UY29683A1 - Sales de 4-metil-n-(3-(4-metil-imidazol-1-il)-5-trifluorometil-fenil)-3-(4-piridin-3-il-pirimidin-2-ilamino)-benzamida - Google Patents

Sales de 4-metil-n-(3-(4-metil-imidazol-1-il)-5-trifluorometil-fenil)-3-(4-piridin-3-il-pirimidin-2-ilamino)-benzamida

Info

Publication number
UY29683A1
UY29683A1 UY29683A UY29683A UY29683A1 UY 29683 A1 UY29683 A1 UY 29683A1 UY 29683 A UY29683 A UY 29683A UY 29683 A UY29683 A UY 29683A UY 29683 A1 UY29683 A1 UY 29683A1
Authority
UY
Uruguay
Prior art keywords
methyl
imidazol
phenyl
salts
benzamida
Prior art date
Application number
UY29683A
Other languages
English (en)
Inventor
Paul W Manley
Wen-Chung Shieh
Paul Allen Sutton
Piotr H Karpinski
Raeann Wu
Stephanie Monnier
Jorg Brozio
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37398525&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY29683(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of UY29683A1 publication Critical patent/UY29683A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Se preparan sales de 4-metil-N-(3-(4-metil-imidazol-1-il)-5-trifluorometil-fenil)-3-(4-piridin-3-il-pirimidin-2-ilamino)-benzamida por diversos procesos
UY29683A 2005-07-20 2006-07-20 Sales de 4-metil-n-(3-(4-metil-imidazol-1-il)-5-trifluorometil-fenil)-3-(4-piridin-3-il-pirimidin-2-ilamino)-benzamida UY29683A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70140605P 2005-07-20 2005-07-20
US71621305P 2005-09-12 2005-09-12

Publications (1)

Publication Number Publication Date
UY29683A1 true UY29683A1 (es) 2007-02-28

Family

ID=37398525

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29683A UY29683A1 (es) 2005-07-20 2006-07-20 Sales de 4-metil-n-(3-(4-metil-imidazol-1-il)-5-trifluorometil-fenil)-3-(4-piridin-3-il-pirimidin-2-ilamino)-benzamida

Country Status (34)

Country Link
US (4) US8163904B2 (es)
EP (2) EP1910336B1 (es)
JP (1) JP5129132B2 (es)
KR (3) KR101755137B1 (es)
CN (1) CN102267981A (es)
AR (1) AR057467A1 (es)
AT (1) ATE514689T1 (es)
AU (1) AU2010241419C1 (es)
BR (1) BRPI0613605A2 (es)
CA (2) CA2615669C (es)
CY (1) CY1111772T1 (es)
DK (1) DK1910336T3 (es)
EC (1) ECSP088118A (es)
ES (1) ES2634291T3 (es)
GT (1) GT200600316A (es)
HK (1) HK1116778A1 (es)
HR (1) HRP20110639T1 (es)
IL (1) IL187787A (es)
JO (1) JO2757B1 (es)
MA (1) MA29686B1 (es)
MX (1) MX2008000892A (es)
MY (1) MY149889A (es)
NO (1) NO341313B1 (es)
NZ (2) NZ564182A (es)
PE (1) PE20070241A1 (es)
PL (1) PL1910336T3 (es)
PT (1) PT1910336E (es)
RU (4) RU2483065C2 (es)
SG (1) SG170772A1 (es)
SI (1) SI1910336T1 (es)
TN (1) TNSN08028A1 (es)
TW (1) TWI455934B (es)
UY (1) UY29683A1 (es)
WO (1) WO2007015871A1 (es)

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WO2013063000A1 (en) 2011-10-28 2013-05-02 Novartis Ag Method of treating gastrointestinal stromal tumors
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EP2779995A1 (en) 2011-11-14 2014-09-24 Novartis AG Immediate release 4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]-n-[5-(4-methyl- 1h-imidazol-1-yl)-3-(trifluoromethyl)phenyl]benzamide formulation
JP2015522070A (ja) 2012-07-11 2015-08-03 ノバルティス アーゲー 消化管間質腫瘍を治療する方法
WO2014059518A1 (en) * 2012-10-15 2014-04-24 Apotex Technologies Inc. Solid forms of nilotinib hydrochloride
AU2013333953B2 (en) * 2012-10-19 2017-08-31 Basf Se Multicomponent crystalline system comprising nilotinib and selected co-crystal formers
EP2792360A1 (en) 2013-04-18 2014-10-22 IP Gesellschaft für Management mbH (1aR,12bS)-8-cyclohexyl-11-fluoro-N-((1-methylcyclopropyl)sulfonyl)-1a-((3-methyl-3,8-diazabicyclo[3.2.1]oct-8-yl)carbonyl)-1,1a,2,2b-tetrahydrocyclopropa[d]indolo[2,1-a][2]benzazepine-5-carboxamide for use in treating HCV
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RU2551359C9 (ru) * 2013-11-28 2021-08-20 Общество с ограниченной ответственностью "Мамонт Фарм" Наноразмерная слабо закристаллизованная модификация 4-метил-N-[3-(4-метилимидазол-1-ил)-5-(трифторметил)фенил]-3-[(4-пиридин-3-илпиримидин-2-ил)амино]бензамида гидрохлорида моногидрата, способ ее получения и фармацевтическая композиция на ее основе
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EP3177610A4 (en) 2014-08-08 2018-01-10 Dr. Reddy's Laboratories Ltd. Process for the preparation of polymorphic forms of nilotinib
RS63029B1 (sr) 2014-08-11 2022-04-29 Sun Pharmaceutical Ind Ltd Nove soli nilotiniba i njihovi polimorfi
EP3271351A1 (en) 2015-03-20 2018-01-24 Cipla Limited Novel polymorphic form x of nilotinib dihydrochloride hydrate
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WO2017149550A1 (en) * 2016-03-02 2017-09-08 Msn Laboratories Private Limited Amorphous form of 4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]-benzamide
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TWI770624B (zh) 2018-06-15 2022-07-11 漢達生技醫藥股份有限公司 尼洛替尼十二烷基硫酸鹽在製備用於治療慢性骨髓性白血病之劑型的用途
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CN113573712A (zh) * 2019-02-18 2021-10-29 斯莱班克制药有限责任公司 尼洛替尼的药物组合物
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Also Published As

Publication number Publication date
CY1111772T1 (el) 2015-10-07
SI1910336T1 (sl) 2011-10-28
ATE514689T1 (de) 2011-07-15
RU2013101749A (ru) 2014-07-27
JO2757B1 (en) 2014-03-15
US20130137712A1 (en) 2013-05-30
JP2009502796A (ja) 2009-01-29
RU2434864C2 (ru) 2011-11-27
RU2605551C2 (ru) 2016-12-20
EP1910336B1 (en) 2011-06-29
NZ564182A (en) 2011-03-31
ES2634291T3 (es) 2017-09-27
TWI455934B (zh) 2014-10-11
HRP20110639T1 (hr) 2011-10-31
NO341313B1 (no) 2017-10-09
PT1910336E (pt) 2011-09-05
RU2008105827A (ru) 2009-08-27
RU2011120363A (ru) 2012-11-27
MX2008000892A (es) 2008-03-18
NZ591142A (en) 2012-09-28
ECSP088118A (es) 2008-02-20
RU2509767C1 (ru) 2014-03-20
AU2010241419B2 (en) 2012-03-29
WO2007015871A1 (en) 2007-02-08
AU2006276205A1 (en) 2007-02-08
US20080200487A1 (en) 2008-08-21
SG170772A1 (en) 2011-05-30
KR101755137B1 (ko) 2017-07-06
CA2615669A1 (en) 2007-02-08
GT200600316A (es) 2007-04-02
AR057467A1 (es) 2007-12-05
EP2186808A1 (en) 2010-05-19
EP2186808B1 (en) 2017-04-19
AU2010241419C1 (en) 2024-05-23
CN102267981A (zh) 2011-12-07
KR20140047737A (ko) 2014-04-22
CA2615669C (en) 2013-11-12
US8163904B2 (en) 2012-04-24
IL187787A (en) 2012-07-31
PE20070241A1 (es) 2007-03-22
KR20080027855A (ko) 2008-03-28
BRPI0613605A2 (pt) 2011-01-18
MA29686B1 (fr) 2008-08-01
RU2483065C2 (ru) 2013-05-27
US8389537B2 (en) 2013-03-05
CA2823946C (en) 2015-12-29
KR20150100946A (ko) 2015-09-02
DK1910336T3 (da) 2011-10-03
JP5129132B2 (ja) 2013-01-23
AU2010241419A1 (en) 2010-12-02
CA2823946A1 (en) 2007-02-08
NO20080897L (no) 2008-02-20
AU2006276205B2 (en) 2010-08-19
US20140038994A1 (en) 2014-02-06
TW200800950A (en) 2008-01-01
US20120270891A1 (en) 2012-10-25
HK1116778A1 (es) 2009-01-02
PL1910336T3 (pl) 2011-11-30
EP1910336A1 (en) 2008-04-16
US8580806B2 (en) 2013-11-12
MY149889A (en) 2013-10-31
US9163005B2 (en) 2015-10-20
TNSN08028A1 (en) 2009-07-14
IL187787A0 (en) 2008-08-07

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