AP2006003768A0 - TetraazabenzoÄeÜazulene derivatives and analogs tehereof - Google Patents

TetraazabenzoÄeÜazulene derivatives and analogs tehereof

Info

Publication number
AP2006003768A0
AP2006003768A0 AP2006003768A AP2006003768A AP2006003768A0 AP 2006003768 A0 AP2006003768 A0 AP 2006003768A0 AP 2006003768 A AP2006003768 A AP 2006003768A AP 2006003768 A AP2006003768 A AP 2006003768A AP 2006003768 A0 AP2006003768 A0 AP 2006003768A0
Authority
AP
ARIPO
Prior art keywords
tetraazabenzoäeüazulene
tehereof
analogs
derivatives
tetraazabenzoäeüazulene derivatives
Prior art date
Application number
AP2006003768A
Other languages
English (en)
Inventor
Kimberly O'keefe Cameron
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of AP2006003768A0 publication Critical patent/AP2006003768A0/xx

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
AP2006003768A 2004-05-25 2005-05-13 TetraazabenzoÄeÜazulene derivatives and analogs tehereof AP2006003768A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US57403304P 2004-05-25 2004-05-25
PCT/IB2005/001469 WO2005116034A1 (fr) 2004-05-25 2005-05-13 Derives de tetraazabenzo[e]azulene et analogues de ceux-ci

Publications (1)

Publication Number Publication Date
AP2006003768A0 true AP2006003768A0 (en) 2006-10-31

Family

ID=34967684

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2006003768A AP2006003768A0 (en) 2004-05-25 2005-05-13 TetraazabenzoÄeÜazulene derivatives and analogs tehereof

Country Status (26)

Country Link
US (2) US7265104B2 (fr)
EP (1) EP1753766A1 (fr)
JP (1) JP4069159B2 (fr)
CN (1) CN1950374A (fr)
AP (1) AP2006003768A0 (fr)
AR (1) AR049187A1 (fr)
AU (1) AU2005247693A1 (fr)
BR (1) BRPI0510273A (fr)
CA (1) CA2568056A1 (fr)
CR (1) CR8753A (fr)
EA (1) EA010888B1 (fr)
EC (1) ECSP067025A (fr)
GE (1) GEP20094723B (fr)
GT (1) GT200500119A (fr)
IL (1) IL178220A0 (fr)
MA (1) MA28605B1 (fr)
NL (1) NL1029105C2 (fr)
NO (1) NO20064288L (fr)
PA (1) PA8634101A1 (fr)
PE (1) PE20060363A1 (fr)
SV (1) SV2006002127A (fr)
TN (1) TNSN06386A1 (fr)
TW (1) TWI297688B (fr)
UA (1) UA84208C2 (fr)
UY (1) UY28915A1 (fr)
WO (1) WO2005116034A1 (fr)

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US20050267100A1 (en) 2005-12-01
TNSN06386A1 (fr) 2008-02-22
JP2008500326A (ja) 2008-01-10
PA8634101A1 (es) 2006-06-02
NL1029105C2 (nl) 2006-06-13
EA010888B1 (ru) 2008-12-30
NO20064288L (no) 2006-10-23
BRPI0510273A (pt) 2007-10-30
IL178220A0 (en) 2006-12-31
AU2005247693A1 (en) 2005-12-08
EA200601773A1 (ru) 2007-06-29
CN1950374A (zh) 2007-04-18
AR049187A1 (es) 2006-07-05
US7358242B2 (en) 2008-04-15
TWI297688B (en) 2008-06-11
PE20060363A1 (es) 2006-05-08
SV2006002127A (es) 2006-02-15
UY28915A1 (es) 2005-12-30
UA84208C2 (en) 2008-09-25
CA2568056A1 (fr) 2005-12-08
TW200609235A (en) 2006-03-16
US7265104B2 (en) 2007-09-04
EP1753766A1 (fr) 2007-02-21
CR8753A (es) 2006-12-13
GT200500119A (es) 2006-01-12
WO2005116034A1 (fr) 2005-12-08
MA28605B1 (fr) 2007-05-02
ECSP067025A (es) 2006-12-29
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JP4069159B2 (ja) 2008-04-02
US20070265193A1 (en) 2007-11-15

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