YU15500A - Postupak za dobijanje cikličnih tioamida - Google Patents
Postupak za dobijanje cikličnih tioamidaInfo
- Publication number
- YU15500A YU15500A YU15500A YUP15500A YU15500A YU 15500 A YU15500 A YU 15500A YU 15500 A YU15500 A YU 15500A YU P15500 A YUP15500 A YU P15500A YU 15500 A YU15500 A YU 15500A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- cyclic thioamides
- preparation cyclic
- preparation
- preparing
- thioamides
- Prior art date
Links
- -1 cyclic thioamides Chemical class 0.000 title abstract 2
- QZAYGJVTTNCVMB-UHFFFAOYSA-N serotonin Chemical compound C1=C(O)C=C2C(CCN)=CNC2=C1 QZAYGJVTTNCVMB-UHFFFAOYSA-N 0.000 abstract 2
- 239000000556 agonist Substances 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000003949 imides Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 229940076279 serotonin Drugs 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C323/24—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/25—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/52—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
- C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Abstract
Ovaj pronalazak se odnosi na postupak za dobijanje jedinjenja formule gde b, Y i R3 su kako je gore definisano, korisnog za dobijanje novih aralkil i aralkiliden heterocikličnih laktama i imida koji su selektivni agonisti i antagonisti sereotonin 1 (5-HT1) receptora.[The present invention relates to a process for preparing a compound of the formula (I) wherewin b, Y and R3 are defined as above, useful for preparing novel aralkyl and aralkylidene heterocyclic lactams and imides which are selective agonists and antagonists of serotonin 1 (5 - HT1) receptors.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US12683199P | 1999-03-30 | 1999-03-30 |
Publications (1)
Publication Number | Publication Date |
---|---|
YU15500A true YU15500A (sh) | 2002-03-18 |
Family
ID=22426907
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
YU15500A YU15500A (sh) | 1999-03-30 | 2000-03-15 | Postupak za dobijanje cikličnih tioamida |
Country Status (26)
Country | Link |
---|---|
US (1) | US6388127B1 (sh) |
EP (1) | EP1041070B1 (sh) |
JP (1) | JP3566175B2 (sh) |
KR (1) | KR100386524B1 (sh) |
CN (2) | CN1163490C (sh) |
AR (1) | AR029744A1 (sh) |
AT (1) | ATE277025T1 (sh) |
AU (1) | AU777097B2 (sh) |
BR (1) | BR0001492A (sh) |
CA (1) | CA2302727C (sh) |
CZ (1) | CZ298140B6 (sh) |
DE (1) | DE60013942T2 (sh) |
DK (1) | DK1041070T3 (sh) |
ES (1) | ES2226715T3 (sh) |
HK (2) | HK1032053A1 (sh) |
HU (1) | HUP0001327A3 (sh) |
ID (1) | ID25428A (sh) |
IL (1) | IL135243A (sh) |
IN (1) | IN188844B (sh) |
PL (1) | PL196446B1 (sh) |
PT (1) | PT1041070E (sh) |
RU (1) | RU2219173C2 (sh) |
TR (1) | TR200000834A2 (sh) |
TW (1) | TW460472B (sh) |
YU (1) | YU15500A (sh) |
ZA (1) | ZA200001536B (sh) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
YU15500A (sh) * | 1999-03-30 | 2002-03-18 | Pfizer Products Inc. | Postupak za dobijanje cikličnih tioamida |
WO2014039715A1 (en) * | 2012-09-07 | 2014-03-13 | University Of Rochester | Methods and compositions for site-specific labeling of peptides and proteins |
US9999921B2 (en) | 2015-06-15 | 2018-06-19 | Gm Global Technology Operatioins Llc | Method of making aluminum or magnesium based composite engine blocks or other parts with in-situ formed reinforced phases through squeeze casting or semi-solid metal forming and post heat treatment |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2755278A (en) * | 1956-07-17 | Thiamori | ||
WO1994003652A1 (en) | 1992-07-31 | 1994-02-17 | Yokota Corporation Co., Ltd. | Method of making metal of high purity from scrap of worked metal |
GB9225377D0 (en) * | 1992-12-04 | 1993-01-27 | Ici Plc | Herbicides |
UA56185C2 (uk) * | 1996-09-30 | 2003-05-15 | Пфайзер Інк. | Аралкіл- та аралкіліденгетероциклічні лактами та іміди, фармацевтична композиція та спосіб лікування |
YU15500A (sh) * | 1999-03-30 | 2002-03-18 | Pfizer Products Inc. | Postupak za dobijanje cikličnih tioamida |
-
2000
- 2000-03-15 YU YU15500A patent/YU15500A/sh unknown
- 2000-03-15 DE DE60013942T patent/DE60013942T2/de not_active Expired - Fee Related
- 2000-03-15 AT AT00302110T patent/ATE277025T1/de not_active IP Right Cessation
- 2000-03-15 PT PT00302110T patent/PT1041070E/pt unknown
- 2000-03-15 ES ES00302110T patent/ES2226715T3/es not_active Expired - Lifetime
- 2000-03-15 EP EP00302110A patent/EP1041070B1/en not_active Expired - Lifetime
- 2000-03-15 DK DK00302110T patent/DK1041070T3/da active
- 2000-03-23 IL IL13524300A patent/IL135243A/xx not_active IP Right Cessation
- 2000-03-27 TW TW089105600A patent/TW460472B/zh not_active IP Right Cessation
- 2000-03-27 ID IDP20000242D patent/ID25428A/id unknown
- 2000-03-27 ZA ZA200001536A patent/ZA200001536B/xx unknown
- 2000-03-27 IN IN273MU2000 patent/IN188844B/en unknown
- 2000-03-28 US US09/536,576 patent/US6388127B1/en not_active Expired - Fee Related
- 2000-03-28 CA CA002302727A patent/CA2302727C/en not_active Expired - Fee Related
- 2000-03-28 AR ARP000101386A patent/AR029744A1/es unknown
- 2000-03-28 BR BR0001492-3A patent/BR0001492A/pt not_active IP Right Cessation
- 2000-03-28 AU AU22635/00A patent/AU777097B2/en not_active Ceased
- 2000-03-29 KR KR10-2000-0015986A patent/KR100386524B1/ko not_active IP Right Cessation
- 2000-03-29 HU HU0001327A patent/HUP0001327A3/hu unknown
- 2000-03-29 PL PL339287A patent/PL196446B1/pl unknown
- 2000-03-29 TR TR2000/00834A patent/TR200000834A2/xx unknown
- 2000-03-29 RU RU2000107951/04A patent/RU2219173C2/ru not_active IP Right Cessation
- 2000-03-29 JP JP2000090837A patent/JP3566175B2/ja not_active Expired - Fee Related
- 2000-03-29 CZ CZ20001142A patent/CZ298140B6/cs not_active IP Right Cessation
- 2000-03-30 CN CNB001048325A patent/CN1163490C/zh not_active Expired - Fee Related
- 2000-03-30 CN CNB2004100014528A patent/CN1290829C/zh not_active Expired - Fee Related
-
2001
- 2001-04-12 HK HK01102637A patent/HK1032053A1/xx not_active IP Right Cessation
-
2004
- 2004-09-17 HK HK04107139A patent/HK1064364A1/xx not_active IP Right Cessation
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