AR076002A1 - Derivados imidazolicos heterociclicos utiles como agentes antivirales para hepatitis c y composiciones farmaceuticas que los comprenden. - Google Patents

Derivados imidazolicos heterociclicos utiles como agentes antivirales para hepatitis c y composiciones farmaceuticas que los comprenden.

Info

Publication number
AR076002A1
AR076002A1 ARP100101038A ARP100101038A AR076002A1 AR 076002 A1 AR076002 A1 AR 076002A1 AR P100101038 A ARP100101038 A AR P100101038A AR P100101038 A ARP100101038 A AR P100101038A AR 076002 A1 AR076002 A1 AR 076002A1
Authority
AR
Argentina
Prior art keywords
alkyl
hydrogen
independently selected
nrarb
cycloalkyl
Prior art date
Application number
ARP100101038A
Other languages
English (en)
Spanish (es)
Inventor
John A Bender
John F Kadow
Piyasena Hewawasam
Jeffrey Lee Romine
Lawrence B Snyder
Van N Nguyen
Omar D Lopez
Nicholas A Meanwell
Makonen Belema
Gan Wang
Lauren Denis R St
Ningning Xu
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42320079&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR076002(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of AR076002A1 publication Critical patent/AR076002A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Virology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ARP100101038A 2009-03-30 2010-03-30 Derivados imidazolicos heterociclicos utiles como agentes antivirales para hepatitis c y composiciones farmaceuticas que los comprenden. AR076002A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US16453109P 2009-03-30 2009-03-30
US12/729,940 US8796466B2 (en) 2009-03-30 2010-03-23 Hepatitis C virus inhibitors

Publications (1)

Publication Number Publication Date
AR076002A1 true AR076002A1 (es) 2011-05-11

Family

ID=42320079

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP100101038A AR076002A1 (es) 2009-03-30 2010-03-30 Derivados imidazolicos heterociclicos utiles como agentes antivirales para hepatitis c y composiciones farmaceuticas que los comprenden.

Country Status (19)

Country Link
US (1) US8796466B2 (enExample)
EP (1) EP2414350B1 (enExample)
JP (1) JP5612660B2 (enExample)
KR (1) KR20120034603A (enExample)
CN (1) CN102448956B (enExample)
AR (1) AR076002A1 (enExample)
AU (1) AU2010234970A1 (enExample)
BR (1) BRPI1013393A2 (enExample)
CA (1) CA2757269A1 (enExample)
CL (1) CL2011002426A1 (enExample)
CO (1) CO6430431A2 (enExample)
EA (1) EA022384B1 (enExample)
IL (1) IL215055A0 (enExample)
MX (1) MX2011009948A (enExample)
NZ (1) NZ595168A (enExample)
PE (1) PE20120546A1 (enExample)
SG (1) SG174521A1 (enExample)
WO (1) WO2010117635A1 (enExample)
ZA (1) ZA201106795B (enExample)

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CO6430431A2 (es) 2012-04-30
EP2414350B1 (en) 2014-11-12
US20110077280A1 (en) 2011-03-31
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CA2757269A1 (en) 2010-10-14
IL215055A0 (en) 2011-11-30
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EA201171152A1 (ru) 2012-10-30
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JP2012522053A (ja) 2012-09-20
SG174521A1 (en) 2011-10-28
MX2011009948A (es) 2011-10-06
WO2010117635A1 (en) 2010-10-14
AU2010234970A1 (en) 2011-10-06
NZ595168A (en) 2013-05-31
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US8796466B2 (en) 2014-08-05
EA022384B1 (ru) 2015-12-30
KR20120034603A (ko) 2012-04-12

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