AR005642A1 - Compuestos antibioticos de cefalosporina, uso de los mismos para preparar composiciones farmaceuticas, dichas composiciones farmaceuticas que los comprenden,compuestos intermediarios de aplicacion en la preparacion de los primeros y metodo para elaborar dichos compuestos intermediarios - Google Patents
Compuestos antibioticos de cefalosporina, uso de los mismos para preparar composiciones farmaceuticas, dichas composiciones farmaceuticas que los comprenden,compuestos intermediarios de aplicacion en la preparacion de los primeros y metodo para elaborar dichos compuestos intermediariosInfo
- Publication number
- AR005642A1 AR005642A1 ARP960104714A ARP960104714A AR005642A1 AR 005642 A1 AR005642 A1 AR 005642A1 AR P960104714 A ARP960104714 A AR P960104714A AR P960104714 A ARP960104714 A AR P960104714A AR 005642 A1 AR005642 A1 AR 005642A1
- Authority
- AR
- Argentina
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions
- application
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
Abstract
Nuevos compuestos antibióticos de cefalosporina de fórmula (I) donde los sustituyentes tienen los valores indicados en la descripción. También seproponen composiciones farmacéuticas de aplicación para el tratamiento de infeccionesbacteriana s, especialmente de aquellas que son debidas a bacteriasresistentes a las beta-lactamas convencionales y, además la preparación de dichos antibióticos y compuestos intermediarios de aplicación en la preparaciónde dichos antibióticosy métodos de aplicación de dichos antibióticos para el tratamiento de infecciones bacterianas.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US538995P | 1995-10-12 | 1995-10-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR005642A1 true AR005642A1 (es) | 1999-07-14 |
Family
ID=21715599
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP960104714A AR005642A1 (es) | 1995-10-12 | 1996-10-11 | Compuestos antibioticos de cefalosporina, uso de los mismos para preparar composiciones farmaceuticas, dichas composiciones farmaceuticas que los comprenden,compuestos intermediarios de aplicacion en la preparacion de los primeros y metodo para elaborar dichos compuestos intermediarios |
Country Status (28)
Country | Link |
---|---|
US (4) | US6057312A (es) |
EP (1) | EP0874854B1 (es) |
JP (1) | JPH11513670A (es) |
KR (2) | KR100491466B1 (es) |
CN (3) | CN1183142C (es) |
AR (1) | AR005642A1 (es) |
AT (1) | ATE210666T1 (es) |
AU (1) | AU708676B2 (es) |
BR (1) | BR9611062A (es) |
CA (1) | CA2234255A1 (es) |
CZ (1) | CZ108998A3 (es) |
DE (1) | DE69618015T2 (es) |
DK (1) | DK0874854T3 (es) |
ES (1) | ES2164924T3 (es) |
HK (3) | HK1017887A1 (es) |
HU (1) | HUP9802545A3 (es) |
IL (1) | IL123983A (es) |
MX (1) | MX9802891A (es) |
MY (1) | MY127641A (es) |
NO (1) | NO323007B1 (es) |
NZ (1) | NZ321135A (es) |
PL (1) | PL192069B1 (es) |
PT (1) | PT874854E (es) |
RO (1) | RO119830B1 (es) |
SK (1) | SK283524B6 (es) |
TW (1) | TW474935B (es) |
WO (1) | WO1997013772A2 (es) |
ZA (1) | ZA968617B (es) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1295935B1 (it) | 1997-10-30 | 1999-05-28 | Acs Dobfar Spa | Derivati aminotiazolici utili nella preparazione di antibiotici b -lattamici |
US6159706A (en) * | 1997-12-23 | 2000-12-12 | Newbiotics, Inc. | Application of enzyme prodrugs as anti-infective agents |
AR029004A1 (es) * | 1999-09-22 | 2003-06-04 | Essential Therapeutics Inc | Compuesto del acido 7-acilamino-3-heteroariltio-3-cefem carboxilico y su uso para la preparacion de una composicion antibacteriana |
US6723716B1 (en) * | 1999-09-22 | 2004-04-20 | Essential Therapeutics, Inc. | 7-acylamino-3-heteroarylthio-3-cephem carboxylic acid antibiotics and prodrugs thereof |
US20030162762A1 (en) * | 2000-07-07 | 2003-08-28 | Chang-Seok Lee | Novel cephalosporin compounds and process for preparing the same |
CA2409329A1 (en) * | 2000-07-07 | 2002-01-17 | Lg Life Sciences Ltd. | Novel cephalosporin compounds and process for preparing the same |
US6599893B2 (en) * | 2000-08-29 | 2003-07-29 | Essential Therapeutics, Inc. | Cephalosporin antibiotics and prodrugs thereof |
AU2001245902B2 (en) * | 2000-09-21 | 2007-08-23 | Trine Pharmaceuticals, Inc. | Prodrugs of a 7-acylamino-3-heteroarylthio-3-cephem carboxylic acid antibiotic |
AU2002234148A1 (en) | 2000-12-29 | 2002-07-16 | Bellsouth Intellectual Property Corporation | Web based messaging system with personalized caller specific messages |
US7119062B1 (en) | 2001-02-23 | 2006-10-10 | Neucoll, Inc. | Methods and compositions for improved articular surgery using collagen |
US6608196B2 (en) | 2001-05-03 | 2003-08-19 | Galileo Pharmaceuticals, Inc. | Process for solid supported synthesis of pyruvate-derived compounds |
ATE408593T1 (de) | 2001-05-03 | 2008-10-15 | Galileo Lab Inc | Pyruvatderivate |
KR20030071311A (ko) * | 2002-02-28 | 2003-09-03 | 주식회사 엘지생명과학 | 신규 세팔로스포린 화합물 및 그의 제조방법 |
AU2003240545A1 (en) * | 2002-06-06 | 2003-12-22 | Therapeutics Corporation Genome | Use of ramoplanin to treat diseases associated with the use of antibiotics |
AU2003274927A1 (en) * | 2002-08-23 | 2004-03-11 | Genome Therapeutics Corporation | Methods and reagents for preventing bacteremias |
US20050043223A1 (en) * | 2003-04-25 | 2005-02-24 | Leach Timothy S. | Methods for reducing or preventing transmission of nosocomial pathogens in a health care facility |
CN107531660A (zh) | 2015-03-13 | 2018-01-02 | 福马治疗股份有限公司 | 作为HDAC8抑制剂的α‑肉桂酰胺化合物和组合物 |
KR102408800B1 (ko) | 2016-03-07 | 2022-06-13 | 머크 샤프 앤드 돔 코포레이션 | 비시클릭 아릴 모노박탐 화합물 및 박테리아 감염의 치료를 위한 그의 사용 방법 |
CN114671892B (zh) * | 2022-04-24 | 2023-04-11 | 江苏海洋大学 | 含7-氨基头孢烷酸的1,3,4-噻二唑衍生物及制法与用途 |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CH605997A5 (es) * | 1974-08-30 | 1978-10-13 | Ciba Geigy Ag | |
US3992377A (en) * | 1974-12-13 | 1976-11-16 | Eli Lilly And Company | 3-Thio-substituted cephalosporin antibiotics |
FR2457297A1 (fr) * | 1979-05-23 | 1980-12-19 | Rhone Poulenc Ind | Nouvelles vinyl-3 cephalosporines, et leur preparation |
FI801640A (fi) * | 1979-05-23 | 1980-11-24 | Rhone Poulenc Ind | Nya tiovinyl-3 kefalosporiner deras framstaellning och dessa innehaollande kompositioner |
FR2494274A2 (fr) * | 1980-11-20 | 1982-05-21 | Rhone Poulenc Ind | Nouvelles thiovinyl-3 cephalosporines, leur preparation et les medicaments qui les contiennent |
GR79043B (es) * | 1982-12-06 | 1984-10-02 | Fujisawa Pharmaceutical Co | |
US4870168A (en) * | 1987-02-26 | 1989-09-26 | Bristol-Myers Company | 3-Unsaturated alkyl cephems from 3-triflyl cephems |
US5025006A (en) * | 1990-06-26 | 1991-06-18 | Merck & Co., Inc. | 2-biphenyl-carbapenem antibacterial agents |
US5077287A (en) * | 1991-01-18 | 1991-12-31 | Eli Lilly And Company | 3-thiazolylthio carbacephem antibacterial agents |
JPH05132488A (ja) * | 1991-08-13 | 1993-05-28 | Meiji Seika Kaisha Ltd | 新規セフアロスポリン誘導体 |
TW427993B (en) * | 1993-09-09 | 2001-04-01 | Fujisawa Pharmaceutical Co | New cephem compounds |
EP0754184A1 (en) * | 1994-04-01 | 1997-01-22 | Microcide Pharmaceuticals, Inc. | Cephalosporin antibiotics |
-
1996
- 1996-10-08 MY MYPI96004152A patent/MY127641A/en unknown
- 1996-10-11 CN CNB001268856A patent/CN1183142C/zh not_active Expired - Fee Related
- 1996-10-11 ZA ZA9608617A patent/ZA968617B/xx unknown
- 1996-10-11 CA CA002234255A patent/CA2234255A1/en not_active Abandoned
- 1996-10-11 WO PCT/US1996/016349 patent/WO1997013772A2/en not_active Application Discontinuation
- 1996-10-11 NZ NZ321135A patent/NZ321135A/xx unknown
- 1996-10-11 ES ES96936406T patent/ES2164924T3/es not_active Expired - Lifetime
- 1996-10-11 RO RO98-00860A patent/RO119830B1/ro unknown
- 1996-10-11 CZ CZ981089A patent/CZ108998A3/cs unknown
- 1996-10-11 US US08/728,233 patent/US6057312A/en not_active Expired - Fee Related
- 1996-10-11 US US08/730,040 patent/US5859256A/en not_active Expired - Fee Related
- 1996-10-11 JP JP9515245A patent/JPH11513670A/ja not_active Ceased
- 1996-10-11 KR KR10-2004-7002598A patent/KR100491466B1/ko not_active IP Right Cessation
- 1996-10-11 KR KR10-1998-0702687A patent/KR100455544B1/ko not_active IP Right Cessation
- 1996-10-11 BR BR9611062A patent/BR9611062A/pt not_active Application Discontinuation
- 1996-10-11 AR ARP960104714A patent/AR005642A1/es not_active Application Discontinuation
- 1996-10-11 US US08/728,232 patent/US6066630A/en not_active Expired - Fee Related
- 1996-10-11 PT PT96936406T patent/PT874854E/pt unknown
- 1996-10-11 HU HU9802545A patent/HUP9802545A3/hu unknown
- 1996-10-11 US US08/730,042 patent/US6087355A/en not_active Expired - Fee Related
- 1996-10-11 EP EP96936406A patent/EP0874854B1/en not_active Expired - Lifetime
- 1996-10-11 DK DK96936406T patent/DK0874854T3/da active
- 1996-10-11 AU AU74417/96A patent/AU708676B2/en not_active Ceased
- 1996-10-11 AT AT96936406T patent/ATE210666T1/de not_active IP Right Cessation
- 1996-10-11 PL PL326150A patent/PL192069B1/pl unknown
- 1996-10-11 DE DE69618015T patent/DE69618015T2/de not_active Expired - Fee Related
- 1996-10-11 SK SK464-98A patent/SK283524B6/sk unknown
- 1996-10-11 CN CN96198934A patent/CN1066735C/zh not_active Expired - Fee Related
- 1996-10-15 TW TW085112602A patent/TW474935B/zh not_active IP Right Cessation
-
1998
- 1998-04-07 IL IL123983A patent/IL123983A/en not_active IP Right Cessation
- 1998-04-08 NO NO19981653A patent/NO323007B1/no unknown
- 1998-04-13 MX MX9802891A patent/MX9802891A/es not_active IP Right Cessation
-
1999
- 1999-06-24 HK HK99102717A patent/HK1017887A1/xx not_active IP Right Cessation
-
2000
- 2000-09-01 CN CNB001268775A patent/CN1179963C/zh not_active Expired - Fee Related
-
2001
- 2001-07-09 HK HK01104714A patent/HK1034191A1/xx not_active IP Right Cessation
- 2001-07-09 HK HK01104713A patent/HK1034248A1/xx not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
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FC | Refusal |