BR0008511A - Sistemas tiazol policìclicos e seu emprego como anoréticos contendo estes compostos - Google Patents

Sistemas tiazol policìclicos e seu emprego como anoréticos contendo estes compostos

Info

Publication number
BR0008511A
BR0008511A BR0008511-1A BR0008511A BR0008511A BR 0008511 A BR0008511 A BR 0008511A BR 0008511 A BR0008511 A BR 0008511A BR 0008511 A BR0008511 A BR 0008511A
Authority
BR
Brazil
Prior art keywords
compounds
anoretics
thiazole systems
polycyclic thiazole
polycyclic
Prior art date
Application number
BR0008511-1A
Other languages
English (en)
Inventor
Gerhard Jaehne
Karl Geisen
Hans-Jochen Lang
Martin Bickel
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of BR0008511A publication Critical patent/BR0008511A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/84—Naphthothiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Patente de Invenção: "SISTEMAS TIAZOL POLICìCLICOS E SEU EMPREGO COMO ANORéTICOS CONTENDO ESTES COMPOSTOS". A invenção refere-se a sistemas tiazol policíclicos bem como aos seus sais fisiologicamente compatíveis e derivados fisiologicamente funcionais. São descritos compostos de fórmula I na qual os radicais têm os significados indicados, bem como seus sais fisiologicamente compatíveis e processos para a sua preparação. Os compostos prestam-se, por exemplo, como anoréticos.
BR0008511-1A 1999-02-26 2000-02-05 Sistemas tiazol policìclicos e seu emprego como anoréticos contendo estes compostos BR0008511A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19908533A DE19908533A1 (de) 1999-02-26 1999-02-26 Polycyclische Thiazol-Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen
PCT/EP2000/000927 WO2000051997A1 (de) 1999-02-26 2000-02-05 Polycyclische thiazol-systeme und ihre verwendung als anorektika

Publications (1)

Publication Number Publication Date
BR0008511A true BR0008511A (pt) 2002-04-02

Family

ID=7899078

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0008511-1A BR0008511A (pt) 1999-02-26 2000-02-05 Sistemas tiazol policìclicos e seu emprego como anoréticos contendo estes compostos

Country Status (18)

Country Link
US (1) US6187801B1 (pt)
EP (1) EP1183247B1 (pt)
JP (1) JP4728485B2 (pt)
KR (1) KR20020000545A (pt)
CN (1) CN1149205C (pt)
AT (1) ATE296295T1 (pt)
AU (1) AU762802B2 (pt)
BR (1) BR0008511A (pt)
CA (1) CA2364903A1 (pt)
CO (1) CO5180595A1 (pt)
DE (2) DE19908533A1 (pt)
DK (1) DK1183247T3 (pt)
ES (1) ES2241574T3 (pt)
HK (1) HK1042300B (pt)
PT (1) PT1183247E (pt)
TW (1) TW593294B (pt)
WO (1) WO2000051997A1 (pt)
ZA (1) ZA200106440B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19908535A1 (de) 1999-02-26 2000-08-31 Aventis Pharma Gmbh Verwendung von polycyclischen Thiazol-Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas
AU2001244136B2 (en) * 2000-02-26 2005-04-14 Sanofi-Aventis Deutschland Gmbh 8,8a-dihydro-indeno[1,2-d]thiazole derivatives with a sulphonamido or sulphono substituent in the 2 position, method for production thereof and use thereof as medicament
DE10142663B4 (de) * 2001-08-31 2004-08-19 Aventis Pharma Deutschland Gmbh C2-Disubstituierte Indan-1-ol-Systeme
KR100712171B1 (ko) * 2004-09-17 2007-05-02 김진우 폐타이어를 이용한 조립식 배관블록
MX2010010659A (es) * 2008-03-31 2010-10-26 Genentech Inc Compuestos de benzopirano y benzoxepina, inhibidores de fosfoinoinositida 3-cinasas y metodos para utilizarlos.
CN104744491B (zh) * 2009-09-28 2017-07-11 霍夫曼-拉罗奇有限公司 苯并氧杂氮杂*pi3k抑制剂化合物和使用方法
CN102762574B (zh) 2009-09-28 2015-12-02 霍夫曼-拉罗奇有限公司 苯并氧杂*pi3k抑制剂化合物和使用方法
US9090628B2 (en) 2011-03-21 2015-07-28 Genentech, Inc. Benzoxazepin compounds selective for PI3K P110 delta and methods of use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2640358A1 (de) * 1976-09-08 1978-03-16 Hoechst Ag Thiazolidinderivate und verfahren zu ihrer herstellung
WO1995024399A1 (fr) * 1994-03-11 1995-09-14 Yamanouchi Pharmaceutical Co., Ltd. Agoniste de recepteur 5-ht3, nouveau derive de thiazole et intermediaire destine a son obtention
JPH1179993A (ja) * 1997-09-05 1999-03-23 Sumitomo Pharmaceut Co Ltd 免疫抑制剤
DE19831878C2 (de) * 1998-07-17 2001-05-17 Aventis Pharma Gmbh Polycyclische Thiazolidin-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE19908535A1 (de) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Verwendung von polycyclischen Thiazol-Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas

Also Published As

Publication number Publication date
ES2241574T3 (es) 2005-11-01
CN1341108A (zh) 2002-03-20
CO5180595A1 (es) 2002-07-30
DE19908533A1 (de) 2000-08-31
HK1042300A1 (en) 2002-08-09
DK1183247T3 (da) 2005-09-19
CA2364903A1 (en) 2000-09-08
KR20020000545A (ko) 2002-01-05
JP2002538150A (ja) 2002-11-12
AU762802B2 (en) 2003-07-03
JP4728485B2 (ja) 2011-07-20
AU2441600A (en) 2000-09-21
EP1183247B1 (de) 2005-05-25
HK1042300B (zh) 2004-12-10
US6187801B1 (en) 2001-02-13
PT1183247E (pt) 2005-07-29
WO2000051997A1 (de) 2000-09-08
ATE296295T1 (de) 2005-06-15
TW593294B (en) 2004-06-21
ZA200106440B (en) 2002-03-06
DE50010403D1 (de) 2005-06-30
CN1149205C (zh) 2004-05-12
EP1183247A1 (de) 2002-03-06

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A, 8A E 9A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 NA RPI2003 DE 26/05/2009.