ATE276252T1 - Aminoheterocyclylamide als pestizide und antiparasitisch wirksame wirkstoffe - Google Patents

Aminoheterocyclylamide als pestizide und antiparasitisch wirksame wirkstoffe

Info

Publication number
ATE276252T1
ATE276252T1 AT00993258T AT00993258T ATE276252T1 AT E276252 T1 ATE276252 T1 AT E276252T1 AT 00993258 T AT00993258 T AT 00993258T AT 00993258 T AT00993258 T AT 00993258T AT E276252 T1 ATE276252 T1 AT E276252T1
Authority
AT
Austria
Prior art keywords
substituents
c6alkyl
c6alkoxy
halogen
phenyl
Prior art date
Application number
AT00993258T
Other languages
English (en)
Inventor
Pierre Ducray
Jacques Bouvier
Maurizio Schwarzenbach
Original Assignee
Novartis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh
Application granted granted Critical
Publication of ATE276252T1 publication Critical patent/ATE276252T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/08—1,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/36—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
AT00993258T 1999-12-02 2000-11-30 Aminoheterocyclylamide als pestizide und antiparasitisch wirksame wirkstoffe ATE276252T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH220799 1999-12-02
PCT/EP2000/012064 WO2001040223A2 (en) 1999-12-02 2000-11-30 Aminoheterocyclylamides as pesticides and antiparasitic agents

Publications (1)

Publication Number Publication Date
ATE276252T1 true ATE276252T1 (de) 2004-10-15

Family

ID=4228396

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00993258T ATE276252T1 (de) 1999-12-02 2000-11-30 Aminoheterocyclylamide als pestizide und antiparasitisch wirksame wirkstoffe

Country Status (18)

Country Link
US (1) US6673820B2 (de)
EP (1) EP1254135B1 (de)
JP (1) JP2003515608A (de)
KR (1) KR100479137B1 (de)
CN (1) CN1196700C (de)
AT (1) ATE276252T1 (de)
AU (1) AU765618B2 (de)
BR (1) BR0016034A (de)
CA (1) CA2390113A1 (de)
DE (1) DE60013910T2 (de)
DK (1) DK1254135T3 (de)
ES (1) ES2228664T3 (de)
MX (1) MXPA02005428A (de)
NZ (1) NZ518931A (de)
PT (1) PT1254135E (de)
RU (1) RU2002117428A (de)
WO (1) WO2001040223A2 (de)
ZA (1) ZA200204337B (de)

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JP2002154904A (ja) * 2000-11-13 2002-05-28 Mitsubishi Chemicals Corp N−チアジアゾリルカルボン酸アミド類およびこれを有効成分とする殺虫、殺ダニ剤
US7196106B2 (en) 2002-11-05 2007-03-27 Merck & Co., Inc Cyanothiophene derivatives, compositions containing such compounds and methods of use
JP2004269515A (ja) * 2003-02-18 2004-09-30 Nippon Nohyaku Co Ltd 置換複素環アミド誘導体、その中間体及び農園芸用薬剤並びにその使用方法
US20050085531A1 (en) * 2003-10-03 2005-04-21 Hodge Carl N. Thiophene-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof
NL2000351C2 (nl) 2005-12-22 2007-09-11 Pfizer Prod Inc Estrogeen-modulatoren.
US20100200021A1 (en) * 2006-02-17 2010-08-12 Nils Adey Slide Conditioning Systems and Methods
WO2008005764A2 (en) * 2006-06-30 2008-01-10 Fmc Corporation Novel zeta-cypermethrin composition
SG10201502484SA (en) 2010-03-30 2015-05-28 Verseon Corp Multisubstituted aromatic compounds as inhibitors of thrombin
EP2560488B1 (de) 2010-04-23 2015-10-28 Cytokinetics, Inc. Bestimmte aminopyrimidine und aminotriazine, zusammensetzungen daraus und verfahren zu ihrer verwendung
AR081331A1 (es) 2010-04-23 2012-08-08 Cytokinetics Inc Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos
AR081626A1 (es) 2010-04-23 2012-10-10 Cytokinetics Inc Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos
CN102067845B (zh) * 2011-01-31 2013-07-17 湖南大学 5-苄基-4-烷基-2-芳氨基噻唑作为制备杀虫剂的应用
US8759380B2 (en) 2011-04-22 2014-06-24 Cytokinetics, Inc. Certain heterocycles, compositions thereof, and methods for their use
LT2782565T (lt) * 2011-11-25 2019-12-27 Bayer Intellectual Property Gmbh Aril- ir hetarilkarboksamidų panaudojimas kaip endoparaziticidų
DK2968297T3 (en) 2013-03-15 2019-01-07 Verseon Inc MULTI-SUBSTITUTED AROMATIC COMPOUNDS AS SERINE PROTEASE INHIBITORS
WO2014149139A2 (en) 2013-03-15 2014-09-25 Verseon, Inc. Halogenopyrazoles as inhibitors of thrombin
JP2017528486A (ja) 2014-09-17 2017-09-28 ヴァーセオン コーポレイション セリンプロテアーゼ阻害剤としてのピラゾリル置換ピリドン化合物
ES2931460T3 (es) 2015-02-27 2022-12-29 Verseon Int Corporation Compuestos de pirazol sustituido como inhibidores de serina proteasa
WO2017005717A1 (en) 2015-07-06 2017-01-12 Bayer Cropscience Aktiengesellschaft Heterocyclic compounds as pesticides
JP2020502168A (ja) * 2016-12-16 2020-01-23 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺有害生物剤としてのチアジアゾール誘導体
MX2019007374A (es) * 2016-12-22 2019-09-18 Bayer Cropscience Ag Heteroarilpirrolonas sustituidas y sus sales y su uso como ingredientes activos herbicidas.
BR112019012822A2 (pt) 2016-12-22 2019-11-26 Bayer Ag 1,2,4-tiadiazolilpirrolonas e 1,2,4-tiadiazolil-hidantoínas e sais das mesmas e uso das mesmas como herbicidas
CN111601802A (zh) 2017-11-28 2020-08-28 拜耳股份有限公司 作为杀虫剂的杂环化合物
EP3846793B1 (de) 2018-09-07 2024-01-24 PIC Therapeutics, Inc. Eif4e-inhibitoren und verwendungen davon
AR121506A1 (es) 2020-03-03 2022-06-08 Pic Therapeutics Inc Inhibidores del eif4e y sus usos
WO2022194841A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
WO2022194842A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
WO2022194843A1 (en) 2021-03-19 2022-09-22 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazoles, salts thereof and their use as herbicidally active substances
CA3229299A1 (en) 2021-08-17 2023-02-23 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazolyl nicotinamides, salts or n-oxides thereof and their use as herbicidally active substances
WO2023020962A1 (en) 2021-08-17 2023-02-23 Bayer Aktiengesellschaft Substituted 1,2,4-thiadiazolyl nicotinamides, salts or n-oxides thereof and their use as herbicidally active substances
MX2024002082A (es) 2021-08-17 2024-03-05 Bayer Ag 1,2,4-tiadiazolil nicotinamidas sustituidas, sus sales o n-oxidos, y su uso como sustancias herbicidamente activas.
US12157732B2 (en) 2021-08-25 2024-12-03 PIC Therapeutics, Inc. eIF4E inhibitors and uses thereof
IL310924A (en) 2021-08-25 2024-04-01 Pic Therapeutics Inc Eif4e inhibitors and uses thereof
EP4238973A1 (de) 2022-03-04 2023-09-06 Bayer AG Substituierte 1,2,4-thiadiazolyl-nicotinamide, salze oder n-oxide davon und ihre verwendung als herbizide wirkstoffe
EP4238972A1 (de) 2022-03-04 2023-09-06 Bayer AG Substituierte 1,2,4-thiadiazolyl-picolinamide, salze oder n-oxide davon und ihre verwendung als herbizide wirkstoffe

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DE1924830A1 (de) 1968-07-06 1970-11-19 Merck Patent Gmbh Neues Verfahren zur Herstellung von 5-Acylamino-isothiazolderivaten
IN140035B (de) 1973-07-19 1976-09-04 Fmc Corp
ES2055808T3 (es) * 1988-03-21 1994-09-01 Ciba Geigy Ag Agente para la proteccion de plantas contra enfermedades.
EP0623282A1 (de) * 1993-05-05 1994-11-09 Shell Internationale Researchmaatschappij B.V. Pestizide Verfahren und Verbindungen
GB9725298D0 (en) 1997-11-28 1998-01-28 Zeneca Ltd Insecticidal thiazole derivatives
JP2000226389A (ja) 1998-11-30 2000-08-15 Mitsubishi Chemicals Corp N−チアジアゾリルピラゾールカルボキサミド誘導体およびこれを有効成分とする殺虫、殺ダニ剤

Also Published As

Publication number Publication date
WO2001040223A2 (en) 2001-06-07
US20030148890A1 (en) 2003-08-07
PT1254135E (pt) 2005-03-31
DE60013910T2 (de) 2005-09-29
DK1254135T3 (da) 2005-01-17
EP1254135A2 (de) 2002-11-06
CA2390113A1 (en) 2001-06-07
JP2003515608A (ja) 2003-05-07
WO2001040223A3 (en) 2001-12-20
ZA200204337B (en) 2003-06-03
EP1254135B1 (de) 2004-09-15
DE60013910D1 (de) 2004-10-21
US6673820B2 (en) 2004-01-06
AU765618B2 (en) 2003-09-25
NZ518931A (en) 2004-02-27
CN1196700C (zh) 2005-04-13
ES2228664T3 (es) 2005-04-16
RU2002117428A (ru) 2003-12-20
KR100479137B1 (ko) 2005-03-31
CN1468235A (zh) 2004-01-14
KR20020058064A (ko) 2002-07-12
WO2001040223B1 (en) 2002-05-30
AU2838901A (en) 2001-06-12
MXPA02005428A (es) 2002-11-29
BR0016034A (pt) 2002-07-30

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