-androstanos insaturados, processos para a sua preparação e composições farmacêuticas contendo estes compostos

Info

Publication number
BR0016737A
BR0016737A BR0016737-1A BR0016737A BR0016737A BR 0016737 A BR0016737 A BR 0016737A BR 0016737 A BR0016737 A BR 0016737A BR 0016737 A BR0016737 A BR 0016737A
Authority
BR
Brazil
Prior art keywords
compounds
cyclopropane
unsaturated
preparation
pharmaceutical compositions
Prior art date
Application number
BR0016737-1A
Other languages
English (en)
Inventor
Sven Ring
Walter Elger
Guenter Kaufmann
Original Assignee
Jenapharm Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jenapharm Gmbh filed Critical Jenapharm Gmbh
Publication of BR0016737A publication Critical patent/BR0016737A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002—Carbocyclic rings fused
    • C07J53/004—3 membered carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/34—Gestagens

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)

Abstract

"14,15-CICLOPROPANO-ANDROSTANOS INSATURADOS, PROCESSOS PARA A SUA PREPARAçãO E COMPOSIçõES FARMACêUTICAS CONTENDO ESTES COMPOSTOS". A invenção refere-se a novos 14,15-ciclopropano-androstanos insaturados da fórmula geral (I), sua preparação e composições farmacêuticas contendo estes compostos. Os compostos da fórmula (I) são compostos de ação gestagênica e/ou androgênica.
BR0016737-1A 1999-12-08 2000-11-21 14,15-ciclopropano-androstanos insaturados, processos para a sua preparação e composições farmacêuticas contendo estes compostos BR0016737A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19959696A DE19959696A1 (de) 1999-12-08 1999-12-08 Ungesättigte 14,15-Cyclopropano-Androstane, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
PCT/EP2000/011557 WO2001042275A1 (de) 1999-12-08 2000-11-21 Ungesättigte 14,15-cyclopropano-androstane, verfahren zu ihrer herstellung und diese verbindungen enthaltende pharmazeutische zusammensetzungen

Publications (1)

Publication Number Publication Date
BR0016737A true BR0016737A (pt) 2002-11-05

Family

ID=7932216

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0016737-1A BR0016737A (pt) 1999-12-08 2000-11-21 14,15-ciclopropano-androstanos insaturados, processos para a sua preparação e composições farmacêuticas contendo estes compostos

Country Status (26)

Country Link
US (2) USRE39862E1 (pt)
EP (1) EP1235850B1 (pt)
JP (1) JP3793088B2 (pt)
KR (1) KR100468341B1 (pt)
CN (1) CN1205219C (pt)
AT (1) ATE275576T1 (pt)
AU (1) AU774384B2 (pt)
BG (1) BG106861A (pt)
BR (1) BR0016737A (pt)
CA (1) CA2393758C (pt)
CZ (1) CZ20022005A3 (pt)
DE (2) DE19959696A1 (pt)
DK (1) DK1235850T3 (pt)
EE (1) EE200200302A (pt)
ES (1) ES2226949T3 (pt)
HU (1) HUP0203655A3 (pt)
IL (2) IL150082A0 (pt)
MX (1) MXPA02005644A (pt)
NO (1) NO323376B1 (pt)
PL (1) PL356061A1 (pt)
PT (1) PT1235850E (pt)
RU (1) RU2244718C2 (pt)
SI (1) SI1235850T1 (pt)
SK (1) SK8092002A3 (pt)
WO (1) WO2001042275A1 (pt)
ZA (1) ZA200205362B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10104327A1 (de) * 2001-01-24 2002-07-25 Schering Ag 11beta-Halogensteroide, deren Herstellung und Verwendung zur Herstellung von Arzneimitteln sowie 11beta-Halogensteroide enthaltende pharmazeutische Präparate

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE31269C (de) * B.GERVAIS in Montmorillon Vienne, Frankreich Transportable Brauerei für Kleinbetrieb
DE33136C (de) * J. KENDAL und M. LAVAL in London Uhr mit zwei Zifferblättern und dazu gehörigem Zeigerstellwerk
NL215687A (pt) * 1956-03-26
CH376097A (de) * 1956-04-23 1964-03-31 Farmaceutici Italia Verfahren zur Herstellung von 4-Halogen-3-keto- 4-steroiden
US2895969A (en) * 1957-09-23 1959-07-21 Syntex Sa Cyclopentanophenanthrene derivatives
GB839908A (en) * 1957-12-24 1960-06-29 Farmaceutici Italia 4,17ª‡-dihydroxy progesterone and its esters and the preparation thereof
GB874572A (en) * 1959-02-18 1961-08-10 Farmaceutici Italia A method for the production of new ketosteroid compounds
GB928714A (en) * 1961-02-10 1963-06-12 Farmaceutici Italia Process for the preparation of 4-hydroxy-3-keto-í¸-steroids
GB991804A (en) * 1962-03-13 1965-05-12 Piero Gomarasca New derivatives of cyclopentanophenanthrene and processes for their preparation
US3239512A (en) * 1964-08-04 1966-03-08 Syntex Corp 17-tetrahydropyranylether of 4-chlorotestosterone
DE19537626A1 (de) * 1995-10-10 1997-04-17 Jenapharm Gmbh Steroide mit einer 14, 15-Methylengruppe
DE19827523A1 (de) * 1998-06-22 1999-12-23 Jenapharm Gmbh Ungesättigte 14,15-Cyclopropano-Androstane, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Präparate

Also Published As

Publication number Publication date
DK1235850T3 (da) 2005-01-17
CZ20022005A3 (cs) 2002-10-16
CN1433425A (zh) 2003-07-30
AU774384B2 (en) 2004-06-24
RU2244718C2 (ru) 2005-01-20
ATE275576T1 (de) 2004-09-15
NO20022712D0 (no) 2002-06-07
CN1205219C (zh) 2005-06-08
KR100468341B1 (ko) 2005-01-27
HUP0203655A2 (hu) 2003-03-28
CA2393758C (en) 2007-06-12
EP1235850B1 (de) 2004-09-08
JP3793088B2 (ja) 2006-07-05
EP1235850A1 (de) 2002-09-04
EE200200302A (et) 2003-06-16
CA2393758A1 (en) 2001-06-14
BG106861A (bg) 2003-02-28
DE19959696A1 (de) 2001-06-21
IL150082A (en) 2007-05-15
NO20022712L (no) 2002-06-07
SI1235850T1 (en) 2005-04-30
NO323376B1 (no) 2007-04-16
MXPA02005644A (es) 2002-12-13
WO2001042275A1 (de) 2001-06-14
AU1703801A (en) 2001-06-18
DE50007708D1 (de) 2004-10-14
ZA200205362B (en) 2003-10-06
PL356061A1 (en) 2004-06-14
IL150082A0 (en) 2002-12-01
KR20030028448A (ko) 2003-04-08
HUP0203655A3 (en) 2004-07-28
US6710039B1 (en) 2004-03-23
USRE39862E1 (en) 2007-09-25
ES2226949T3 (es) 2005-04-01
SK8092002A3 (en) 2003-05-02
JP2003516416A (ja) 2003-05-13
PT1235850E (pt) 2005-01-31

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: SCHERING AG (DE)

Free format text: TRANSFERIDO DE: JENAPHARM GMBH AND CO. KG

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O, 10, 13 E 25 DA LPI.

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.