ZA9810993B - A process for the preparation of ring-opened epothilone intermediates which are useful for the preparation of epothilone analogs. - Google Patents

A process for the preparation of ring-opened epothilone intermediates which are useful for the preparation of epothilone analogs.

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Publication number
ZA9810993B
ZA9810993B ZA9810993A ZA9810993A ZA9810993B ZA 9810993 B ZA9810993 B ZA 9810993B ZA 9810993 A ZA9810993 A ZA 9810993A ZA 9810993 A ZA9810993 A ZA 9810993A ZA 9810993 B ZA9810993 B ZA 9810993B
Authority
ZA
South Africa
Prior art keywords
preparation
epothilone
useful
ring
intermediates
Prior art date
Application number
ZA9810993A
Other languages
English (en)
Inventor
Soong-Hoon Kim
Robert M Borzilleri
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ZA9810993B publication Critical patent/ZA9810993B/xx

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    • C07D303/02—Compounds containing oxirane rings
    • C07D303/38—Compounds containing oxirane rings with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

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ZA9810993A 1997-12-04 1998-12-01 A process for the preparation of ring-opened epothilone intermediates which are useful for the preparation of epothilone analogs. ZA9810993B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6755097P 1997-12-04 1997-12-04

Publications (1)

Publication Number Publication Date
ZA9810993B true ZA9810993B (en) 2000-06-01

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ID=22076753

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Application Number Title Priority Date Filing Date
ZA9810993A ZA9810993B (en) 1997-12-04 1998-12-01 A process for the preparation of ring-opened epothilone intermediates which are useful for the preparation of epothilone analogs.

Country Status (10)

Country Link
US (1) US6365749B1 (xx)
EP (1) EP1035824A4 (xx)
JP (1) JP2003522722A (xx)
AR (1) AR017808A1 (xx)
AU (1) AU739380B2 (xx)
CA (1) CA2312098C (xx)
PE (1) PE134099A1 (xx)
UY (1) UY25279A1 (xx)
WO (1) WO1999027890A2 (xx)
ZA (1) ZA9810993B (xx)

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UY25279A1 (es) 1999-07-19
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