IS7003A - Arómatisk súlfonhýdroxýamöt og notkun þeirra til tálmunar próteasa - Google Patents

Arómatisk súlfonhýdroxýamöt og notkun þeirra til tálmunar próteasa

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Publication number
IS7003A
IS7003A IS7003A IS7003A IS7003A IS 7003 A IS7003 A IS 7003A IS 7003 A IS7003 A IS 7003A IS 7003 A IS7003 A IS 7003A IS 7003 A IS7003 A IS 7003A
Authority
IS
Iceland
Prior art keywords
hydroxyamides
protease inhibition
aromatic sulfone
sulfone
aromatic
Prior art date
Application number
IS7003A
Other languages
English (en)
Inventor
E. Barta Thomas
P. Becker Daniel
J. Bedell Louis
L. Boehm Terri
N. Carro Jeffery
A. Decrescenzo Gary
M. Fobian Yvette
N. Freskos John
L. Hockerman Susan
J. Kassab Darren
A. Kolodziej Steve
J. Mcdonald Joseph
A. Mischke Deborah
B. Norton Monica
G. Rico Joseph
J. Talley John
I. Villamil Clara
Jane Wang Lijuan
Original Assignee
Pharmacia Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corporation filed Critical Pharmacia Corporation
Publication of IS7003A publication Critical patent/IS7003A/is

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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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IS7003A 2001-05-11 2003-10-29 Arómatisk súlfonhýdroxýamöt og notkun þeirra til tálmunar próteasa IS7003A (is)

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US20040110805A1 (en) 2004-06-10
IL158454A0 (en) 2004-05-12
HRP20030901A2 (en) 2005-10-31
BR0209525A (pt) 2004-03-09
ECSP034839A (es) 2003-12-24
WO2002092588A3 (en) 2003-02-27
US6890928B2 (en) 2005-05-10
US20040010019A1 (en) 2004-01-15
NO20034995D0 (no) 2003-11-10
EA200301116A1 (ru) 2004-06-24
CR7146A (es) 2008-02-11
US20050101641A1 (en) 2005-05-12
CZ20032913A3 (cs) 2004-05-12
NO20034995L (no) 2003-12-16
CA2446586A1 (en) 2002-11-21
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AP2003002908A0 (en) 2003-12-31
MXPA03010326A (es) 2004-07-30
AR040928A1 (es) 2005-04-27
PL367487A1 (en) 2005-02-21
CO5540386A2 (es) 2005-07-29
WO2002092588A2 (en) 2002-11-21
CN1764655A (zh) 2006-04-26
JP2004530691A (ja) 2004-10-07
YU85403A (sh) 2006-03-03
HUP0304069A2 (hu) 2004-04-28
KR20040018368A (ko) 2004-03-03
BG108285A (bg) 2004-09-30
US6689794B2 (en) 2004-02-10
EP1385836A2 (en) 2004-02-04

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