BR0012192A - Derivado de ácido quinolinocarboxìlico ou seus sais - Google Patents

Derivado de ácido quinolinocarboxìlico ou seus sais

Info

Publication number
BR0012192A
BR0012192A BR0012192-4A BR0012192A BR0012192A BR 0012192 A BR0012192 A BR 0012192A BR 0012192 A BR0012192 A BR 0012192A BR 0012192 A BR0012192 A BR 0012192A
Authority
BR
Brazil
Prior art keywords
salts
derived
extremely high
quinolinocarboxylic
quinolinocarboxylic acid
Prior art date
Application number
BR0012192-4A
Other languages
English (en)
Inventor
Akira Yazaki
Yoshiko Niino
Yasuhiro Kuramoto
Yuzo Hirao
Yoshihiro Ohshita
Norihiro Hayashi
Hirotaka Amano
Original Assignee
Wakunaga Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wakunaga Pharma Co Ltd filed Critical Wakunaga Pharma Co Ltd
Publication of BR0012192A publication Critical patent/BR0012192A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

"DERIVADO DE áCIDO QUINOLINOCARBOXìLICO OU SEUS SAIS". A presente invenção refere-se a ácido 1-(6-amino-3,5difluoropiridin-2-il)-8-bromo-7-(3-etilaminoazetidin-1-il)6- fluoro-4-oxo-1,4-di-hidroquinolino-3-carboxílico ou um de seus sais, bem como a um remédio que o contém. Este composto possui funções características e, quando administrado oralmente, apresenta meia-vida em sangue e biodisponibilidade extremamente altas, retendo propriedades de efeitos anti-microbianos extremamente altos e baixa toxicidade. Ele pode ser amplamente utilizado como preventivo, terapêutico e similares para diversas doenças infecciosas de seres humanos e animais.
BR0012192-4A 1999-07-01 2000-06-22 Derivado de ácido quinolinocarboxìlico ou seus sais BR0012192A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP18749299 1999-07-01
PCT/JP2000/004096 WO2001002390A1 (fr) 1999-07-01 2000-06-22 Derive d'acide quinolinecarboxylique et ses sels

Publications (1)

Publication Number Publication Date
BR0012192A true BR0012192A (pt) 2002-06-18

Family

ID=16207019

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0012192-4A BR0012192A (pt) 1999-07-01 2000-06-22 Derivado de ácido quinolinocarboxìlico ou seus sais

Country Status (25)

Country Link
US (1) US6858625B1 (pt)
EP (1) EP1193266B1 (pt)
JP (1) JP3477465B2 (pt)
KR (1) KR100628414B1 (pt)
CN (1) CN1157389C (pt)
AT (1) ATE248162T1 (pt)
AU (1) AU766014B2 (pt)
BR (1) BR0012192A (pt)
CA (1) CA2376760C (pt)
CZ (1) CZ302033B6 (pt)
DE (1) DE60004846T2 (pt)
DK (1) DK1193266T3 (pt)
ES (1) ES2206257T3 (pt)
HK (1) HK1047103B (pt)
HU (1) HUP0201549A3 (pt)
IL (2) IL147043A0 (pt)
MX (1) MXPA02000103A (pt)
NO (1) NO321803B1 (pt)
NZ (1) NZ516201A (pt)
PT (1) PT1193266E (pt)
RU (1) RU2236408C2 (pt)
SK (1) SK285814B6 (pt)
TW (1) TW576832B (pt)
WO (1) WO2001002390A1 (pt)
ZA (1) ZA200110357B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3477466B2 (ja) 1999-09-02 2003-12-10 湧永製薬株式会社 キノリンカルボン酸誘導体又はその塩
US7172535B2 (en) * 2004-10-28 2007-02-06 Volmar John F Upper back exercise machine and method of use
MX2007005892A (es) 2004-11-17 2007-06-19 Wakunaga Pharma Co Ltd Derivados de acido piridonacarboxilico novedosos y sales de los mismos.
US8497378B2 (en) * 2008-09-24 2013-07-30 Rib-X Pharmaceuticals, Inc. Process for making quinolone compounds

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO177302C (no) * 1989-03-16 1995-08-23 Esteve Labor Dr Analogifremgangsmåte til fremstilling av terapeutisk aktive substituerte azetidinylkinolon(naftyridon)karboksylsyrederivater
CA2168764C (en) * 1993-08-13 2000-01-18 Sung June Yoon Novel quinolone carboxylic acid derivatives
CA2290712C (en) * 1995-09-22 2003-09-09 Wakunaga Pharmaceutical Co., Ltd. Novel pyridonecarboxylic acid derivatives or their salts, and antibacterial agents containing the same as their effective components
EP0897919B1 (en) * 1996-04-19 2004-06-16 Wakunaga Pharmaceutical Co., Ltd. Novel pyridonecarboxylic acid derivatives or salts thereof and antibacterial agents containing the same as the active ingredient
KR100516379B1 (ko) 1996-11-28 2005-09-26 와쿠나가 세이야쿠 가부시키 가이샤 신규 피리돈카르복실산 유도체 또는 그의 염 및 이를 유효 성분으로 하는 의약
DE19652239A1 (de) * 1996-12-16 1998-06-18 Bayer Ag Verwendung von 7-(2-Oxa-5,8-diazabicyclo[4.3.0]non-8-yl)-chinolon- und -naphthyridoncarbonsäure-Derivaten zur Therapie von Helicobacter-pylori-Infektionen und den damit assoziierten gastroduodenalen Erkrankungen
JPH11292873A (ja) 1998-04-07 1999-10-26 Dainippon Pharmaceut Co Ltd キノロンカルボン酸誘導体の製造方法およびその中間体

Also Published As

Publication number Publication date
DK1193266T3 (da) 2003-11-24
SK285814B6 (sk) 2007-08-02
SK19162001A3 (sk) 2002-06-04
CA2376760C (en) 2008-11-25
NO20016378D0 (no) 2001-12-27
CZ302033B6 (cs) 2010-09-08
CN1157389C (zh) 2004-07-14
PT1193266E (pt) 2003-12-31
NO20016378L (no) 2002-02-28
MXPA02000103A (es) 2003-07-21
DE60004846T2 (de) 2004-06-03
CN1358183A (zh) 2002-07-10
ZA200110357B (en) 2002-12-18
US6858625B1 (en) 2005-02-22
CZ20014598A3 (cs) 2002-05-15
TW576832B (en) 2004-02-21
AU5567900A (en) 2001-01-22
KR100628414B1 (ko) 2006-09-26
ATE248162T1 (de) 2003-09-15
KR20020020733A (ko) 2002-03-15
WO2001002390A1 (fr) 2001-01-11
HK1047103A1 (en) 2003-02-07
EP1193266A4 (en) 2002-08-14
HK1047103B (zh) 2005-04-08
IL147043A (en) 2007-07-04
ES2206257T3 (es) 2004-05-16
IL147043A0 (en) 2002-08-14
NZ516201A (en) 2003-06-30
DE60004846D1 (de) 2003-10-02
RU2236408C2 (ru) 2004-09-20
NO321803B1 (no) 2006-07-03
CA2376760A1 (en) 2001-01-11
HUP0201549A3 (en) 2003-11-28
JP3477465B2 (ja) 2003-12-10
EP1193266B1 (en) 2003-08-27
EP1193266A1 (en) 2002-04-03
AU766014B2 (en) 2003-10-09
HUP0201549A2 (en) 2002-08-28

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Legal Events

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B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O, 10 (VIII), 11 E 13 DA LPI

B09T Decision of refusal: decision cancelled [chapter 9.2.1 patent gazette]

Free format text: REFERENTE A RPI 2039 DE 02/02/2010.

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) 8O, 11, 13, 24 E 25 DA LPI.

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.