ATE208374T1 - Beta-laktam und cepham verbindungen und ihre herstellung - Google Patents

Beta-laktam und cepham verbindungen und ihre herstellung

Info

Publication number
ATE208374T1
ATE208374T1 AT93903302T AT93903302T ATE208374T1 AT E208374 T1 ATE208374 T1 AT E208374T1 AT 93903302 T AT93903302 T AT 93903302T AT 93903302 T AT93903302 T AT 93903302T AT E208374 T1 ATE208374 T1 AT E208374T1
Authority
AT
Austria
Prior art keywords
lactam
beta
optionally substituted
production
compound
Prior art date
Application number
AT93903302T
Other languages
English (en)
Inventor
Shigeru Torii
Hideo Tanaka
Mitio Sasaoka
Takashi Shiroi
Yutaka Kameyama
Original Assignee
Otsuka Kagaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP03031092A external-priority patent/JP3227497B2/ja
Priority claimed from JP03031192A external-priority patent/JP3265381B2/ja
Application filed by Otsuka Kagaku Kk filed Critical Otsuka Kagaku Kk
Application granted granted Critical
Publication of ATE208374T1 publication Critical patent/ATE208374T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C07D205/095Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4 and with a nitrogen atom directly attached in position 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
AT93903302T 1992-02-18 1993-02-03 Beta-laktam und cepham verbindungen und ihre herstellung ATE208374T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP03031092A JP3227497B2 (ja) 1992-02-18 1992-02-18 β−ラクタム化合物及びその製造法
JP03031192A JP3265381B2 (ja) 1992-02-18 1992-02-18 2−置換メチル−3−セフェム化合物及びその製造法並びに2−エキソメチレンセフェム誘導体の製造法
PCT/JP1993/000131 WO1993016043A1 (en) 1992-02-18 1993-02-03 β-LACTAM COMPOUND AND CEPHEM COMPOUND, AND PRODUCTION THEREOF

Publications (1)

Publication Number Publication Date
ATE208374T1 true ATE208374T1 (de) 2001-11-15

Family

ID=26368636

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93903302T ATE208374T1 (de) 1992-02-18 1993-02-03 Beta-laktam und cepham verbindungen und ihre herstellung

Country Status (5)

Country Link
US (2) US5470972A (de)
EP (1) EP0592677B1 (de)
AT (1) ATE208374T1 (de)
DE (1) DE69331089T2 (de)
WO (1) WO1993016043A1 (de)

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JP6552412B2 (ja) 2013-09-05 2019-07-31 国立大学法人 宮崎大学 ヒトインテグリンa6b4と特異的に反応する抗体
TWI695011B (zh) 2014-06-18 2020-06-01 美商梅爾莎納醫療公司 抗her2表位之單株抗體及其使用之方法
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WO2022075439A1 (ja) 2020-10-08 2022-04-14 国立大学法人東海国立大学機構 抗トランスフェリンレセプター抗体の薬効又は感受性の判定方法
CN117836003A (zh) 2021-08-26 2024-04-05 株式会社英仙蛋白质科学 Ros(活性氧类)产生增强剂
WO2023116911A1 (zh) 2021-12-24 2023-06-29 百奥泰生物制药股份有限公司 抗FRα抗体及其抗体药物偶联物和用途
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Also Published As

Publication number Publication date
EP0592677A4 (en) 1994-07-06
DE69331089T2 (de) 2002-07-18
EP0592677B1 (de) 2001-11-07
DE69331089D1 (de) 2001-12-13
WO1993016043A1 (en) 1993-08-19
US5470972A (en) 1995-11-28
EP0592677A1 (de) 1994-04-20
US5693792A (en) 1997-12-02

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Legal Events

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REN Ceased due to non-payment of the annual fee