ZA857132B - Preparation of(threo)-1-aryl-2-acylamido-3-fluoro-1-propanols - Google Patents

Preparation of(threo)-1-aryl-2-acylamido-3-fluoro-1-propanols

Info

Publication number
ZA857132B
ZA857132B ZA857132A ZA857132A ZA857132B ZA 857132 B ZA857132 B ZA 857132B ZA 857132 A ZA857132 A ZA 857132A ZA 857132 A ZA857132 A ZA 857132A ZA 857132 B ZA857132 B ZA 857132B
Authority
ZA
South Africa
Prior art keywords
propanols
acylamido
threo
fluoro
aryl
Prior art date
Application number
ZA857132A
Other languages
English (en)
Inventor
Tattanahali Lakshm Nagabhushan
Stuart Walter Mccombie
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of ZA857132B publication Critical patent/ZA857132B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D301/00—Preparation of oxiranes
    • C07D301/02—Synthesis of the oxirane ring
    • C07D301/03—Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds
    • C07D301/14—Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds with organic peracids, or salts, anhydrides or esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/34—Compounds containing oxirane rings with hydrocarbon radicals, substituted by sulphur, selenium or tellurium atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
ZA857132A 1984-09-19 1985-09-17 Preparation of(threo)-1-aryl-2-acylamido-3-fluoro-1-propanols ZA857132B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/651,980 US4582918A (en) 1984-09-19 1984-09-19 Preparation of intermediates for (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols

Publications (1)

Publication Number Publication Date
ZA857132B true ZA857132B (en) 1986-05-28

Family

ID=24615030

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA857132A ZA857132B (en) 1984-09-19 1985-09-17 Preparation of(threo)-1-aryl-2-acylamido-3-fluoro-1-propanols

Country Status (18)

Country Link
US (1) US4582918A (fr)
EP (1) EP0200739B1 (fr)
JP (1) JPS62500519A (fr)
KR (1) KR900001509B1 (fr)
AR (1) AR245445A1 (fr)
AT (1) ATE44735T1 (fr)
AU (1) AU577622B2 (fr)
CA (1) CA1262553A (fr)
DE (1) DE3571613D1 (fr)
DK (1) DK173703B1 (fr)
ES (1) ES8702339A1 (fr)
HU (1) HU196198B (fr)
IE (1) IE58491B1 (fr)
IL (1) IL76432A (fr)
NZ (1) NZ213508A (fr)
SG (1) SG39092G (fr)
WO (1) WO1986001799A1 (fr)
ZA (1) ZA857132B (fr)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4973750A (en) * 1984-09-19 1990-11-27 Schering Corporation Preparation of (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols
DE3543021A1 (de) * 1985-12-05 1987-06-11 Boehringer Mannheim Gmbh Verbesserte verfahren zur herstellung von d-threo-1-(p-methylsulfonylphenyl) -2-dichloracetamido-propandiol-1,3-(thiamphenicol) sowie verwendung geeigneter zwischenprodukte
US5084583A (en) * 1989-10-12 1992-01-28 E. I. Du Pont De Nemours And Company Epoxidation of fluorine containing olefins
IT1249048B (it) 1991-02-21 1995-02-11 Zambon Spa Processo per la preparazione di trans-(5r)-2-ossazoline -2,4,5, trisostituite
US5346828A (en) * 1991-03-27 1994-09-13 Celgene Corporation Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenylpropionic acids using d-threonine aldolase
IL134144A (en) * 1999-02-19 2004-02-08 Akzo Nobel Nv Process for the preparation of a-droxy organic acids
EP1487785A2 (fr) * 2002-03-08 2004-12-22 Schering-Plough Ltd. Antibiotiques de type florfenicol
US20040202762A1 (en) * 2003-04-08 2004-10-14 Ducharme Paul E Smoked nonfibrous casing
US7126005B2 (en) 2003-10-06 2006-10-24 Aurobindo Pharma Limited Process for preparing florfenicol
PT1776109E (pt) * 2004-08-13 2009-03-25 Schering Plough Ltd Formulação farmacêutica que compreende um antibiótico, um triazol e um corticosteróide
BRPI0515917A (pt) 2004-09-23 2008-08-12 Schering Plough Ltd controle de parasitas em animais pelo uso de novos derivados de éter de oxima de trifluorometanossulfonanilida
JP4750126B2 (ja) * 2004-11-19 2011-08-17 シェーリング−プラウ・リミテッド 殺寄生虫薬２−フェニル−３−（１ｈ−ピロール−２−イル）アクリロニトリル誘導体の使用による動物における寄生虫の制御
PT1830885E (pt) * 2004-12-21 2008-12-22 Intervet Int Bv Composição veterinária injectável
AR054380A1 (es) * 2005-06-09 2007-06-20 Schering Plough Ltd Control de parasitos en animales con derivados de n- ((feniloxi) fenil) -1,1,1-trifluorometansulfonamida y de n-(fenilsulfanil) fenil) -1,1,1-trifluorometansulfonamida
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US7518017B2 (en) 2006-02-17 2009-04-14 Idexx Laboratories Fenicol compounds and methods synthesizing 2-trifluoroacetamido-3-substituted propiophenone compounds
MX2009006282A (es) * 2006-12-13 2009-06-23 Schering Plough Ltd Profarmacos solubles en agua de florfenicol y sus analogos.
US8044230B2 (en) * 2006-12-13 2011-10-25 Intervet Inc. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
US20090062397A1 (en) * 2007-04-27 2009-03-05 Schering-Plough Animal Health Corporation Compounds and methods for enhancing solubility of florfenicol and structurally-related antibiotics using cyclodextrins
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
ES2666187T3 (es) 2007-06-27 2018-05-03 E. I. Du Pont De Nemours And Company Procedimiento de control de plagas en animales
CN101909600A (zh) * 2007-11-09 2010-12-08 英特维特国际股份有限公司 速释固体制剂、其制备及其应用
TWI468407B (zh) 2008-02-06 2015-01-11 Du Pont 中離子農藥
EP2321269B1 (fr) * 2008-07-30 2018-09-19 Intervet International B.V. Procede de preparation de composes aminodiol d'oxazoline proteges utiles comme produits intermediaires dans la production de florfenicol
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
AU2010279587A1 (en) 2009-08-05 2012-02-09 E. I. Du Pont De Nemours And Company Mesoionic pesticides
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
EP2461684A2 (fr) 2009-08-05 2012-06-13 E. I. du Pont de Nemours and Company Pesticides mésoioniques
BRPI1002023A2 (pt) 2010-03-01 2011-10-25 Nanocore Biotecnologia S A forma farmacêutica sólida de dissolução rápida para tratamento de infecções bacterianas
MY156670A (en) 2010-05-27 2016-03-15 Du Pont Crystalline form of 4-[5-[3-chloro-5-(trifluoromethly)phenyl]-4,5-dihydro-5-(trifluoromethyl)-3-isoxazolyl]-n-[2-oxo-2-[(2,2,2-trifluoroethyl) amino]ethyl]-1-naphthalenecarboxamide
JP5716349B2 (ja) * 2010-10-22 2015-05-13 住友化学株式会社 エポキシアルコール化合物の取得方法、並びにエポキシアルコール化合物及びトリアゾール化合物の製造方法
WO2012087630A1 (fr) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Composés de pyridine et de pyrimidine utilisés pour lutter contre des nuisibles invertébrés
WO2013158422A1 (fr) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Composés hétérocycliques pour la lutte contre des animaux nuisibles invertébrés

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD83161A (fr) *
US3849482A (en) * 1967-10-30 1974-11-19 Merck & Co Inc Amine salts of cis-propenylphosphonic acid
LU79970A1 (fr) * 1978-07-13 1980-02-14 Continental Pharma Procede de preparation de derives de 1-phenyl-1-propanol
ES8104203A1 (es) * 1979-02-05 1981-04-16 Schering Corp Un procedimiento para la preparacion de un compuesto d-(treo-1-aril-2-acilamido-3-fluor-1-propanol
US4235892A (en) * 1979-02-05 1980-11-25 Schering Corporation, Patent Dept. 1-Aryl-2-acylamido-3-fluoro-1-propanols, methods for their use as antibacterial agents and compositions useful therefor

Also Published As

Publication number Publication date
IL76432A (en) 1989-02-28
DK224086D0 (da) 1986-05-14
AR245445A1 (es) 1994-01-31
HU196198B (en) 1988-10-28
EP0200739A1 (fr) 1986-11-12
AU4809785A (en) 1986-04-08
IE58491B1 (en) 1993-09-22
KR900001509B1 (ko) 1990-03-12
ES547083A0 (es) 1986-12-16
JPS62500519A (ja) 1987-03-05
DE3571613D1 (en) 1989-08-24
ES8702339A1 (es) 1986-12-16
CA1262553A (fr) 1989-10-31
DK173703B1 (da) 2001-07-09
IL76432A0 (en) 1986-01-31
WO1986001799A1 (fr) 1986-03-27
IE852296L (en) 1986-03-19
SG39092G (en) 1992-05-22
AU577622B2 (en) 1988-09-29
ATE44735T1 (de) 1989-08-15
EP0200739B1 (fr) 1989-07-19
KR870700614A (ko) 1987-12-30
US4582918A (en) 1986-04-15
NZ213508A (en) 1989-05-29
HUT45243A (en) 1988-06-28
JPH0529216B2 (fr) 1993-04-28
DK224086A (da) 1986-05-14

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