PT1157015E - Utilizacao de sistemas 2-amino-triazole policiclicos para a preparacao de medicamentos para tratamento de perturbacoes lipometabolicas, da obesidade e da diabetes tipo ii - Google Patents

Utilizacao de sistemas 2-amino-triazole policiclicos para a preparacao de medicamentos para tratamento de perturbacoes lipometabolicas, da obesidade e da diabetes tipo ii

Info

Publication number
PT1157015E
PT1157015E PT00910642T PT00910642T PT1157015E PT 1157015 E PT1157015 E PT 1157015E PT 00910642 T PT00910642 T PT 00910642T PT 00910642 T PT00910642 T PT 00910642T PT 1157015 E PT1157015 E PT 1157015E
Authority
PT
Portugal
Prior art keywords
polycyclic
preparation
perturbacoes
lipometabolic
obesity
Prior art date
Application number
PT00910642T
Other languages
English (en)
Inventor
Karl Geisen
Gerhard Jahne
Lang Hans-Jochen
Bickel Martin
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of PT1157015E publication Critical patent/PT1157015E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT00910642T 1999-02-26 2000-02-05 Utilizacao de sistemas 2-amino-triazole policiclicos para a preparacao de medicamentos para tratamento de perturbacoes lipometabolicas, da obesidade e da diabetes tipo ii PT1157015E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19908538A DE19908538A1 (de) 1999-02-26 1999-02-26 Polycyclische 2-Amino-Thiazol Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen

Publications (1)

Publication Number Publication Date
PT1157015E true PT1157015E (pt) 2005-08-31

Family

ID=7899082

Family Applications (1)

Application Number Title Priority Date Filing Date
PT00910642T PT1157015E (pt) 1999-02-26 2000-02-05 Utilizacao de sistemas 2-amino-triazole policiclicos para a preparacao de medicamentos para tratamento de perturbacoes lipometabolicas, da obesidade e da diabetes tipo ii

Country Status (15)

Country Link
US (1) US6251922B1 (pt)
EP (1) EP1157015B1 (pt)
JP (1) JP4728484B2 (pt)
KR (1) KR20010102390A (pt)
CN (1) CN1148362C (pt)
AT (1) ATE295357T1 (pt)
AU (1) AU763111B2 (pt)
BR (1) BR0008510A (pt)
CA (1) CA2364900A1 (pt)
DE (2) DE19908538A1 (pt)
ES (1) ES2240070T3 (pt)
HK (1) HK1043117B (pt)
PT (1) PT1157015E (pt)
WO (1) WO2000051995A1 (pt)
ZA (1) ZA200106198B (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19908537A1 (de) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Verwendung von polycyclischen 2-Amino-Thiazol Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas
WO2002009701A1 (en) * 2000-08-01 2002-02-07 University Of Virginia Patent Foundation Use of selective adenosine a1 receptor agonists, antagonists and allosteric enhancers to manipulate angiogenesis
CA2471989A1 (en) * 2002-01-16 2003-07-31 University Of Virginia Patent Foundation 2-aminothiazole allosteric enhancers of a1 adenosine receptors
PE20091720A1 (es) * 2008-03-31 2009-11-26 Genentech Inc Compuestos de benzopirano y benzoxepina como inhibidores de pi3k
PL2483278T3 (pl) 2009-09-28 2014-05-30 Hoffmann La Roche Związki benzoksazepinowe stanowiące inhibitor pi3k i ich zastosowanie w leczeniu nowotworu
MX2012003641A (es) 2009-09-28 2012-04-30 Hoffmann La Roche Compuestos de benzoxepina inhibidores de la pi3x y metodos de uso.
WO2011059784A1 (en) * 2009-10-29 2011-05-19 Bristol-Myers Squibb Company Tricyclic heterocyclic compounds
BR112013024122A2 (pt) 2011-03-21 2019-09-24 Hoffmann La Roche compostos de benzoxazepina seletivos para p110 delta pi3k e métodos de uso
WO2018045149A1 (en) 2016-09-02 2018-03-08 Bristol-Myers Squibb Company Substituted tricyclic heterocyclic compounds
US11046646B2 (en) 2017-08-09 2021-06-29 Bristol-Myers Squibb Company Alkylphenyl compounds
WO2019032631A1 (en) 2017-08-09 2019-02-14 Bristol-Myers Squibb Company OXIME ETHER COMPOUNDS

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4082773A (en) * 1972-07-03 1978-04-04 E. R. Squibb & Sons, Inc. Tricyclic tetrahydro naphthaleneols and related compounds
DE2640358A1 (de) * 1976-09-08 1978-03-16 Hoechst Ag Thiazolidinderivate und verfahren zu ihrer herstellung
CA1292226C (en) * 1986-01-16 1991-11-19 Terumi Hachiya Indenothiazole derivative and process for preparing the same
IE68593B1 (en) 1989-12-06 1996-06-26 Sanofi Sa Heterocyclic substituted acylaminothiazoles their preparation and pharmaceutical compositions containing them
TW416953B (en) * 1996-09-25 2001-01-01 Takeda Chemical Industries Ltd Tricyclic compounds for eliciting a prostaglandin I2 receptor agonistic effect, their production and use
AU3289299A (en) * 1998-02-19 1999-09-06 Tularik Inc. Antiviral agents
DE19831878C2 (de) * 1998-07-17 2001-05-17 Aventis Pharma Gmbh Polycyclische Thiazolidin-2-yliden Amine, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
DE19908537A1 (de) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Verwendung von polycyclischen 2-Amino-Thiazol Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas

Also Published As

Publication number Publication date
CN1148362C (zh) 2004-05-05
ZA200106198B (en) 2002-05-03
BR0008510A (pt) 2002-02-05
ES2240070T3 (es) 2005-10-16
HK1043117A1 (en) 2002-09-06
JP4728484B2 (ja) 2011-07-20
JP2002538148A (ja) 2002-11-12
HK1043117B (zh) 2004-10-08
US6251922B1 (en) 2001-06-26
ATE295357T1 (de) 2005-05-15
EP1157015B1 (de) 2005-05-11
CN1344263A (zh) 2002-04-10
DE50010285D1 (de) 2005-06-16
AU763111B2 (en) 2003-07-10
KR20010102390A (ko) 2001-11-15
DE19908538A1 (de) 2000-08-31
EP1157015A1 (de) 2001-11-28
AU3278200A (en) 2000-09-21
WO2000051995A1 (de) 2000-09-08
CA2364900A1 (en) 2000-09-08

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