AU2017292818B2 - Solid forms of an sGC stimulator - Google Patents

Solid forms of an sGC stimulator Download PDF

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Publication number
AU2017292818B2
AU2017292818B2 AU2017292818A AU2017292818A AU2017292818B2 AU 2017292818 B2 AU2017292818 B2 AU 2017292818B2 AU 2017292818 A AU2017292818 A AU 2017292818A AU 2017292818 A AU2017292818 A AU 2017292818A AU 2017292818 B2 AU2017292818 B2 AU 2017292818B2
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disease
pulmonary
compound
diseases
hypertension
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AU2017292818A1 (en
Inventor
Ahmad Hashash
Robert C. Livingston
Kwame Wiredu NTI-ADDAE
Vasu SETHURAMAN
Song Xue
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Cyclerion Therapeutics Inc
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Cyclerion Therapeutics Inc
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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