ATE116135T1 - Einschlusskomplex von nimesulide mit cyclodextrinen. - Google Patents

Einschlusskomplex von nimesulide mit cyclodextrinen.

Info

Publication number
ATE116135T1
ATE116135T1 AT91909437T AT91909437T ATE116135T1 AT E116135 T1 ATE116135 T1 AT E116135T1 AT 91909437 T AT91909437 T AT 91909437T AT 91909437 T AT91909437 T AT 91909437T AT E116135 T1 ATE116135 T1 AT E116135T1
Authority
AT
Austria
Prior art keywords
nimesulide
cyclodextrins
inclusion complex
cyclodextrin
comprised
Prior art date
Application number
AT91909437T
Other languages
English (en)
Inventor
Giuseppe Bietti
Enrica Dubini
Grazia Maffione
Aldo Vidi
Original Assignee
Boehringer Ingelheim Italia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Italia filed Critical Boehringer Ingelheim Italia
Application granted granted Critical
Publication of ATE116135T1 publication Critical patent/ATE116135T1/de

Links

Classifications

    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nanotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Biotechnology (AREA)
  • General Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Medical Informatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Ceramic Products (AREA)
  • Fats And Perfumes (AREA)
  • Ink Jet (AREA)
  • Ink Jet Recording Methods And Recording Media Thereof (AREA)
  • Slide Fasteners, Snap Fasteners, And Hook Fasteners (AREA)
  • Manufacture And Refinement Of Metals (AREA)
AT91909437T 1990-05-22 1991-05-20 Einschlusskomplex von nimesulide mit cyclodextrinen. ATE116135T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT02039390A IT1248475B (it) 1990-05-22 1990-05-22 Composti di inclusione di nimesulide con ciclodestrine

Publications (1)

Publication Number Publication Date
ATE116135T1 true ATE116135T1 (de) 1995-01-15

Family

ID=11166307

Family Applications (1)

Application Number Title Priority Date Filing Date
AT91909437T ATE116135T1 (de) 1990-05-22 1991-05-20 Einschlusskomplex von nimesulide mit cyclodextrinen.

Country Status (15)

Country Link
EP (1) EP0534995B1 (de)
JP (1) JP3417942B2 (de)
KR (1) KR100198046B1 (de)
AT (1) ATE116135T1 (de)
AU (1) AU655183B2 (de)
DE (1) DE69106361T2 (de)
DK (1) DK0534995T3 (de)
ES (1) ES2065687T3 (de)
FI (1) FI102462B (de)
GR (1) GR3015468T3 (de)
HK (1) HK1006413A1 (de)
HU (1) HU214336B (de)
IT (1) IT1248475B (de)
NO (1) NO304730B1 (de)
WO (1) WO1991017774A1 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1255462B (it) * 1992-07-28 1995-11-02 Grazia Maffione Metodo di preparazione di composti di inclusione di nimesulide con ciclodestrine
HU210922B (en) * 1993-05-24 1995-09-28 Europharmaceuticals Sa Nimesulide alkali salt cyclodextrin inclusion complexes their preparation and pharmaceutical compositions containing them
BE1008307A3 (fr) * 1994-06-16 1996-04-02 Europharmaceuticals Sa Sel de nimesulide hydrosoluble, solution aqueuse le contenant, sa preparation et son utilisation.
US5837735A (en) * 1994-10-05 1998-11-17 Helsinn Healthcare S.A. Antiinflammatory agent for external use
HUP9601442A3 (en) * 1995-07-25 1999-03-29 Panacea Biotec Ltd Nes antinflammatory and analgetic pharmaceutical compositions, containing nimesulid for transdermal use, and process for producing them
RO116040B1 (ro) 1995-10-05 2000-10-30 Hisamitsu Pharmaceutical Co Compozitie antiinflamatoare pentru uz extern
HUP9601443A3 (en) * 1996-05-29 1999-03-29 Panacea Biotec Ltd Injectable analgetic pharmaceutical compositions for intramuscular use containing nimesulid, and process for producing them
IN186315B (de) * 1996-12-12 2001-08-04 Panacea Biotec Ltd
IT1291895B1 (it) 1997-04-24 1999-01-21 Errekappa Euroterapici S P A Preparazione farmaceutica fluida a base di nimesulide per uso orale e rinofaringeo
WO1999041233A1 (en) * 1998-02-17 1999-08-19 Micio Pharma Chemical Aktiengesellschaft A watersoluble nimesulide adduct also for injectable use
IT1298732B1 (it) * 1998-03-13 2000-02-02 Recordati Chem Pharm Composizioni farmaceutiche orali assumibili senza liquidi,contenenti complessi di inclusione
KR100395247B1 (ko) * 2000-08-30 2003-08-21 디디에스텍주식회사 비자극성 캡사이신 경피 투여 제형
EP1902705A1 (de) * 2006-09-22 2008-03-26 Pharmatex Italia Srl Injizierbare pharmazeutische Lösungen mit Nimesulid

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR206496A1 (es) * 1972-07-03 1976-07-30 Riker Laboratories Inc Procedimiento para la preparacion de 2-fenoxi-4-nitro-alquil o haloalquilsulfonanilidas

Also Published As

Publication number Publication date
DE69106361T2 (de) 1995-05-18
FI102462B1 (fi) 1998-12-15
DE69106361D1 (de) 1995-02-09
HK1006413A1 (en) 1999-02-26
FI925224A (fi) 1992-11-18
FI102462B (fi) 1998-12-15
DK0534995T3 (da) 1995-05-01
IT1248475B (it) 1995-01-19
GR3015468T3 (en) 1995-06-30
JP3417942B2 (ja) 2003-06-16
NO924492L (no) 1993-01-20
ES2065687T3 (es) 1995-02-16
HU214336B (hu) 1998-03-02
AU7866591A (en) 1991-12-10
JPH06502842A (ja) 1994-03-31
AU655183B2 (en) 1994-12-08
FI925224A0 (fi) 1992-11-18
NO304730B1 (no) 1999-02-08
EP0534995A1 (de) 1993-04-07
EP0534995B1 (de) 1994-12-28
HUT65418A (en) 1994-06-28
NO924492D0 (no) 1992-11-20
KR937000160A (ko) 1993-03-13
HU9203649D0 (en) 1993-03-29
WO1991017774A1 (en) 1991-11-28
KR100198046B1 (ko) 1999-06-15
IT9020393A0 (de) 1990-05-22
IT9020393A1 (it) 1991-11-22

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
EEIH Change in the person of patent owner
EEIH Change in the person of patent owner
REN Ceased due to non-payment of the annual fee