HUP0304069A2 - Aromás szulfon-hidroxamátok és proteázgátlókként való alkalmazásuk - Google Patents

Aromás szulfon-hidroxamátok és proteázgátlókként való alkalmazásuk

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Publication number
HUP0304069A2
HUP0304069A2 HU0304069A HUP0304069A HUP0304069A2 HU P0304069 A2 HUP0304069 A2 HU P0304069A2 HU 0304069 A HU0304069 A HU 0304069A HU P0304069 A HUP0304069 A HU P0304069A HU P0304069 A2 HUP0304069 A2 HU P0304069A2
Authority
HU
Hungary
Prior art keywords
protease inhibitors
aromatic sulfone
sulfone hydroxamates
hydroxamates
aromatic
Prior art date
Application number
HU0304069A
Other languages
English (en)
Inventor
Thomas E. Barta
Daniel P. Becker
Louis J. Bedell
Terri L. Boehm
Jeffery N. Carroll
Gary A. Decrescenzo
Yvette M. Fobian
John N. Freskos
Susan L. Hockerman
Darren J. Kassab
Steve A. Kolodziej
Joseph J. Mcdonald
Deborah A. Mischke
Monica B. Norton
Joseph G. Rico
John J. Talley
Clara I. Villamil
Tijuan Jane Wang
Original Assignee
Pharmacia Corp.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp. filed Critical Pharmacia Corp.
Publication of HUP0304069A2 publication Critical patent/HUP0304069A2/hu

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
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US20040110805A1 (en) 2004-06-10
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OA12602A (en) 2006-06-09
HRP20030901A2 (en) 2005-10-31
MXPA03010326A (es) 2004-07-30
ZA200308525B (en) 2005-02-17
CR7146A (es) 2008-02-11
IL158454A0 (en) 2004-05-12
ECSP034839A (es) 2003-12-24
JP2004530691A (ja) 2004-10-07
PL367487A1 (en) 2005-02-21
KR20040018368A (ko) 2004-03-03
WO2002092588A3 (en) 2003-02-27
US6689794B2 (en) 2004-02-10
BR0209525A (pt) 2004-03-09
YU85403A (sh) 2006-03-03
BG108285A (bg) 2004-09-30
AP2003002908A0 (en) 2003-12-31
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NO20034995L (no) 2003-12-16
EP1385836A2 (en) 2004-02-04
IS7003A (is) 2003-10-29
US6890928B2 (en) 2005-05-10
CN1764655A (zh) 2006-04-26
US20040010019A1 (en) 2004-01-15
WO2002092588A2 (en) 2002-11-21
CZ20032913A3 (cs) 2004-05-12
CO5540386A2 (es) 2005-07-29
CA2446586A1 (en) 2002-11-21
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