GT201300263A - Combinación de un inhibidor de cinasa de fosfatidilinositol-3 (pi3k) y un inhibidor de mtor - Google Patents

Combinación de un inhibidor de cinasa de fosfatidilinositol-3 (pi3k) y un inhibidor de mtor

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Publication number
GT201300263A
GT201300263A GT201300263A GT201300263A GT201300263A GT 201300263 A GT201300263 A GT 201300263A GT 201300263 A GT201300263 A GT 201300263A GT 201300263 A GT201300263 A GT 201300263A GT 201300263 A GT201300263 A GT 201300263A
Authority
GT
Guatemala
Prior art keywords
inhibitor
pi3k
combination
phosfatidylinositol
motor
Prior art date
Application number
GT201300263A
Other languages
English (en)
Inventor
Fritsch Christine
Garcia-Echeverria Carlos
Huang Xizhong
Maira Sauveur-Michel
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Publication date
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Application filed filed Critical
Publication of GT201300263A publication Critical patent/GT201300263A/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
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    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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Abstract

LA PRESENTE INVENCIÓN SE REFIERE A UNA COMBINACIÓN FARMACÉUTICA QUE COMPRENDE UN COMPUESTO INHIBIDOR DE CINASA DE FOSFATIDIL-INOSITOL-3 (PI3K), EL CUAL ES UN DERIVADO DE 2-CARBOXAMIDA-CICLOAMINO-UREA, O UNA SAL FARMACÉUTICAMENTE ACEPTABLE DEL MISMO.
GT201300263A 2011-04-25 2013-10-25 Combinación de un inhibidor de cinasa de fosfatidilinositol-3 (pi3k) y un inhibidor de mtor GT201300263A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161478572P 2011-04-25 2011-04-25

Publications (1)

Publication Number Publication Date
GT201300263A true GT201300263A (es) 2015-11-24

Family

ID=46018130

Family Applications (1)

Application Number Title Priority Date Filing Date
GT201300263A GT201300263A (es) 2011-04-25 2013-10-25 Combinación de un inhibidor de cinasa de fosfatidilinositol-3 (pi3k) y un inhibidor de mtor

Country Status (25)

Country Link
US (3) US20140066474A1 (es)
EP (1) EP2701703A1 (es)
JP (2) JP6086902B2 (es)
KR (1) KR101925656B1 (es)
CN (1) CN103491955B (es)
AR (1) AR086481A1 (es)
AU (2) AU2012250010A1 (es)
BR (1) BR112013027486A2 (es)
CA (1) CA2833962A1 (es)
CL (1) CL2013003078A1 (es)
CO (1) CO6801759A2 (es)
EA (1) EA025948B1 (es)
EC (1) ECSP13012994A (es)
GT (1) GT201300263A (es)
IL (1) IL229008A (es)
MA (1) MA35038B1 (es)
MX (1) MX2013012385A (es)
NZ (1) NZ615593A (es)
PE (1) PE20140601A1 (es)
SG (1) SG193919A1 (es)
TN (1) TN2013000392A1 (es)
TW (1) TWI602567B (es)
UA (1) UA110961C2 (es)
WO (1) WO2012148846A1 (es)
ZA (1) ZA201306973B (es)

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WO2015148626A1 (en) * 2014-03-26 2015-10-01 Millennium Pharmaceuticals, Inc. Treatment of fibrotic disorders
EP3200772B1 (en) * 2014-10-03 2022-08-03 Novartis AG Pharmaceutical compositions comprising alpelisib
US20160339030A1 (en) * 2015-05-19 2016-11-24 University Of Maryland, Baltimore Treatment agents for inhibiting hiv and cancer in hiv infected patients
GB202010627D0 (en) * 2020-07-10 2020-08-26 Qbd (Qs-Ip) Ltd Blocking method

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MX2013012385A (es) 2013-11-04
JP2017061527A (ja) 2017-03-30
KR20140012147A (ko) 2014-01-29
TW201244716A (en) 2012-11-16
CA2833962A1 (en) 2012-11-01
US20140066474A1 (en) 2014-03-06
ECSP13012994A (es) 2013-12-31
KR101925656B1 (ko) 2018-12-05
SG193919A1 (en) 2013-11-29
AU2012250010A1 (en) 2013-10-10
PE20140601A1 (es) 2014-05-24
JP6086902B2 (ja) 2017-03-01
BR112013027486A2 (pt) 2017-02-14
NZ615593A (en) 2015-05-29
TN2013000392A1 (en) 2015-01-20
AR086481A1 (es) 2013-12-18
MA35038B1 (fr) 2014-04-03
WO2012148846A1 (en) 2012-11-01
ZA201306973B (en) 2014-06-25
AU2016202372B2 (en) 2017-07-20
TWI602567B (zh) 2017-10-21
CL2013003078A1 (es) 2014-05-30
EA025948B1 (ru) 2017-02-28
CN103491955A (zh) 2014-01-01
EP2701703A1 (en) 2014-03-05
UA110961C2 (uk) 2016-03-10
JP2014513097A (ja) 2014-05-29
CO6801759A2 (es) 2013-11-29
US20180085362A1 (en) 2018-03-29
AU2016202372A1 (en) 2016-05-05
EA201391565A1 (ru) 2014-02-28
US20170095463A1 (en) 2017-04-06
IL229008A (en) 2017-11-30
IL229008A0 (en) 2013-12-31
CN103491955B (zh) 2015-12-23

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