AU2014233240B2 - Convergent processes for preparing macrolide antibacterial agents - Google Patents

Convergent processes for preparing macrolide antibacterial agents Download PDF

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Publication number
AU2014233240B2
AU2014233240B2 AU2014233240A AU2014233240A AU2014233240B2 AU 2014233240 B2 AU2014233240 B2 AU 2014233240B2 AU 2014233240 A AU2014233240 A AU 2014233240A AU 2014233240 A AU2014233240 A AU 2014233240A AU 2014233240 B2 AU2014233240 B2 AU 2014233240B2
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compound
formula
salt
prepare
contacting
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AU2014233240A1 (en
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David E. Pereira
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Cempra Pharmaceuticals Inc
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Cempra Pharmaceuticals Inc
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU2014233240A 2013-03-15 2014-03-15 Convergent processes for preparing macrolide antibacterial agents Ceased AU2014233240B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361786914P 2013-03-15 2013-03-15
US61/786,914 2013-03-15
PCT/US2014/029932 WO2014145210A1 (en) 2013-03-15 2014-03-15 Convergent processes for preparing macrolide antibacterial agents

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AU2014233240A1 AU2014233240A1 (en) 2015-10-01
AU2014233240B2 true AU2014233240B2 (en) 2018-08-09

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AU2014233240A Ceased AU2014233240B2 (en) 2013-03-15 2014-03-15 Convergent processes for preparing macrolide antibacterial agents

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US (3) US9751908B2 (enExample)
EP (1) EP2968384A4 (enExample)
JP (1) JP6675973B2 (enExample)
KR (1) KR20160020403A (enExample)
CN (1) CN105188712A (enExample)
AU (1) AU2014233240B2 (enExample)
BR (1) BR112015023670A2 (enExample)
CA (1) CA2907085A1 (enExample)
HK (2) HK1218864A1 (enExample)
MX (1) MX356772B (enExample)
RU (1) RU2015138797A (enExample)
WO (1) WO2014145210A1 (enExample)
ZA (1) ZA201507551B (enExample)

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EP2968384A1 (en) 2016-01-20
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