AR012997A1 - Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene. - Google Patents

Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene.

Info

Publication number
AR012997A1
AR012997A1 ARP980102883A ARP980102883A AR012997A1 AR 012997 A1 AR012997 A1 AR 012997A1 AR P980102883 A ARP980102883 A AR P980102883A AR P980102883 A ARP980102883 A AR P980102883A AR 012997 A1 AR012997 A1 AR 012997A1
Authority
AR
Argentina
Prior art keywords
insulin
thiazolidin
amino
methyl
preparation
Prior art date
Application number
ARP980102883A
Other languages
English (en)
Spanish (es)
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of AR012997A1 publication Critical patent/AR012997A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/28Insulins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
ARP980102883A 1997-06-18 1998-06-17 Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene. AR012997A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9712866.4A GB9712866D0 (en) 1997-06-18 1997-06-18 Novel method of treatment

Publications (1)

Publication Number Publication Date
AR012997A1 true AR012997A1 (es) 2000-11-22

Family

ID=10814527

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP980102883A AR012997A1 (es) 1997-06-18 1998-06-17 Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4- diona e insulina para la preparacion de medicamentos, y composicionfarmaceutica que los contiene.
ARP980102886A AR015894A1 (es) 1997-06-18 1998-06-17 Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4-diona e insulina para la preparacion de un medicamento y composicion farmaceuticaque contiene dichos compuestos

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP980102886A AR015894A1 (es) 1997-06-18 1998-06-17 Uso de 5-[4-[2-(n-metil-n-(2-piridil)amino)etoxi]bencil]tiazolidin-2,4-diona e insulina para la preparacion de un medicamento y composicion farmaceuticaque contiene dichos compuestos

Country Status (30)

Country Link
EP (1) EP0999837A1 (pt)
JP (1) JP2002504138A (pt)
KR (1) KR20010013843A (pt)
CN (1) CN1133431C (pt)
AP (1) AP1287A (pt)
AR (2) AR012997A1 (pt)
AU (1) AU8216398A (pt)
BG (1) BG104059A (pt)
BR (1) BR9810444A (pt)
CA (1) CA2294141A1 (pt)
CO (1) CO4940454A1 (pt)
DZ (1) DZ2521A1 (pt)
EA (1) EA004800B1 (pt)
GB (1) GB9712866D0 (pt)
HU (1) HUP0003260A3 (pt)
ID (1) ID23951A (pt)
IL (1) IL133143A0 (pt)
IN (1) IN189723B (pt)
MA (1) MA26511A1 (pt)
NO (1) NO996265D0 (pt)
OA (1) OA11517A (pt)
PE (1) PE104499A1 (pt)
PL (1) PL343123A1 (pt)
SK (1) SK179399A3 (pt)
TR (1) TR199903095T2 (pt)
TW (1) TW587937B (pt)
UA (1) UA70299C2 (pt)
UY (1) UY25050A1 (pt)
WO (1) WO1998057636A1 (pt)
ZA (1) ZA985237B (pt)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6291495B1 (en) * 1997-02-24 2001-09-18 Robert B. Rieveley Method and composition for the treatment of diabetes
TWI249401B (en) 1999-04-14 2006-02-21 Takeda Chemical Industries Ltd Agent for improving ketosis
US6815457B1 (en) 1999-04-23 2004-11-09 Smithkline Beecham P.L.C. Thiazolidinedione derivative and its use as antidiabetic
WO2000078333A2 (en) * 1999-06-21 2000-12-28 Eli Lilly And Company Synergetic use of thiazolidinediones with glucagon-like peptide-1 and agonists thereof to treat non-insulin dependant diabetes
WO2001000223A2 (en) * 1999-06-25 2001-01-04 Minimed Inc. Multiple agent diabetes therapy
US6468507B1 (en) * 2000-05-01 2002-10-22 Aeropharm Technology, Inc. Non-aqueous aerosol formulation comprising rosiglitazone maleate, a non-aqueous carrier, and an amino acid stabilizer
GB0023970D0 (en) * 2000-09-29 2000-11-15 Smithkline Beecham Plc Novel pharmaceutical
US6852694B2 (en) 2001-02-21 2005-02-08 Medtronic Minimed, Inc. Stabilized insulin formulations
US6531461B1 (en) 2001-06-04 2003-03-11 Louis Obyo Obyo Nelson Medicament for the treatment of diabetes
WO2002100396A1 (en) * 2001-06-07 2002-12-19 Wyeth COMBINATION OF A PTPase INHIBITOR AND A THIAZOLIDINEDIONE AGENT
US6737401B2 (en) 2001-06-28 2004-05-18 Metronic Minimed, Inc. Methods of evaluating protein formulation stability and surfactant-stabilized insulin formulations derived therefrom
KR100699614B1 (ko) * 2002-11-08 2007-03-23 에프. 호프만-라 로슈 아게 퍼옥시좀 증식자 활성화된 수용체 작용제로서의 치환된4-알콕시옥사졸 유도체
US7264813B2 (en) * 2003-09-24 2007-09-04 Nikken Sohonsha Corporation Therapeutic uses of Dunaliella powder
CN102389427A (zh) * 2011-10-10 2012-03-28 成都恒瑞制药有限公司 含有罗格列酮和盐酸西替利嗪的固体口服制剂

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ283339B6 (cs) * 1993-09-15 1998-03-18 Sankyo Company Limited Použití thiazolidinových derivátů pro výrobu léčivého přípravku pro léčení zhoršené tolerance glukosy pro zabránění nebo zpoždění nástupu diabetes mellitus nezávislé na inzulinu
CZ32998A3 (cs) * 1995-08-10 1998-10-14 Warner-Lambert Company Výroba léčiva pro snížení množství exogenního insulinu
EP1426048A3 (en) * 1995-09-18 2004-06-16 Ligand Pharmaceuticals, Inc. Treating hypertriglyceridemia with RXR agonists in combination with a PPARgamma agonist

Also Published As

Publication number Publication date
DZ2521A1 (fr) 2003-02-08
EA004800B1 (ru) 2004-08-26
EA200000042A1 (ru) 2000-08-28
CN1133431C (zh) 2004-01-07
IN189723B (pt) 2003-04-19
SK179399A3 (en) 2000-11-07
ID23951A (id) 2000-06-08
WO1998057636A1 (en) 1998-12-23
CO4940454A1 (es) 2000-07-24
CN1260715A (zh) 2000-07-19
AR015894A1 (es) 2001-05-30
BG104059A (en) 2000-10-31
PE104499A1 (es) 2000-01-13
JP2002504138A (ja) 2002-02-05
UA70299C2 (en) 2004-10-15
PL343123A1 (en) 2001-07-30
GB9712866D0 (en) 1997-08-20
HUP0003260A3 (en) 2001-12-28
ZA985237B (en) 2000-02-17
IL133143A0 (en) 2001-03-19
TR199903095T2 (xx) 2000-08-21
OA11517A (en) 2004-02-04
UY25050A1 (es) 2000-09-29
HUP0003260A2 (hu) 2001-05-28
BR9810444A (pt) 2000-09-05
NO996265L (no) 1999-12-17
EP0999837A1 (en) 2000-05-17
NO996265D0 (no) 1999-12-17
KR20010013843A (ko) 2001-02-26
AP1287A (en) 2004-06-26
AP9901718A0 (en) 1999-12-31
TW587937B (en) 2004-05-21
MA26511A1 (fr) 2004-12-20
CA2294141A1 (en) 1998-12-23
AU8216398A (en) 1999-01-04

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