UA77757C2 - Heterocyclic tripeptides as hepatitis c virus inhibitors - Google Patents
Heterocyclic tripeptides as hepatitis c virus inhibitors Download PDFInfo
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- UA77757C2 UA77757C2 UA20040807171A UA20040807171A UA77757C2 UA 77757 C2 UA77757 C2 UA 77757C2 UA 20040807171 A UA20040807171 A UA 20040807171A UA 20040807171 A UA20040807171 A UA 20040807171A UA 77757 C2 UA77757 C2 UA 77757C2
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0808—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms, e.g. Val, Ile, Leu
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Gastroenterology & Hepatology (AREA)
- Epidemiology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA002369970A CA2369970A1 (en) | 2002-02-01 | 2002-02-01 | Hepatitis c inhibitor tri-peptides |
PCT/CA2003/000091 WO2003064416A1 (en) | 2002-02-01 | 2003-01-24 | Heterocyclic tripeptides as hepatitis c inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
UA77757C2 true UA77757C2 (en) | 2007-01-15 |
Family
ID=27626567
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UA20040807171A UA77757C2 (en) | 2002-02-01 | 2003-01-24 | Heterocyclic tripeptides as hepatitis c virus inhibitors |
Country Status (30)
Country | Link |
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US (1) | US20030191067A1 (no) |
EP (1) | EP1474423B1 (no) |
JP (1) | JP4073872B2 (no) |
KR (1) | KR20040081167A (no) |
CN (1) | CN1304416C (no) |
AR (1) | AR038382A1 (no) |
AT (1) | ATE369364T1 (no) |
AU (1) | AU2003202348B2 (no) |
BR (1) | BR0307517A (no) |
CA (1) | CA2369970A1 (no) |
CO (1) | CO5611112A2 (no) |
DE (1) | DE60315420T2 (no) |
EA (1) | EA007739B1 (no) |
EC (1) | ECSP045224A (no) |
ES (1) | ES2290425T3 (no) |
HK (1) | HK1078870A1 (no) |
HR (1) | HRP20040696A2 (no) |
MX (1) | MXPA04007446A (no) |
MY (1) | MY133719A (no) |
NO (1) | NO326421B1 (no) |
NZ (1) | NZ534730A (no) |
PE (1) | PE20030854A1 (no) |
PL (1) | PL371283A1 (no) |
RS (1) | RS67104A (no) |
SA (1) | SA03240006B1 (no) |
TW (1) | TWI274056B (no) |
UA (1) | UA77757C2 (no) |
UY (1) | UY27638A1 (no) |
WO (1) | WO2003064416A1 (no) |
ZA (1) | ZA200406014B (no) |
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WO2015103490A1 (en) | 2014-01-03 | 2015-07-09 | Abbvie, Inc. | Solid antiviral dosage forms |
US20170066779A1 (en) | 2014-03-05 | 2017-03-09 | Idenix Pharmaceuticals Llc | Solid forms of a flaviviridae virus inhibitor compound and salts thereof |
US20170135990A1 (en) | 2014-03-05 | 2017-05-18 | Idenix Pharmaceuticals Llc | Pharmaceutical compositions comprising a 5,5-fused heteroarylene flaviviridae inhibitor and their use for treating or preventing flaviviridae infection |
US20170066795A1 (en) | 2014-03-05 | 2017-03-09 | Idenix Pharmaceuticals Llc | Solid prodrug forms of 2'-chloro-2'-methyl uridine for hcv |
EP3131914B1 (en) | 2014-04-16 | 2023-05-10 | Idenix Pharmaceuticals LLC | 3'-substituted methyl or alkynyl nucleosides for the treatment of hcv |
RU2650610C1 (ru) * | 2017-02-28 | 2018-04-16 | Васильевич Иващенко Александр | Противовирусная композиция и способ ее применения |
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US6323180B1 (en) * | 1998-08-10 | 2001-11-27 | Boehringer Ingelheim (Canada) Ltd | Hepatitis C inhibitor tri-peptides |
UA74546C2 (en) * | 1999-04-06 | 2006-01-16 | Boehringer Ingelheim Ca Ltd | Macrocyclic peptides having activity relative to hepatitis c virus, a pharmaceutical composition and use of the pharmaceutical composition |
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2002
- 2002-02-01 CA CA002369970A patent/CA2369970A1/en not_active Abandoned
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2003
- 2003-01-24 CN CNB038061619A patent/CN1304416C/zh not_active Expired - Fee Related
- 2003-01-24 WO PCT/CA2003/000091 patent/WO2003064416A1/en active IP Right Grant
- 2003-01-24 AT AT03700745T patent/ATE369364T1/de active
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- 2003-01-24 PL PL03371283A patent/PL371283A1/xx not_active Application Discontinuation
- 2003-01-24 EP EP03700745A patent/EP1474423B1/en not_active Expired - Lifetime
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- 2003-01-24 ES ES03700745T patent/ES2290425T3/es not_active Expired - Lifetime
- 2003-01-24 DE DE60315420T patent/DE60315420T2/de not_active Expired - Lifetime
- 2003-01-24 UA UA20040807171A patent/UA77757C2/uk unknown
- 2003-01-24 JP JP2003564039A patent/JP4073872B2/ja not_active Expired - Fee Related
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- 2003-01-24 KR KR10-2004-7011888A patent/KR20040081167A/ko active IP Right Grant
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- 2003-01-24 AU AU2003202348A patent/AU2003202348B2/en not_active Ceased
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- 2003-01-31 UY UY27638A patent/UY27638A1/es not_active Application Discontinuation
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2004
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