AR005642A1 - Compuestos antibioticos de cefalosporina, uso de los mismos para preparar composiciones farmaceuticas, dichas composiciones farmaceuticas que los comprenden,compuestos intermediarios de aplicacion en la preparacion de los primeros y metodo para elaborar dichos compuestos intermediarios - Google Patents

Compuestos antibioticos de cefalosporina, uso de los mismos para preparar composiciones farmaceuticas, dichas composiciones farmaceuticas que los comprenden,compuestos intermediarios de aplicacion en la preparacion de los primeros y metodo para elaborar dichos compuestos intermediarios

Info

Publication number
AR005642A1
AR005642A1 ARP960104714A ARP960104714A AR005642A1 AR 005642 A1 AR005642 A1 AR 005642A1 AR P960104714 A ARP960104714 A AR P960104714A AR P960104714 A ARP960104714 A AR P960104714A AR 005642 A1 AR005642 A1 AR 005642A1
Authority
AR
Argentina
Prior art keywords
preparation
pharmaceutical compositions
compositions
application
compounds
Prior art date
Application number
ARP960104714A
Other languages
English (en)
Original Assignee
Essential Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Essential Therapeutics Inc filed Critical Essential Therapeutics Inc
Publication of AR005642A1 publication Critical patent/AR005642A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)

Abstract

Nuevos compuestos antibióticos de cefalosporina de fórmula (I) donde los sustituyentes tienen los valores indicados en la descripción. También seproponen composiciones farmacéuticas de aplicación para el tratamiento de infeccionesbacteriana s, especialmente de aquellas que son debidas a bacteriasresistentes a las beta-lactamas convencionales y, además la preparación de dichos antibióticos y compuestos intermediarios de aplicación en la preparaciónde dichos antibióticosy métodos de aplicación de dichos antibióticos para el tratamiento de infecciones bacterianas.
ARP960104714A 1995-10-12 1996-10-11 Compuestos antibioticos de cefalosporina, uso de los mismos para preparar composiciones farmaceuticas, dichas composiciones farmaceuticas que los comprenden,compuestos intermediarios de aplicacion en la preparacion de los primeros y metodo para elaborar dichos compuestos intermediarios AR005642A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US538995P 1995-10-12 1995-10-12

Publications (1)

Publication Number Publication Date
AR005642A1 true AR005642A1 (es) 1999-07-14

Family

ID=21715599

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP960104714A AR005642A1 (es) 1995-10-12 1996-10-11 Compuestos antibioticos de cefalosporina, uso de los mismos para preparar composiciones farmaceuticas, dichas composiciones farmaceuticas que los comprenden,compuestos intermediarios de aplicacion en la preparacion de los primeros y metodo para elaborar dichos compuestos intermediarios

Country Status (27)

Country Link
US (4) US6066630A (es)
EP (1) EP0874854B1 (es)
JP (1) JPH11513670A (es)
KR (2) KR100491466B1 (es)
CN (3) CN1183142C (es)
AR (1) AR005642A1 (es)
AT (1) ATE210666T1 (es)
AU (1) AU708676B2 (es)
BR (1) BR9611062A (es)
CA (1) CA2234255A1 (es)
CZ (1) CZ108998A3 (es)
DE (1) DE69618015T2 (es)
DK (1) DK0874854T3 (es)
ES (1) ES2164924T3 (es)
HU (1) HUP9802545A3 (es)
IL (1) IL123983A (es)
MX (1) MX9802891A (es)
MY (1) MY127641A (es)
NO (1) NO323007B1 (es)
NZ (1) NZ321135A (es)
PL (1) PL192069B1 (es)
PT (1) PT874854E (es)
RO (1) RO119830B1 (es)
SK (1) SK283524B6 (es)
TW (1) TW474935B (es)
WO (1) WO1997013772A2 (es)
ZA (1) ZA968617B (es)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1295935B1 (it) 1997-10-30 1999-05-28 Acs Dobfar Spa Derivati aminotiazolici utili nella preparazione di antibiotici b -lattamici
US6159706A (en) * 1997-12-23 2000-12-12 Newbiotics, Inc. Application of enzyme prodrugs as anti-infective agents
US6723716B1 (en) * 1999-09-22 2004-04-20 Essential Therapeutics, Inc. 7-acylamino-3-heteroarylthio-3-cephem carboxylic acid antibiotics and prodrugs thereof
AR029004A1 (es) * 1999-09-22 2003-06-04 Essential Therapeutics Inc Compuesto del acido 7-acilamino-3-heteroariltio-3-cefem carboxilico y su uso para la preparacion de una composicion antibacteriana
JP2004505896A (ja) * 2000-07-07 2004-02-26 エルジー・ライフ・サイエンシーズ・リミテッド 新規なセファロスポリン化合物およびその製造方法
WO2002004464A1 (en) * 2000-07-07 2002-01-17 Lg Life Sciences Ltd Novel cephalosporin compounds and process for preparing the same
US6599893B2 (en) * 2000-08-29 2003-07-29 Essential Therapeutics, Inc. Cephalosporin antibiotics and prodrugs thereof
EP1320533A4 (en) * 2000-09-21 2004-12-15 Essential Therapeutics Inc 7-ACYLAMINO-3-HETEROARYLTHIO-3-CEPHEM CARBOXYLIC ANTIBIOTIC PREDICTIONS
AU2002234148A1 (en) 2000-12-29 2002-07-16 Bellsouth Intellectual Property Corporation Web based messaging system with personalized caller specific messages
US7119062B1 (en) 2001-02-23 2006-10-10 Neucoll, Inc. Methods and compositions for improved articular surgery using collagen
EP1392639B1 (en) 2001-05-03 2008-09-17 Galileo Laboratories, Inc. Pyruvate derivatives
US6608196B2 (en) 2001-05-03 2003-08-19 Galileo Pharmaceuticals, Inc. Process for solid supported synthesis of pyruvate-derived compounds
KR20030071311A (ko) * 2002-02-28 2003-09-03 주식회사 엘지생명과학 신규 세팔로스포린 화합물 및 그의 제조방법
AU2003240545A1 (en) * 2002-06-06 2003-12-22 Therapeutics Corporation Genome Use of ramoplanin to treat diseases associated with the use of antibiotics
WO2004017925A2 (en) * 2002-08-23 2004-03-04 Genome Therapeutics Corporation Methods and reagents for preventing bacteremias
CA2523573A1 (en) * 2003-04-25 2004-11-11 Oscient Pharmaceuticals Corporation Methods for reducing or preventing transmission of nosocomial pathogens in a health care facility
EA201792028A1 (ru) 2015-03-13 2018-04-30 Форма Терапьютикс, Инк. Альфа-цинамидные соединения и композиции как ингибиторы hdac8
WO2017155765A1 (en) * 2016-03-07 2017-09-14 Merck Sharp & Dohme Corp. Bicyclic aryl monobactam compounds and methods of use thereof for the treatment of bacterial infections
CN114671892B (zh) * 2022-04-24 2023-04-11 江苏海洋大学 含7-氨基头孢烷酸的1,3,4-噻二唑衍生物及制法与用途
CN121181575B (zh) * 2025-11-24 2026-02-24 重庆汉佩生物科技有限公司 一种抗菌化合物和应用以及制备方法

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CH605997A5 (es) * 1974-08-30 1978-10-13 Ciba Geigy Ag
US3992377A (en) * 1974-12-13 1976-11-16 Eli Lilly And Company 3-Thio-substituted cephalosporin antibiotics
SE8003820L (sv) * 1979-05-23 1980-11-24 Rhone Poulenc Ind Nya 3-tiovinylcefalosporiner, forfaranden for framstellning av desamma och farmaceutiska kompositioner innehallande desamma
FR2457297A1 (fr) * 1979-05-23 1980-12-19 Rhone Poulenc Ind Nouvelles vinyl-3 cephalosporines, et leur preparation
FR2494274A2 (fr) * 1980-11-20 1982-05-21 Rhone Poulenc Ind Nouvelles thiovinyl-3 cephalosporines, leur preparation et les medicaments qui les contiennent
GR79043B (es) * 1982-12-06 1984-10-02 Fujisawa Pharmaceutical Co
US4847373A (en) * 1987-02-26 1989-07-11 Bristol-Myers Company Production of 3-allyl- and 3-butenyl-3-cephems
US5025006A (en) * 1990-06-26 1991-06-18 Merck & Co., Inc. 2-biphenyl-carbapenem antibacterial agents
US5077287A (en) * 1991-01-18 1991-12-31 Eli Lilly And Company 3-thiazolylthio carbacephem antibacterial agents
JPH05132488A (ja) * 1991-08-13 1993-05-28 Meiji Seika Kaisha Ltd 新規セフアロスポリン誘導体
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Also Published As

Publication number Publication date
CN1183142C (zh) 2005-01-05
CN1291611A (zh) 2001-04-18
MY127641A (en) 2006-12-29
NO981653D0 (no) 1998-04-08
US6087355A (en) 2000-07-11
PT874854E (pt) 2002-06-28
CN1204336A (zh) 1999-01-06
EP0874854A2 (en) 1998-11-04
IL123983A (en) 2007-03-08
MX9802891A (es) 1998-09-30
PL192069B1 (pl) 2006-08-31
US6066630A (en) 2000-05-23
WO1997013772A2 (en) 1997-04-17
ES2164924T3 (es) 2002-03-01
PL326150A1 (en) 1998-08-31
BR9611062A (pt) 1999-07-13
AU708676B2 (en) 1999-08-12
SK283524B6 (sk) 2003-09-11
TW474935B (en) 2002-02-01
EP0874854B1 (en) 2001-12-12
US5859256A (en) 1999-01-12
HK1034191A1 (en) 2001-10-19
KR20040047794A (ko) 2004-06-05
CZ108998A3 (cs) 1998-07-15
CA2234255A1 (en) 1997-04-17
CN1066735C (zh) 2001-06-06
KR100455544B1 (ko) 2005-01-15
HK1034248A1 (en) 2001-10-19
NZ321135A (en) 2000-01-28
WO1997013772A3 (en) 1997-06-05
JPH11513670A (ja) 1999-11-24
RO119830B1 (ro) 2005-04-29
KR19990064201A (ko) 1999-07-26
HUP9802545A3 (en) 2001-01-29
ZA968617B (en) 1997-10-21
DE69618015D1 (de) 2002-01-24
CN1179963C (zh) 2004-12-15
US6057312A (en) 2000-05-02
HK1017887A1 (zh) 1999-12-03
NO323007B1 (no) 2006-12-18
ATE210666T1 (de) 2001-12-15
NO981653L (no) 1998-06-11
CN1291612A (zh) 2001-04-18
SK46498A3 (en) 1998-10-07
HUP9802545A2 (hu) 1999-05-28
DK0874854T3 (da) 2002-03-25
DE69618015T2 (de) 2002-05-16
AU7441796A (en) 1997-04-30
KR100491466B1 (ko) 2005-05-25

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