AU2004268941A1 - Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases - Google Patents

Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases Download PDF

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Publication number
AU2004268941A1
AU2004268941A1 AU2004268941A AU2004268941A AU2004268941A1 AU 2004268941 A1 AU2004268941 A1 AU 2004268941A1 AU 2004268941 A AU2004268941 A AU 2004268941A AU 2004268941 A AU2004268941 A AU 2004268941A AU 2004268941 A1 AU2004268941 A1 AU 2004268941A1
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Prior art keywords
substituted
compound
group
formula
heterocycle
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Abandoned
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AU2004268941A
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Inventor
Timothy James Davis
Sunil K.C. Kumar
Jagadish Sircar
Wenbin Ying
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Avanir Pharmaceuticals Inc
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Avanir Pharmaceuticals Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34272569&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2004268941(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Avanir Pharmaceuticals Inc filed Critical Avanir Pharmaceuticals Inc
Publication of AU2004268941A1 publication Critical patent/AU2004268941A1/en
Abandoned legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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    • A61P37/02—Immunomodulators
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P7/06—Antianaemics
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Endocrinology (AREA)
  • Transplantation (AREA)
  • Psychology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Virology (AREA)
  • Dermatology (AREA)
AU2004268941A 2003-08-22 2004-08-09 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases Abandoned AU2004268941A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US49744303P 2003-08-22 2003-08-22
US60/497,443 2003-08-22
PCT/US2004/025683 WO2005021546A1 (en) 2003-08-22 2004-08-09 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases

Publications (1)

Publication Number Publication Date
AU2004268941A1 true AU2004268941A1 (en) 2005-03-10

Family

ID=34272569

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AU2004268941A Abandoned AU2004268941A1 (en) 2003-08-22 2004-08-09 Substituted naphthyridine derivatives as inhibitors of macrophage migration inhibitory factor and their use in the treatment of human diseases

Country Status (13)

Country Link
US (2) US20050124604A1 (https=)
EP (1) EP1656376A1 (https=)
JP (1) JP2007503388A (https=)
CN (1) CN1839133A (https=)
AR (1) AR045471A1 (https=)
AU (1) AU2004268941A1 (https=)
BR (1) BRPI0413695A (https=)
CA (1) CA2531506A1 (https=)
MX (1) MXJL06000006A (https=)
PE (1) PE20051112A1 (https=)
TW (1) TW200524928A (https=)
UY (1) UY28483A1 (https=)
WO (1) WO2005021546A1 (https=)

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EP1656376A1 (en) 2006-05-17
TW200524928A (en) 2005-08-01
MXJL06000006A (es) 2006-05-04
US20050124604A1 (en) 2005-06-09
JP2007503388A (ja) 2007-02-22
UY28483A1 (es) 2005-03-31
CN1839133A (zh) 2006-09-27
CA2531506A1 (en) 2005-03-10
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WO2005021546A1 (en) 2005-03-10
AR045471A1 (es) 2005-10-26

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