UY33151A - Pirrolidinonas heteroaromáticas fusionadas - Google Patents

Pirrolidinonas heteroaromáticas fusionadas

Info

Publication number
UY33151A
UY33151A UY33151A UY33151A UY33151A UY 33151 A UY33151 A UY 33151A UY 33151 A UY33151 A UY 33151A UY 33151 A UY33151 A UY 33151A UY 33151 A UY33151 A UY 33151A
Authority
UY
Uruguay
Prior art keywords
pirrolidinones
fusioned
heteroaromatic
heteroaromatic pirrolidinones
fusioned heteroaromatic
Prior art date
Application number
UY33151A
Other languages
English (en)
Spanish (es)
Inventor
Yasuyoshi Arikawa
Victoria Feher
Betty Lam
Zhe Nie
Qing Dong
Benjamin Jones
Christopher Smith
Masashi Takahashi
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43618073&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY33151(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of UY33151A publication Critical patent/UY33151A/es

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/527Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim spiro-condensed
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    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
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  • Diabetes (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
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  • Neurology (AREA)
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  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Transplantation (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Oncology (AREA)
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UY33151A 2009-12-23 2010-12-22 Pirrolidinonas heteroaromáticas fusionadas UY33151A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28996909P 2009-12-23 2009-12-23
US38696410P 2010-09-27 2010-09-27

Publications (1)

Publication Number Publication Date
UY33151A true UY33151A (es) 2011-07-29

Family

ID=43618073

Family Applications (1)

Application Number Title Priority Date Filing Date
UY33151A UY33151A (es) 2009-12-23 2010-12-22 Pirrolidinonas heteroaromáticas fusionadas

Country Status (42)

Country Link
US (7) US9181255B2 (OSRAM)
EP (4) EP2516434B1 (OSRAM)
JP (7) JP5658274B2 (OSRAM)
KR (1) KR101790255B1 (OSRAM)
CN (1) CN102753548B (OSRAM)
AR (1) AR081797A1 (OSRAM)
AU (1) AU2010333804B2 (OSRAM)
BR (1) BR112012015651B1 (OSRAM)
CA (1) CA2786950C (OSRAM)
CL (1) CL2012001745A1 (OSRAM)
CO (1) CO6592058A2 (OSRAM)
CR (1) CR20120392A (OSRAM)
CY (1) CY1116736T1 (OSRAM)
DK (1) DK2516434T3 (OSRAM)
DO (1) DOP2012000180A (OSRAM)
EA (1) EA021568B1 (OSRAM)
EC (1) ECSP12012057A (OSRAM)
ES (1) ES2545616T3 (OSRAM)
GE (1) GEP20156243B (OSRAM)
HR (1) HRP20150878T1 (OSRAM)
HU (1) HUE025177T2 (OSRAM)
IL (1) IL220509A (OSRAM)
JO (1) JO3108B1 (OSRAM)
MA (1) MA33909B1 (OSRAM)
ME (1) ME02186B (OSRAM)
MX (1) MX2012007402A (OSRAM)
MY (1) MY159257A (OSRAM)
NZ (1) NZ601267A (OSRAM)
PE (1) PE20130188A1 (OSRAM)
PH (1) PH12012501311A1 (OSRAM)
PL (1) PL2516434T3 (OSRAM)
PT (1) PT2516434E (OSRAM)
RS (1) RS54180B1 (OSRAM)
SG (1) SG181857A1 (OSRAM)
SI (1) SI2516434T1 (OSRAM)
SM (1) SMT201500199B (OSRAM)
TN (1) TN2012000316A1 (OSRAM)
TW (1) TWI457339B (OSRAM)
UA (1) UA107100C2 (OSRAM)
UY (1) UY33151A (OSRAM)
WO (1) WO2011079051A1 (OSRAM)
ZA (1) ZA201205428B (OSRAM)

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US9181255B2 (en) 2009-12-23 2015-11-10 Takeda Pharmaceutical Company Limited Fused heteroaromatic pyrrolidinones as SYK inhibitors
WO2012130780A1 (en) * 2011-03-28 2012-10-04 F. Hoffmann-La Roche Ag Thiazolopyrimidine compounds
WO2012177714A1 (en) 2011-06-22 2012-12-27 Takeda Pharmaceutical Company Limited Substituted 6-aza-isoindolin-1-one derivatives
WO2014051653A1 (en) 2012-09-27 2014-04-03 Portola Pharmaceuticals, Inc. Bicyclic dihydropyridone kinase inhibitors
US9469654B2 (en) 2012-09-27 2016-10-18 Portola Pharmaceuticals, Inc. Bicyclic oxa-lactam kinase inhibitors
HRP20181367T4 (hr) 2012-11-01 2021-11-26 Infinity Pharmaceuticals, Inc. Liječenje raka korištenjem modulatora izoforme pi3 kinaze
US20160024051A1 (en) 2013-03-15 2016-01-28 Infinity Pharmaceuticals, Inc. Salts and solid forms of isoquinolinones and composition comprising and methods of using the same
EP3003309B1 (en) 2013-05-30 2020-09-09 Infinity Pharmaceuticals, Inc. Treatment of cancers using pi3 kinase isoform modulators
US9376441B2 (en) 2013-07-31 2016-06-28 Gilead Sciences, Inc. Substituted pyrrolidines as SYK inhibitors
US9751888B2 (en) 2013-10-04 2017-09-05 Infinity Pharmaceuticals, Inc. Heterocyclic compounds and uses thereof
MX389256B (es) 2013-10-04 2025-03-20 Infinity Pharmaceuticals Inc Compuestos heterociclicos y usos de los mismos.
US20160244452A1 (en) 2013-10-21 2016-08-25 Infinity Pharmaceuticals, Inc. Heterocyclic compounds and uses thereof
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