ZA200209484B - Arylmethylamine derivatives for use as tryptase inhibitors. - Google Patents

Arylmethylamine derivatives for use as tryptase inhibitors. Download PDF

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Publication number
ZA200209484B
ZA200209484B ZA200209484A ZA200209484A ZA200209484B ZA 200209484 B ZA200209484 B ZA 200209484B ZA 200209484 A ZA200209484 A ZA 200209484A ZA 200209484 A ZA200209484 A ZA 200209484A ZA 200209484 B ZA200209484 B ZA 200209484B
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South Africa
Prior art keywords
compound
phenyl
piperidin
aryl
heteroaryl
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ZA200209484A
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English (en)
Inventor
Peter C Astles
Olivier Houille
Heinz Pauls
Guyan Liang
James Pribish
Paul R Eastwood
Julian Levell
Mark Czekaj
Yong Gong
Kent Neuenschwander
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Aventis Pharma Inc
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Publication of ZA200209484B publication Critical patent/ZA200209484B/en

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ZA200209484A 2000-05-22 2002-11-21 Arylmethylamine derivatives for use as tryptase inhibitors. ZA200209484B (en)

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KR101182690B1 (ko) * 2004-03-02 2012-09-14 아벤티스 파마슈티칼스 인크. 트립타제 억제제의 제조방법
DOP2005000039A (es) * 2004-03-26 2005-10-31 Aventis Pharma Inc Hidrocloruro de [4-(5-aminometil-2-fluoro-fenil)- piperidin-1-il]-(4-bomo-3-metil-5-propoxi-tiofen-2-il)-metanona como un inhibidor de la triptasa de mastocitos
US7423176B2 (en) * 2004-04-13 2008-09-09 Cephalon, Inc. Bicyclic aromatic sulfinyl derivatives
EP1812071A2 (en) * 2004-10-13 2007-08-01 PTC Therapeutics, Inc. Compounds for nonsense suppression, use of these compounds for the manufacture of a medicament for treating somatic mutation-related diseases
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