AU2012250010A1 - Combination of a phosphatidylinositol-3-kinase (PI3K) inhibitor and a mTOR inhibitor - Google Patents

Combination of a phosphatidylinositol-3-kinase (PI3K) inhibitor and a mTOR inhibitor Download PDF

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Publication number
AU2012250010A1
AU2012250010A1 AU2012250010A AU2012250010A AU2012250010A1 AU 2012250010 A1 AU2012250010 A1 AU 2012250010A1 AU 2012250010 A AU2012250010 A AU 2012250010A AU 2012250010 A AU2012250010 A AU 2012250010A AU 2012250010 A1 AU2012250010 A1 AU 2012250010A1
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AU
Australia
Prior art keywords
compound
combination
alkyl
substituted
deuterium
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Abandoned
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AU2012250010A
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English (en)
Inventor
Christine Fritsch
Carlos Garcia-Echeverria
Xizhong Huang
Sauveur-Michel Maira
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Novartis AG
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Novartis AG
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46018130&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2012250010(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis AG filed Critical Novartis AG
Publication of AU2012250010A1 publication Critical patent/AU2012250010A1/en
Priority to AU2016202372A priority Critical patent/AU2016202372B2/en
Abandoned legal-status Critical Current

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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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AU2012250010A 2011-04-25 2012-04-23 Combination of a phosphatidylinositol-3-kinase (PI3K) inhibitor and a mTOR inhibitor Abandoned AU2012250010A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2016202372A AU2016202372B2 (en) 2011-04-25 2016-04-14 Combination of a phosphatidylinositol-3-kinase (PI3K) inhibitor and a mTOR inhibitor

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161478572P 2011-04-25 2011-04-25
US61/478,572 2011-04-25
PCT/US2012/034647 WO2012148846A1 (en) 2011-04-25 2012-04-23 Combination of a phosphatidylinositol-3-kinase (pi3k) inhibitor and a mtor inhibitor

Related Child Applications (1)

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AU2016202372A Division AU2016202372B2 (en) 2011-04-25 2016-04-14 Combination of a phosphatidylinositol-3-kinase (PI3K) inhibitor and a mTOR inhibitor

Publications (1)

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AU2012250010A1 true AU2012250010A1 (en) 2013-10-10

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Family Applications (2)

Application Number Title Priority Date Filing Date
AU2012250010A Abandoned AU2012250010A1 (en) 2011-04-25 2012-04-23 Combination of a phosphatidylinositol-3-kinase (PI3K) inhibitor and a mTOR inhibitor
AU2016202372A Ceased AU2016202372B2 (en) 2011-04-25 2016-04-14 Combination of a phosphatidylinositol-3-kinase (PI3K) inhibitor and a mTOR inhibitor

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AU2016202372A Ceased AU2016202372B2 (en) 2011-04-25 2016-04-14 Combination of a phosphatidylinositol-3-kinase (PI3K) inhibitor and a mTOR inhibitor

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US (3) US20140066474A1 (cg-RX-API-DMAC7.html)
EP (1) EP2701703A1 (cg-RX-API-DMAC7.html)
JP (2) JP6086902B2 (cg-RX-API-DMAC7.html)
KR (1) KR101925656B1 (cg-RX-API-DMAC7.html)
CN (1) CN103491955B (cg-RX-API-DMAC7.html)
AR (1) AR086481A1 (cg-RX-API-DMAC7.html)
AU (2) AU2012250010A1 (cg-RX-API-DMAC7.html)
BR (1) BR112013027486A2 (cg-RX-API-DMAC7.html)
CA (1) CA2833962A1 (cg-RX-API-DMAC7.html)
CL (1) CL2013003078A1 (cg-RX-API-DMAC7.html)
CO (1) CO6801759A2 (cg-RX-API-DMAC7.html)
EA (1) EA025948B1 (cg-RX-API-DMAC7.html)
EC (1) ECSP13012994A (cg-RX-API-DMAC7.html)
GT (1) GT201300263A (cg-RX-API-DMAC7.html)
IL (1) IL229008A (cg-RX-API-DMAC7.html)
MA (1) MA35038B1 (cg-RX-API-DMAC7.html)
MX (1) MX2013012385A (cg-RX-API-DMAC7.html)
NZ (1) NZ615593A (cg-RX-API-DMAC7.html)
PE (1) PE20140601A1 (cg-RX-API-DMAC7.html)
PH (1) PH12013502077A1 (cg-RX-API-DMAC7.html)
SG (1) SG193919A1 (cg-RX-API-DMAC7.html)
TN (1) TN2013000392A1 (cg-RX-API-DMAC7.html)
TW (1) TWI602567B (cg-RX-API-DMAC7.html)
UA (1) UA110961C2 (cg-RX-API-DMAC7.html)
WO (1) WO2012148846A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA201306973B (cg-RX-API-DMAC7.html)

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EP3068435A1 (en) * 2013-11-13 2016-09-21 Novartis AG Mtor inhibitors for enhancing the immune response
RU2016135413A (ru) * 2014-02-11 2018-03-14 Новартис Аг Фармацевтические комбинации, включающие ингибитор pi3k, для лечения рака
WO2015148626A1 (en) * 2014-03-26 2015-10-01 Millennium Pharmaceuticals, Inc. Treatment of fibrotic disorders
BR112017004694A2 (pt) * 2014-10-03 2017-12-05 Novartis Ag composições farmacêuticas compreendendo alpelisibe
US20160339030A1 (en) * 2015-05-19 2016-11-24 University Of Maryland, Baltimore Treatment agents for inhibiting hiv and cancer in hiv infected patients
JP6691337B2 (ja) * 2016-02-29 2020-04-28 学校法人北里研究所 膀胱癌患者の予後を予測するための方法

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