ZA200510298B - Pyrido[2,1-a]-isoquinoline derivatives as DPP-IV inhibitors - Google Patents
Pyrido[2,1-a]-isoquinoline derivatives as DPP-IV inhibitors Download PDFInfo
- Publication number
- ZA200510298B ZA200510298B ZA200510298A ZA200510298A ZA200510298B ZA 200510298 B ZA200510298 B ZA 200510298B ZA 200510298 A ZA200510298 A ZA 200510298A ZA 200510298 A ZA200510298 A ZA 200510298A ZA 200510298 B ZA200510298 B ZA 200510298B
- Authority
- ZA
- South Africa
- Prior art keywords
- pyrido
- dimethoxy
- hexahydro
- amino
- isoquinolin
- Prior art date
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- 108010067722 Dipeptidyl Peptidase 4 Proteins 0.000 title claims description 14
- 102100025012 Dipeptidyl peptidase 4 Human genes 0.000 title claims description 14
- 239000003112 inhibitor Substances 0.000 title description 5
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- NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical compound C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 claims description 4
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Classifications
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
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- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Public Health (AREA)
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- Urology & Nephrology (AREA)
- Emergency Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP03013404 | 2003-06-20 |
Publications (1)
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2011
- 2011-01-12 HR HR20110018T patent/HRP20110018T1/hr unknown
- 2011-01-27 CY CY20111100091T patent/CY1111425T1/el unknown
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