ZA200907099B - Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals - Google Patents

Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals

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Publication number
ZA200907099B
ZA200907099B ZA2009/07099A ZA200907099A ZA200907099B ZA 200907099 B ZA200907099 B ZA 200907099B ZA 2009/07099 A ZA2009/07099 A ZA 2009/07099A ZA 200907099 A ZA200907099 A ZA 200907099A ZA 200907099 B ZA200907099 B ZA 200907099B
Authority
ZA
South Africa
Prior art keywords
pharmaceuticals
production
receptor ligands
vanilloid receptor
novel vanilloid
Prior art date
Application number
ZA2009/07099A
Other languages
English (en)
Inventor
Robert Frank
Gregor Bahrenberg
Thomas Christoph
Klaus Schiene
Vry Jean De
Derek John Saunders
Bernd Sundermann
Jeewoo Lee
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE102007018149A external-priority patent/DE102007018149A1/de
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of ZA200907099B publication Critical patent/ZA200907099B/en

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    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D215/14—Radicals substituted by oxygen atoms
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ZA2009/07099A 2007-04-16 2009-10-12 Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals ZA200907099B (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE102007018149A DE102007018149A1 (de) 2007-04-16 2007-04-16 Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
US12/103,667 US8084484B2 (en) 2007-04-16 2008-04-15 Vanilloid receptor ligands, pharmaceutical compositions containing them, process for making them, and use thereof for treating pain and other conditions
EP2008002997 2008-04-15
PCT/EP2008/003027 WO2008125342A2 (de) 2007-04-16 2008-04-16 Vanilloid-rezeptor-liganden und ihre verwendung zur herstellung von arzneimitteln

Publications (1)

Publication Number Publication Date
ZA200907099B true ZA200907099B (en) 2013-03-27

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Application Number Title Priority Date Filing Date
ZA2009/07099A ZA200907099B (en) 2007-04-16 2009-10-12 Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals

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JP (1) JP2010523727A (ko)
KR (1) KR20100016593A (ko)
CN (1) CN101679370A (ko)
AU (1) AU2008238250B2 (ko)
BR (1) BRPI0810035A2 (ko)
CA (1) CA2683461A1 (ko)
CO (1) CO6241154A2 (ko)
EC (1) ECSP099692A (ko)
IL (1) IL201505A0 (ko)
MX (1) MX2009011149A (ko)
NZ (1) NZ580411A (ko)
RU (1) RU2498982C2 (ko)
WO (1) WO2008125342A2 (ko)
ZA (1) ZA200907099B (ko)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102007018149A1 (de) 2007-04-16 2008-10-23 Grünenthal GmbH Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
MX2011011797A (es) 2009-05-07 2011-11-29 Gruenenthal Gmbh Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides.
US8946204B2 (en) 2009-05-07 2015-02-03 Gruenenthal Gmbh Substituted phenylureas and phenylamides as vanilloid receptor ligands
MX2014000964A (es) 2011-07-26 2014-03-27 Gruenenthal Gmbh Derivados aza heterociclicos sustituidos.
BR112014001714A2 (pt) 2011-07-26 2017-02-14 Gruenenthal Gmbh derivados de carboxamida e ureia aromáticos bicíclicos substituídos como ligantes de receptor vaniloide
AR088701A1 (es) * 2011-11-09 2014-06-25 Gruenenthal Gmbh Derivados de carboxamida y urea basados en pirazolilo, sustituidos, que contienen una porcion fenilo sustituida con un grupo que contiene n como ligandos del receptor de vanilloide
AU2013230425B2 (en) * 2012-03-05 2017-05-25 Dr.Reddy's Laboratories Ltd. Substituted heterocyclic acetamides as kappa opioid receptor (kor) agonists
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