BR0008519A - Aplicação de sistemas tiazol policìclicos para apreparação de medicamentos para a profilaxia outratamento da obesidade - Google Patents

Aplicação de sistemas tiazol policìclicos para apreparação de medicamentos para a profilaxia outratamento da obesidade

Info

Publication number
BR0008519A
BR0008519A BR0008519-7A BR0008519A BR0008519A BR 0008519 A BR0008519 A BR 0008519A BR 0008519 A BR0008519 A BR 0008519A BR 0008519 A BR0008519 A BR 0008519A
Authority
BR
Brazil
Prior art keywords
treatment
obesity
prophylaxis
drugs
preparation
Prior art date
Application number
BR0008519-7A
Other languages
English (en)
Inventor
Gerhard Jaehne
Karl Geisen
Hans-Jochen Lang
Martin Bickel
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of BR0008519A publication Critical patent/BR0008519A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

Patente de Invenção: "APLICAçãO DE SISTEMAS TIAZOLPOLICìCLICOS PARA A PREPARAçãO DE MEDICAMENTOSPARA A PROFILAXIA OU TRATAMENTO DA OBESIDADE". áinvenção refere-se ao emprego de sistemas tiazol policíclicos bemcomo aos seus sais fisiologicamente compatíveis e derivadosfisiologicamente funcionais para a preparação de medicamentospara a profilaxia ou tratamento da obesidade. é descrita aaplicação dos compostos da fórmula I na qual os radicais têm ossignificados indicados, bem como seus sais fisiologicamentecompatíveis e derivados fisiologicamente funcionais para apreparação de um medicamento para a profilaxia ou tratamento daobesidade.
BR0008519-7A 1999-02-26 2000-02-05 Aplicação de sistemas tiazol policìclicos para apreparação de medicamentos para a profilaxia outratamento da obesidade BR0008519A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19908535A DE19908535A1 (de) 1999-02-26 1999-02-26 Verwendung von polycyclischen Thiazol-Systemen zur Herstellung von Medikamenten zur Prophylaxe oder Behandlung von Obesitas
PCT/EP2000/000928 WO2000051579A2 (de) 1999-02-26 2000-02-05 Verwendung von polycyclischen thiazol-systemen zur herstellung von medikamenten zur prophylaxe oder behandlung von obesitas

Publications (1)

Publication Number Publication Date
BR0008519A true BR0008519A (pt) 2001-11-13

Family

ID=7899079

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0008519-7A BR0008519A (pt) 1999-02-26 2000-02-05 Aplicação de sistemas tiazol policìclicos para apreparação de medicamentos para a profilaxia outratamento da obesidade

Country Status (15)

Country Link
US (1) US6329407B1 (pt)
EP (1) EP1156805B1 (pt)
JP (1) JP4728482B2 (pt)
KR (1) KR20010103775A (pt)
CN (1) CN1141940C (pt)
AT (1) ATE273006T1 (pt)
AU (1) AU766813B2 (pt)
BR (1) BR0008519A (pt)
CA (1) CA2362364A1 (pt)
DE (2) DE19908535A1 (pt)
ES (1) ES2221836T3 (pt)
HK (1) HK1044467B (pt)
PT (1) PT1156805E (pt)
WO (1) WO2000051579A2 (pt)
ZA (1) ZA200106439B (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19908533A1 (de) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Polycyclische Thiazol-Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen
FR2870742B1 (fr) * 2004-05-28 2008-03-14 Expanscience Laboratoires Sa Utilisation d'alkyle furannes pour la preparation d'un medicament destine au traitement du diabete, de l'obesite et pour le traitement cosmetique de la cellulite et de la surcharge ponderale
MX2010010659A (es) * 2008-03-31 2010-10-26 Genentech Inc Compuestos de benzopirano y benzoxepina, inhibidores de fosfoinoinositida 3-cinasas y metodos para utilizarlos.
CN104744491B (zh) * 2009-09-28 2017-07-11 霍夫曼-拉罗奇有限公司 苯并氧杂氮杂*pi3k抑制剂化合物和使用方法
CN102762574B (zh) 2009-09-28 2015-12-02 霍夫曼-拉罗奇有限公司 苯并氧杂*pi3k抑制剂化合物和使用方法
US9090628B2 (en) 2011-03-21 2015-07-28 Genentech, Inc. Benzoxazepin compounds selective for PI3K P110 delta and methods of use
US10689955B1 (en) 2019-03-05 2020-06-23 SWM International Inc. Intelligent downhole perforating gun tube and components
US11078762B2 (en) 2019-03-05 2021-08-03 Swm International, Llc Downhole perforating gun tube and components
US11268376B1 (en) 2019-03-27 2022-03-08 Acuity Technical Designs, LLC Downhole safety switch and communication protocol
US11619119B1 (en) 2020-04-10 2023-04-04 Integrated Solutions, Inc. Downhole gun tube extension

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2640358A1 (de) * 1976-09-08 1978-03-16 Hoechst Ag Thiazolidinderivate und verfahren zu ihrer herstellung
NO923126L (no) * 1991-08-13 1993-02-15 Fuji Photo Film Co Ltd Preparat og metode for behandling av canser
US5565479A (en) * 1992-09-14 1996-10-15 Yamanouchi Pharmaceutical Co., Ltd. Condensed thiazole derivative, production process thereof and pharmaceutical composition thereof
WO1995024399A1 (fr) * 1994-03-11 1995-09-14 Yamanouchi Pharmaceutical Co., Ltd. Agoniste de recepteur 5-ht3, nouveau derive de thiazole et intermediaire destine a son obtention
GB9517381D0 (en) * 1995-08-24 1995-10-25 Pharmacia Spa Aryl and heteroaryl piperazine derivatives
DE19908533A1 (de) * 1999-02-26 2000-08-31 Aventis Pharma Gmbh Polycyclische Thiazol-Systeme, Verfahren zu ihrer Herstellung und Arzneimittel enthaltend diese Verbindungen

Also Published As

Publication number Publication date
ZA200106439B (en) 2002-03-06
KR20010103775A (ko) 2001-11-23
EP1156805A2 (de) 2001-11-28
ES2221836T3 (es) 2005-01-16
ATE273006T1 (de) 2004-08-15
CN1341021A (zh) 2002-03-20
WO2000051579A3 (de) 2001-01-11
WO2000051579A2 (de) 2000-09-08
DE50007381D1 (de) 2004-09-16
HK1044467B (zh) 2004-08-20
US6329407B1 (en) 2001-12-11
AU2441700A (en) 2000-09-21
JP2002538101A (ja) 2002-11-12
PT1156805E (pt) 2004-10-29
CN1141940C (zh) 2004-03-17
CA2362364A1 (en) 2000-09-08
EP1156805B1 (de) 2004-08-11
JP4728482B2 (ja) 2011-07-20
HK1044467A1 (en) 2002-10-25
AU766813B2 (en) 2003-10-23
DE19908535A1 (de) 2000-08-31

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 7A, 8A E 9A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 NA RPI2003 DE 26/05/2009.