AP403A - N-t-butyl-androst-3,5-diene-17b-carboxyamide-3-carboxylic acid polymorph A. - Google Patents

N-t-butyl-androst-3,5-diene-17b-carboxyamide-3-carboxylic acid polymorph A. Download PDF

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Publication number
AP403A
AP403A APAP/P/1993/000497A AP9300497A AP403A AP 403 A AP403 A AP 403A AP 9300497 A AP9300497 A AP 9300497A AP 403 A AP403 A AP 403A
Authority
AP
ARIPO
Prior art keywords
polymorph
diene
androst
carboxylic acid
carboxamide
Prior art date
Application number
APAP/P/1993/000497A
Other languages
English (en)
Other versions
AP9300497A0 (en
Inventor
Neil Howard Baine
Neville Lewis Holder
Donald Nathaniel Kline
Robert Lee Webb
Gary Edward Zuber
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of AP9300497A0 publication Critical patent/AP9300497A0/xx
Application granted granted Critical
Publication of AP403A publication Critical patent/AP403A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
APAP/P/1993/000497A 1992-03-24 1993-03-18 N-t-butyl-androst-3,5-diene-17b-carboxyamide-3-carboxylic acid polymorph A. AP403A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929206413A GB9206413D0 (en) 1992-03-24 1992-03-24 N-t-butyl-androst-3,5-diene-17b-carboxamide-3-carboxylic acid polymorph a

Publications (2)

Publication Number Publication Date
AP9300497A0 AP9300497A0 (en) 1993-04-30
AP403A true AP403A (en) 1995-08-24

Family

ID=10712749

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1993/000497A AP403A (en) 1992-03-24 1993-03-18 N-t-butyl-androst-3,5-diene-17b-carboxyamide-3-carboxylic acid polymorph A.

Country Status (29)

Country Link
EP (1) EP0633892B1 (de)
JP (1) JP2736169B2 (de)
CN (1) CN1078723A (de)
AP (1) AP403A (de)
AT (1) ATE180490T1 (de)
AU (1) AU669522B2 (de)
BG (1) BG99062A (de)
BR (1) BR9306139A (de)
CA (1) CA2132535A1 (de)
CZ (1) CZ286266B6 (de)
DE (1) DE69325094T2 (de)
DK (1) DK0633892T3 (de)
ES (1) ES2134260T3 (de)
FI (1) FI114709B (de)
GB (1) GB9206413D0 (de)
GR (1) GR3030779T3 (de)
HU (1) HUT68120A (de)
IL (1) IL105102A (de)
MA (1) MA22841A1 (de)
MX (1) MX9301656A (de)
NO (1) NO943547D0 (de)
NZ (1) NZ252008A (de)
OA (1) OA10100A (de)
PL (1) PL172523B1 (de)
RU (1) RU94041839A (de)
SI (1) SI9300140A (de)
SK (1) SK113894A3 (de)
WO (1) WO1993019081A1 (de)
ZA (1) ZA932014B (de)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4910226A (en) * 1987-04-29 1990-03-20 Smithkline Beckman Corporation Steroid 5-alpha-reductase inhibitors
IL104602A (en) * 1992-02-07 1997-07-13 Smithkline Beecham Corp Process for the preparation of 3-carbonylandrostadiene- 17-carboxamides and intermediates for this process

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
Bioorganic Chemistry, 1989, METCALF et al. pp. 372-376 *
Journal of Steroid Biochemistry, 1989, LEVY et al. pp. 571-575 *

Also Published As

Publication number Publication date
FI944414A (fi) 1994-09-23
EP0633892B1 (de) 1999-05-26
ATE180490T1 (de) 1999-06-15
RU94041839A (ru) 1996-08-10
AP9300497A0 (en) 1993-04-30
ES2134260T3 (es) 1999-10-01
OA10100A (en) 1996-12-18
SI9300140A (en) 1993-09-30
DK0633892T3 (da) 2000-04-10
EP0633892A1 (de) 1995-01-18
IL105102A0 (en) 1994-08-26
BG99062A (en) 1995-08-28
NO943547L (no) 1994-09-23
ZA932014B (en) 1994-09-22
FI944414A0 (fi) 1994-09-23
EP0633892A4 (de) 1995-05-17
HUT68120A (en) 1995-05-29
NZ252008A (en) 1996-06-25
MX9301656A (es) 1994-02-28
JPH07505370A (ja) 1995-06-15
AU4044893A (en) 1993-10-21
DE69325094T2 (de) 1999-11-18
FI114709B (fi) 2004-12-15
IL105102A (en) 1997-02-18
DE69325094D1 (de) 1999-07-01
MA22841A1 (fr) 1993-10-01
WO1993019081A1 (en) 1993-09-30
NO943547D0 (no) 1994-09-23
AU669522B2 (en) 1996-06-13
CA2132535A1 (en) 1993-09-30
BR9306139A (pt) 1998-06-23
CZ231994A3 (en) 1995-01-18
GR3030779T3 (en) 1999-11-30
GB9206413D0 (en) 1992-05-06
JP2736169B2 (ja) 1998-04-02
SK113894A3 (en) 1995-04-12
HU9402740D0 (en) 1994-12-28
CZ286266B6 (cs) 2000-03-15
CN1078723A (zh) 1993-11-24
PL172523B1 (pl) 1997-10-31

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