ATE384731T1 - Nukleinsäurebindende verbindungen mit pyrazolo 3, 4-d pyrimidinanalogen von purin-2,6-diamin und ihre verwendung - Google Patents

Nukleinsäurebindende verbindungen mit pyrazolo 3, 4-d pyrimidinanalogen von purin-2,6-diamin und ihre verwendung

Info

Publication number
ATE384731T1
ATE384731T1 AT01956576T AT01956576T ATE384731T1 AT E384731 T1 ATE384731 T1 AT E384731T1 AT 01956576 T AT01956576 T AT 01956576T AT 01956576 T AT01956576 T AT 01956576T AT E384731 T1 ATE384731 T1 AT E384731T1
Authority
AT
Austria
Prior art keywords
nucleic acid
acid binding
purine
pyrazolo
diamine
Prior art date
Application number
AT01956576T
Other languages
German (de)
English (en)
Inventor
Frank Seela
Frank Bergmann
Der Eltz Herbert Von
Dieter Heindl
Christoph Seidel
Georg Becher
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of ATE384731T1 publication Critical patent/ATE384731T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H21/00—Compounds containing two or more mononucleotide units having separate phosphate or polyphosphate groups linked by saccharide radicals of nucleoside groups, e.g. nucleic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T436/00—Chemistry: analytical and immunological testing
    • Y10T436/14—Heterocyclic carbon compound [i.e., O, S, N, Se, Te, as only ring hetero atom]
    • Y10T436/142222—Hetero-O [e.g., ascorbic acid, etc.]
    • Y10T436/143333—Saccharide [e.g., DNA, etc.]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • General Health & Medical Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT01956576T 2000-08-03 2001-07-31 Nukleinsäurebindende verbindungen mit pyrazolo 3, 4-d pyrimidinanalogen von purin-2,6-diamin und ihre verwendung ATE384731T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00116816 2000-08-03
EP01109438 2001-04-24

Publications (1)

Publication Number Publication Date
ATE384731T1 true ATE384731T1 (de) 2008-02-15

Family

ID=26071249

Family Applications (1)

Application Number Title Priority Date Filing Date
AT01956576T ATE384731T1 (de) 2000-08-03 2001-07-31 Nukleinsäurebindende verbindungen mit pyrazolo 3, 4-d pyrimidinanalogen von purin-2,6-diamin und ihre verwendung

Country Status (9)

Country Link
US (2) US7238795B2 (enExample)
EP (1) EP1307469B1 (enExample)
JP (1) JP4331476B2 (enExample)
AT (1) ATE384731T1 (enExample)
AU (1) AU2001278517A1 (enExample)
CA (1) CA2416631C (enExample)
DE (1) DE60132596T2 (enExample)
ES (1) ES2300346T3 (enExample)
WO (1) WO2002012263A1 (enExample)

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Also Published As

Publication number Publication date
JP4331476B2 (ja) 2009-09-16
EP1307469B1 (en) 2008-01-23
EP1307469A1 (en) 2003-05-07
CA2416631A1 (en) 2002-02-14
DE60132596D1 (de) 2008-03-13
US7238795B2 (en) 2007-07-03
US8057997B2 (en) 2011-11-15
AU2001278517A1 (en) 2002-02-18
US20110021365A1 (en) 2011-01-27
WO2002012263A1 (en) 2002-02-14
CA2416631C (en) 2011-11-22
JP2004505988A (ja) 2004-02-26
ES2300346T3 (es) 2008-06-16
US20030198982A1 (en) 2003-10-23
DE60132596T2 (de) 2009-02-19

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