ATE163850T1 - Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen - Google Patents

Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen

Info

Publication number
ATE163850T1
ATE163850T1 AT93909884T AT93909884T ATE163850T1 AT E163850 T1 ATE163850 T1 AT E163850T1 AT 93909884 T AT93909884 T AT 93909884T AT 93909884 T AT93909884 T AT 93909884T AT E163850 T1 ATE163850 T1 AT E163850T1
Authority
AT
Austria
Prior art keywords
pct
rectal administration
agonistic
pharmaceutical compositions
sec
Prior art date
Application number
AT93909884T
Other languages
German (de)
English (en)
Inventor
Nadine Merlet
Isabelle Richard
Isabelle Thielemans
Original Assignee
Glaxo Wellcome Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Wellcome Lab filed Critical Glaxo Wellcome Lab
Application granted granted Critical
Publication of ATE163850T1 publication Critical patent/ATE163850T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
AT93909884T 1992-05-07 1993-05-03 Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen ATE163850T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929209882A GB9209882D0 (en) 1992-05-07 1992-05-07 Compositions

Publications (1)

Publication Number Publication Date
ATE163850T1 true ATE163850T1 (de) 1998-03-15

Family

ID=10715158

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93909884T ATE163850T1 (de) 1992-05-07 1993-05-03 Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen

Country Status (33)

Country Link
US (1) US5705506A (OSRAM)
EP (1) EP0639072B1 (OSRAM)
JP (1) JPH07506570A (OSRAM)
KR (1) KR100253111B1 (OSRAM)
AT (1) ATE163850T1 (OSRAM)
AU (1) AU670083B2 (OSRAM)
BE (1) BE1007024A5 (OSRAM)
BG (1) BG62120B1 (OSRAM)
BR (1) BR1100108A (OSRAM)
CA (1) CA2135179C (OSRAM)
CH (1) CH685920A5 (OSRAM)
CY (1) CY2039B1 (OSRAM)
CZ (1) CZ283512B6 (OSRAM)
DE (1) DE69317418T2 (OSRAM)
ES (1) ES2113533T3 (OSRAM)
FR (1) FR2690847B1 (OSRAM)
GB (2) GB9209882D0 (OSRAM)
GR (1) GR3026584T3 (OSRAM)
HK (1) HK95697A (OSRAM)
HU (2) HU227338B1 (OSRAM)
IE (1) IE75203B1 (OSRAM)
IL (1) IL105468A (OSRAM)
IT (1) IT1261471B (OSRAM)
NO (1) NO306700B1 (OSRAM)
NZ (1) NZ252132A (OSRAM)
OA (1) OA10109A (OSRAM)
RO (1) RO112993B1 (OSRAM)
RU (1) RU2118527C1 (OSRAM)
SG (1) SG46649A1 (OSRAM)
TW (1) TW231970B (OSRAM)
UA (1) UA37206C2 (OSRAM)
WO (1) WO1993021916A1 (OSRAM)
ZA (1) ZA933178B (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2434297A (en) * 1996-05-23 1997-12-09 Alcon Laboratories, Inc. The use of 5-ht1b/1d agonists to treat ocular pain
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
KR100440553B1 (ko) * 1998-03-26 2004-07-15 후지사와 야꾸힝 고교 가부시키가이샤 서방성 제제
WO2000051624A2 (en) * 1999-03-05 2000-09-08 The Trustees Of University Technology Corporation Methods and compositions useful in inhibiting apoptosis
AR056690A1 (es) * 2005-10-14 2007-10-17 Athersys Inc Derivados de indol como inhibidores de indol como inhibidores del receptor 3 de histamina para el tartamiento de trastornos del sueno y cognitivos obesidad y otros trastornos de snc
SI2124556T1 (sl) 2006-10-09 2015-01-30 Charleston Laboratories, Inc. Farmacevtske sestave
CA2749273C (en) 2008-01-09 2018-09-04 Charleston Laboratories, Inc. Pharmaceutical oral dosage form comprising a triptan and an antiemetic
EP3311667A1 (en) 2009-07-08 2018-04-25 Charleston Laboratories, Inc. Pharmaceutical compositions
EP2627328B1 (en) 2010-10-15 2016-09-14 Contera Pharma APS Combinations of serotonin receptor agonists for treatment of movement disorders
HUE037732T2 (hu) 2012-04-18 2018-09-28 Contera Pharma Aps A mozgászavarok fejlett kezelésére alkalmas, szájon át szedhetõ gyógyszerészeti készítmény
JP2019507181A (ja) 2016-03-04 2019-03-14 チャールストン ラボラトリーズ，インコーポレイテッド 医薬組成物
EP3481385B1 (en) 2016-07-11 2025-09-03 Contera Pharma A/S Pulsatile drug delivery system for treating morning akinesia

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
NZ197998A (en) * 1980-08-12 1985-08-16 Glaxo Group Ltd 5-amino(methyl)-1h-indol-3-ylalkaneamines
IT1170387B (it) * 1982-06-07 1987-06-03 Glaxo Group Ltd Composti eterociclici, procedimento per prepararli e composizioni farmaceutiche che li contengono
HU196752B (en) * 1983-12-06 1989-01-30 Glaxo Group Ltd Process for production of medical compositions containing indole-derivatives and these compounds
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
GB2162522B (en) * 1984-08-01 1988-02-24 Glaxo Group Ltd An indole derivative
US4785016A (en) * 1984-12-04 1988-11-15 Glaxo Group Limited Indole derivatives
GB8431426D0 (en) * 1984-12-13 1985-01-23 Glaxo Group Ltd Chemical compounds
DE3678805D1 (de) * 1985-11-08 1991-05-23 Glaxo Group Ltd Indolderivate.
ES2058292T3 (es) * 1987-08-13 1994-11-01 Glaxo Group Ltd Derivados de indol.
ATE156823T1 (de) * 1990-06-07 1997-08-15 Zeneca Ltd Therapeutische heterocyclische verbindungen

Also Published As

Publication number Publication date
GR3026584T3 (en) 1998-07-31
CH685920A5 (fr) 1995-11-15
EP0639072B1 (en) 1998-03-11
GB9309209D0 (en) 1993-06-16
SG46649A1 (en) 1998-02-20
CA2135179A1 (en) 1993-11-11
GB2266665B (en) 1996-05-22
NO944214L (no) 1994-11-07
CZ283512B6 (cs) 1998-04-15
GB2266665A (en) 1993-11-10
WO1993021916A1 (en) 1993-11-11
NZ252132A (en) 1996-09-25
IT1261471B (it) 1996-05-23
OA10109A (en) 1996-12-18
IL105468A (en) 1998-09-24
NO306700B1 (no) 1999-12-13
ZA933178B (en) 1994-01-10
CA2135179C (en) 2000-12-05
BE1007024A5 (fr) 1995-02-21
FR2690847B1 (fr) 1995-06-09
HUT71418A (en) 1995-11-28
ITRM930286A1 (it) 1994-11-06
HK95697A (en) 1997-08-08
HU211638A9 (en) 1995-12-28
DE69317418D1 (de) 1998-04-16
BG99167A (bg) 1995-06-30
CY2039B1 (en) 1998-04-30
IE930339A1 (en) 1993-11-17
BR1100108A (pt) 1999-12-07
UA37206C2 (uk) 2001-05-15
KR100253111B1 (en) 2000-07-01
NO944214D0 (no) 1994-11-04
CZ272394A3 (en) 1995-10-18
RU2118527C1 (ru) 1998-09-10
IE75203B1 (en) 1997-08-27
DE69317418T2 (de) 1998-07-30
IL105468A0 (en) 1993-08-18
AU4064093A (en) 1993-11-29
AU670083B2 (en) 1996-07-04
TW231970B (OSRAM) 1994-10-11
ITRM930286A0 (it) 1993-05-06
FR2690847A1 (fr) 1993-11-12
JPH07506570A (ja) 1995-07-20
BG62120B1 (bg) 1999-03-31
HU227338B1 (en) 2011-04-28
GB9209882D0 (en) 1992-06-24
ES2113533T3 (es) 1998-05-01
EP0639072A1 (en) 1995-02-22
RO112993B1 (ro) 1998-03-30
US5705506A (en) 1998-01-06

Similar Documents

Publication Publication Date Title
FR2714378B1 (fr) Dérivés de l'indol-2-one substitués en 3 par un groupe azoté, leur préparation, les compositions pharmaceutiques en contenant.
HUP0100266A2 (hu) NMDA-receptor-antagonista hatású 1-aminoalkilciklohexánszármazékok, a vegyületeket tartalmazó gyógyszerkészítmények és előállításaik
DK0889877T3 (da) Meta-substituerede phenylenderivater og deres anvendelse som alfav-beta3-integrin-antagonister eller -inhibitorer
ES2160949T3 (es) Derivados de fenilen-sulfonamida sustituidos en meta.
MX9301032A (es) Compuestos farmaceuticos y procedimento para su preparacion
ATE163850T1 (de) Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen
KR870003974A (ko) 비시클로 치환된 페닐아세토니트릴 유도체
ZA971279B (en) Use of 5ht4 receptor antagonists for overcoming gastrointestinal effects of serotonin reuptake inhinitors
NO306345B1 (no) Piperidin-derivater med PAF antagonist-aktivitet, anvendelse derav og farmasöytisk blanding
ATE148989T1 (de) Partielle agonisten der strychnin unempfindlichen glycinmodulierenden stelle des n-methyl-d- aspartat-rezeptor-komplexes als neuropsycho- pharmakologische wirkstoffe
KR950000663A (ko) 트리테르펜 유도체 및 이를 함유하는 엔도텔린-수용체 길항물질
NO972623D0 (no) Framasöytisk blanding omfattende lamotrigin
SE9702002D0 (sv) Novel compounds
FR2724933B1 (OSRAM)
FI950209A0 (fi) Farmakologisesti aktiiviset alfa-(tertiaarinen-amino-metyyli)-bentseenimetanolijohdannaiset
TW371661B (en) Novel intermediates and their use to prepare N,N'-bridged bisindolylmaleimides
NO20010907L (no) Medikament inneholdende platinakompleksforbindelser og anvendelse derav
ATE141248T1 (de) Neue bis-phenyl-hexene
KR910007526A (ko) 인터류킨-1 생합성 억제제로의 3-치화된-2-옥신돌 유도체

Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification