BG63164B1 - 9-n-етенил производни на 9(s)-еритромициламин - Google Patents

9-n-етенил производни на 9(s)-еритромициламин Download PDF

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Publication number
BG63164B1
BG63164B1 BG101996A BG10199697A BG63164B1 BG 63164 B1 BG63164 B1 BG 63164B1 BG 101996 A BG101996 A BG 101996A BG 10199697 A BG10199697 A BG 10199697A BG 63164 B1 BG63164 B1 BG 63164B1
Authority
BG
Bulgaria
Prior art keywords
alkyl group
group
formula
compound
different
Prior art date
Application number
BG101996A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG101996A (en
Inventor
Nedjelko Kujundzic
Dina Pavlovic
Gabrijela Kobrehel
Gorjana Lazarevski
Zeljko Kelneric
Original Assignee
Pliva Farmaceutska,Kemijska,Prehrambena Ikozmeticka Industrija, Dionicko Drustvo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pliva Farmaceutska,Kemijska,Prehrambena Ikozmeticka Industrija, Dionicko Drustvo filed Critical Pliva Farmaceutska,Kemijska,Prehrambena Ikozmeticka Industrija, Dionicko Drustvo
Publication of BG101996A publication Critical patent/BG101996A/xx
Publication of BG63164B1 publication Critical patent/BG63164B1/bg

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
BG101996A 1996-10-28 1997-10-27 9-n-етенил производни на 9(s)-еритромициламин BG63164B1 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HR960497A HRP960497B1 (en) 1996-10-28 1996-10-28 9-n-ethenyl derivatives of 9(s)-erythromycylamine

Publications (2)

Publication Number Publication Date
BG101996A BG101996A (en) 1998-11-30
BG63164B1 true BG63164B1 (bg) 2001-05-31

Family

ID=10946479

Family Applications (1)

Application Number Title Priority Date Filing Date
BG101996A BG63164B1 (bg) 1996-10-28 1997-10-27 9-n-етенил производни на 9(s)-еритромициламин

Country Status (18)

Country Link
US (1) US5854219A (xx)
EP (1) EP0838470B1 (xx)
JP (1) JPH10182689A (xx)
CN (1) CN1059212C (xx)
AT (1) ATE229028T1 (xx)
BG (1) BG63164B1 (xx)
CA (1) CA2217417C (xx)
CZ (1) CZ293429B6 (xx)
DE (1) DE69717583T2 (xx)
ES (1) ES2188847T3 (xx)
HR (1) HRP960497B1 (xx)
HU (1) HUP9701744A1 (xx)
PL (1) PL185878B1 (xx)
PT (1) PT838470E (xx)
RU (1) RU2170739C2 (xx)
SI (1) SI9700267B (xx)
SK (1) SK283535B6 (xx)
UA (1) UA54390C2 (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
OA11670A (en) * 1998-11-03 2005-01-12 Pfizer Prod Inc Novel macrolide antibiotics.
KR100428703B1 (ko) * 2000-02-02 2004-04-30 한국과학기술연구원 헬리코박터 파이로리의 성장 억제 효과를 지닌 신규 마크로라이드 화합물
US20020132782A1 (en) * 2001-01-18 2002-09-19 Zhenkun Ma 9-amino erythromycin derivatives with antibacterial activity
US7582611B2 (en) * 2005-05-24 2009-09-01 Pfizer Inc. Motilide compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE759251A (fr) * 1969-11-21 1971-05-21 Lilly Co Eli Derives n-arylidene de l'erythromycylamine
GB1345524A (en) * 1970-09-30 1974-01-30 Lilly Industries Ltd N-heteroarylidene erythomycylamines
DE2515076A1 (de) * 1975-04-07 1976-10-28 Thomae Gmbh Dr K Neue erythromycinderivate, deren salze und verfahren zu ihrer herstellung
DE2515026C2 (de) * 1975-04-07 1982-09-23 Jordan, Alfred, 1000 Berlin Kontaktanordnung zum Einfügen einer Schmelzsicherung in eine Leitungsverbindung
JPS61132941A (ja) * 1984-12-03 1986-06-20 Ricoh Co Ltd 複写装置
IL81395A0 (en) * 1986-02-03 1987-08-31 Lilly Co Eli Novel derivatives of erythromycylamine

Also Published As

Publication number Publication date
DE69717583D1 (de) 2003-01-16
CZ338997A3 (cs) 1998-06-17
SI9700267A (sl) 1998-04-30
SK144997A3 (en) 1998-08-05
CA2217417C (en) 2004-07-06
HU9701744D0 (en) 1997-12-29
HUP9701744A1 (hu) 1998-05-28
EP0838470A1 (en) 1998-04-29
HRP960497B1 (en) 2003-08-31
HRP960497A2 (en) 1999-02-28
PT838470E (pt) 2003-03-31
ES2188847T3 (es) 2003-07-01
EP0838470B1 (en) 2002-12-04
CN1182090A (zh) 1998-05-20
DE69717583T2 (de) 2003-09-25
ATE229028T1 (de) 2002-12-15
SI9700267B (sl) 2002-02-28
US5854219A (en) 1998-12-29
CZ293429B6 (cs) 2004-04-14
RU2170739C2 (ru) 2001-07-20
PL322862A1 (en) 1998-05-11
SK283535B6 (sk) 2003-09-11
JPH10182689A (ja) 1998-07-07
CN1059212C (zh) 2000-12-06
CA2217417A1 (en) 1998-04-28
BG101996A (en) 1998-11-30
UA54390C2 (uk) 2003-03-17
PL185878B1 (pl) 2003-08-29

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