BG108285A - Ароматни сулфон хидроксамати и тяхното използване като протеазни инхибитори - Google Patents

Ароматни сулфон хидроксамати и тяхното използване като протеазни инхибитори Download PDF

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Publication number
BG108285A
BG108285A BG108285A BG10828503A BG108285A BG 108285 A BG108285 A BG 108285A BG 108285 A BG108285 A BG 108285A BG 10828503 A BG10828503 A BG 10828503A BG 108285 A BG108285 A BG 108285A
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BG
Bulgaria
Prior art keywords
alkyl
carbocyclyl
group
substituted
heterocyclyl
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BG108285A
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Bulgarian (bg)
English (en)
Inventor
Thomas E. Barta
Daniel P. Becker
Louis J. Bedell
Terri L. Boehm
Jeffery N. Carroll
Gary A. Decrescenzo
Yvette M. Fobian
John N. Freskos
Susan L. Hockerman
Darren J. Kassab
Steve A. Kolodziej
Joseph J. Mcdonald
Deborah A. Mischke
Monica B. Norton
Joseph G. Rico
John J. Talley
Clara I. Villamil
Lijuan J. Wang
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Pharmacia Corporation
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Application filed by Pharmacia Corporation filed Critical Pharmacia Corporation
Publication of BG108285A publication Critical patent/BG108285A/bg

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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US20050101641A1 (en) 2005-05-12
IS7003A (is) 2003-10-29
US20040010019A1 (en) 2004-01-15
EP1385836A2 (fr) 2004-02-04
IL158454A0 (en) 2004-05-12
OA12602A (en) 2006-06-09
CA2446586A1 (fr) 2002-11-21
CN1764655A (zh) 2006-04-26
YU85403A (sh) 2006-03-03
KR20040018368A (ko) 2004-03-03
US6689794B2 (en) 2004-02-10
WO2002092588A2 (fr) 2002-11-21
ZA200308525B (en) 2005-02-17
JP2004530691A (ja) 2004-10-07
MXPA03010326A (es) 2004-07-30
HRP20030901A2 (en) 2005-10-31
EA200301116A1 (ru) 2004-06-24
ECSP034839A (es) 2003-12-24
CR7146A (es) 2008-02-11
HUP0304069A2 (hu) 2004-04-28
BR0209525A (pt) 2004-03-09
PL367487A1 (en) 2005-02-21
CO5540386A2 (es) 2005-07-29
NO20034995L (no) 2003-12-16
CZ20032913A3 (cs) 2004-05-12
NO20034995D0 (no) 2003-11-10
AR040928A1 (es) 2005-04-27
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US6890928B2 (en) 2005-05-10
AP2003002908A0 (en) 2003-12-31

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