BE869833A - 2,3-polymethylene-4-oxo-4h-pyrido(1,2-a) pyrimidines utiles comme medicaments et procede pour leur preparation - Google Patents

2,3-polymethylene-4-oxo-4h-pyrido(1,2-a) pyrimidines utiles comme medicaments et procede pour leur preparation

Info

Publication number
BE869833A
BE869833A BE189955A BE189955A BE869833A BE 869833 A BE869833 A BE 869833A BE 189955 A BE189955 A BE 189955A BE 189955 A BE189955 A BE 189955A BE 869833 A BE869833 A BE 869833A
Authority
BE
Belgium
Prior art keywords
polymethylene
pyrido
oxo
preparation
medicinal products
Prior art date
Application number
BE189955A
Other languages
English (en)
French (fr)
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of BE869833A publication Critical patent/BE869833A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BE189955A 1977-08-19 1978-08-18 2,3-polymethylene-4-oxo-4h-pyrido(1,2-a) pyrimidines utiles comme medicaments et procede pour leur preparation BE869833A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU77CI1766A HU182009B (en) 1977-08-19 1977-08-19 Process for producing substituted pirido-square bracket-1,2-a-square bracket closed-pyrimidines, pyrrolo-square bracket-1,2-a-square bracket closed-pyrimidines

Publications (1)

Publication Number Publication Date
BE869833A true BE869833A (fr) 1978-12-18

Family

ID=10994668

Family Applications (1)

Application Number Title Priority Date Filing Date
BE189955A BE869833A (fr) 1977-08-19 1978-08-18 2,3-polymethylene-4-oxo-4h-pyrido(1,2-a) pyrimidines utiles comme medicaments et procede pour leur preparation

Country Status (21)

Country Link
US (1) US4220771A (sv)
JP (1) JPS5459299A (sv)
AT (1) AT371818B (sv)
BE (1) BE869833A (sv)
CA (1) CA1117525A (sv)
CH (1) CH638207A5 (sv)
CS (1) CS240351B1 (sv)
DD (1) DD138902A5 (sv)
DE (1) DE2836449A1 (sv)
DK (1) DK157021C (sv)
ES (1) ES473182A1 (sv)
FI (1) FI67547C (sv)
FR (1) FR2416893A1 (sv)
GB (1) GB2003870B (sv)
GR (1) GR65275B (sv)
HU (1) HU182009B (sv)
NL (1) NL7808571A (sv)
PL (1) PL116688B1 (sv)
SE (1) SE436279B (sv)
SU (1) SU749365A3 (sv)
YU (1) YU196578A (sv)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4348396A (en) * 1978-01-23 1982-09-07 Hoffmann-La Roche Inc. Substituted 11-oxo-11H-pyrido[2,1-b]quinazolines and method of inhibiting allergic reactions with them
US4395549A (en) * 1981-10-02 1983-07-26 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. 6-Hydrazono-pyrido[2,1-b] quinazoline-11 ones
ES521739A0 (es) * 1982-04-29 1984-07-01 Erba Farmitalia Procedimiento para preparar derivados cicloalifaticos condensados de pirido(1,2-a)pirimidinas sustituidas.
HU191192B (en) * 1982-11-16 1987-01-28 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt,Hu Process for producing new azepino /1,2-a/ pyrimidine derivatives of bronchodilating activity and acid additional salts thereof and pharmaceiutical compositions containing them
CA2113115A1 (en) * 1991-07-29 1993-02-18 Vlad E. Gregor Quinazoline derivatives as acetylcholinesterase inhibitors
US5892917A (en) * 1995-09-27 1999-04-06 Microsoft Corporation System for log record and log expansion with inserted log records representing object request for specified object corresponding to cached object copies
WO2011075699A2 (en) * 2009-12-18 2011-06-23 Sunovion Pharmaceuticals Inc. Compounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1088968B (de) 1958-07-03 1960-09-15 Bayer Ag Verfahren zur Herstellung von mehrkernigen, heterocyclischen, einen 4-Oxo-3, 4-dihydro-pyrimidinring enthaltenden Verbindungen
US2992221A (en) * 1958-07-03 1961-07-11 Petersen Siegfried Polymethylene-oxoquinazolines and their production
US3271396A (en) * 1964-08-17 1966-09-06 Squibb & Sons Inc Pyrido-quinazoline derivatives
DE1803785A1 (de) * 1968-10-18 1970-06-04 Hoechst Ag Verfahren zur Herstellung von 1,2-disubstituierten 6-Oxo-1.4.5.6-tetrahydropyrimidinen
US3790573A (en) * 1971-11-11 1974-02-05 Smithkline Corp Imidazo and pyrimido(2,1-b)quinazolines
US3965100A (en) * 1975-02-26 1976-06-22 E. R. Squibb & Sons, Inc. 2,3-Dihydrocyclopenta[d]pyrido[1,2-a]pyrimidin-10(1H)-one and its derivatives
US4033961A (en) * 1975-10-07 1977-07-05 Warner-Lambert Company Pyrido[2-1-b]quinazolin-ones and their methods of preparation
DE2557425A1 (de) * 1975-12-19 1977-06-30 Boehringer Sohn Ingelheim Chinazolonderivate
JPH0297996A (ja) * 1988-10-05 1990-04-10 Toshiba Corp 画像データ変換回路

Also Published As

Publication number Publication date
FR2416893A1 (fr) 1979-09-07
GB2003870A (en) 1979-03-21
CH638207A5 (de) 1983-09-15
PL209131A1 (pl) 1979-06-04
ATA597178A (de) 1982-12-15
DK157021C (da) 1990-04-02
CA1117525A (en) 1982-02-02
ES473182A1 (es) 1979-04-01
AT371818B (de) 1983-08-10
HU182009B (en) 1983-12-28
YU196578A (en) 1983-10-31
CS240351B1 (en) 1986-02-13
DE2836449A1 (de) 1979-03-22
GR65275B (en) 1980-07-31
SU749365A3 (ru) 1980-07-15
GB2003870B (en) 1982-07-21
US4220771A (en) 1980-09-02
FI67547B (fi) 1984-12-31
FR2416893B1 (sv) 1983-07-22
DK367378A (da) 1979-02-20
FI782517A (fi) 1979-02-20
JPS5459299A (en) 1979-05-12
NL7808571A (nl) 1979-02-21
DD138902A5 (de) 1979-11-28
SE7808771L (sv) 1979-02-20
DE2836449C2 (sv) 1990-09-06
FI67547C (fi) 1985-04-10
SE436279B (sv) 1984-11-26
DK157021B (da) 1989-10-30
CS541878A1 (en) 1985-05-15
PL116688B1 (en) 1981-06-30

Similar Documents

Publication Publication Date Title
BE841390A (fr) Diamino-2,4 bromo-5 chloro-6 pyrimidines utilisables comme medicaments et procede pour leur preparation
BE895708A (fr) Urees et thio-urees substituees, leur procede de preparation et leur application therapeutique comme medicaments anti-atherosclereux
BE877889A (fr) Nouveaux derives de la pyrimidone, procedes pour leur preparation et leur utilisation comme medicaments
BE891092A (fr) Derives de benzofuranne-2 substitues utiles comme medicaments et procede de leur preparation
BE880153A (fr) Derives de 7-oxo-4-thia-1-aza-bicyclo- (3,2,0) -heptane, procede pour les preparer et leur application comme medicaments
BE865015A (fr) Pseudotrisaccharides, leur procede de preparation et medicament les contenant
MY8600271A (en) Novel mercaptoimidazole derivatives process for their preparation, mercapto-imidazole derivatives for the treatment of inflammatory disorders, and pharmaceutical products containing them
BE860614A (fr) Hydroxylamines alkylees, leur procede de preparation et leur emploi comme medicaments
FR2569195B1 (fr) Derives du 7-carboxymethoxyphenylacetamido-3-cepheme utiles comme medicaments antibacteriens et procedes pour leur preparation
LU79356A1 (fr) Preparation d'interphenylene 8-aza-9-dioxathia-11,12-secoprostaglandines utiles comme medicaments
FR2521134B1 (fr) Urees et thio-urees substituees, leur procede de preparation et leur application therapeutique comme medicaments anti-atherosclereux
BE869833A (fr) 2,3-polymethylene-4-oxo-4h-pyrido(1,2-a) pyrimidines utiles comme medicaments et procede pour leur preparation
IL55862A0 (en) Novel 6-oxygenated-3,20-dioxo-pregnane derivatives, process for the preparation thereof, and pharmaceutical compositionss containing them
PT65456B (fr) Procede de preparation de dihyro-1,4 pyridines utilisablesnotamment comme medicaments antihypertenseurs et antiangoreux
BE883576A (fr) Nouveaux derives d'hydroxyamino-eburnane leur procede de preparation, intermediaires utiles et utilisation comme medicament et comme intermediaire
BE875106A (fr) Medicaments anticomplementaires en partie antinephretiques, de type soya-sapogenol b et leur procede de preparation
FR2526022B1 (fr) Derives de l'ergoline, procede pour les preparer et leur emploi comme medicaments
BE859120A (fr) Procede pour la preparation de steroides polyhalogenes utiles comme medicaments
BE861137A (fr) Ortho-aminoacetophenones utiles comme medicaments et procede pour leur preparation
BE870687A (fr) Nouvelles monoalkylanilines substituees en position 4 utiles comme medicaments et procedes pour leur preparation
BE862302A (fr) Nouvelles oximes 0-alkylees, leur procede de preparation et leur emploi comme medicaments
BE866588A (fr) Derives de 2-benzyl-perhydroazepines, procede pour leur preparation et application comme medicaments
IL53685A (en) N2-arylsulfonyl-l-argininamides and the pharmaceutical salts thereof,process for their preparation and pharmaceutical compositions containing them
FR2520742B1 (fr) 1,3,4-thiadiazolo(3,2-a)pyrimidines substituees utiles comme medicaments et procede de leur preparation
BE863596A (fr) 2,9-dioxatricyclo (4,3,1,03,7) decanes,procede pour leur preparation et utilisation comme medicaments

Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT

Effective date: 19910831