UA129890C2 - ТІЄНО[3,2-b]ПІРИДИН-7-АМІНОВІ СПОЛУКИ ДЛЯ ЛІКУВАННЯ СІМЕЙНОЇ ДИЗАВТОНОМІЇ - Google Patents

ТІЄНО[3,2-b]ПІРИДИН-7-АМІНОВІ СПОЛУКИ ДЛЯ ЛІКУВАННЯ СІМЕЙНОЇ ДИЗАВТОНОМІЇ

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Publication number
UA129890C2
UA129890C2 UAA202105103A UAA202105103A UA129890C2 UA 129890 C2 UA129890 C2 UA 129890C2 UA A202105103 A UAA202105103 A UA A202105103A UA A202105103 A UAA202105103 A UA A202105103A UA 129890 C2 UA129890 C2 UA 129890C2
Authority
UA
Ukraine
Prior art keywords
chloro
methyl
amino
pyridin
amine
Prior art date
Application number
UAA202105103A
Other languages
English (en)
Ukrainian (uk)
Inventor
Наньцзин ЧЖАН
Майкл А. Арнольд
Амал Дакка
Ґарі Мітчелл Керп
Гари Митчелл Керп
Том Туан Луонґ
Том Туан Луонг
Джейна Наресімхен
Джэйна Наресимхен
Ніколай А. Наришкін
Николай А. Наришкин
Цзяши ВАН
Сяоянь Чжан
Original Assignee
ПіТіСі ТЕРАПЬЮТИКС, ІНК.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ПіТіСі ТЕРАПЬЮТИКС, ІНК. filed Critical ПіТіСі ТЕРАПЬЮТИКС, ІНК.
Publication of UA129890C2 publication Critical patent/UA129890C2/uk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
UAA202105103A 2019-02-13 2020-02-10 ТІЄНО[3,2-b]ПІРИДИН-7-АМІНОВІ СПОЛУКИ ДЛЯ ЛІКУВАННЯ СІМЕЙНОЇ ДИЗАВТОНОМІЇ UA129890C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201962805283P 2019-02-13 2019-02-13
PCT/US2020/017430 WO2020167628A1 (en) 2019-02-13 2020-02-10 Thioeno[3,2-b] pyridin-7-amine compounds for treating familial dysautonomia

Publications (1)

Publication Number Publication Date
UA129890C2 true UA129890C2 (uk) 2025-09-03

Family

ID=69960696

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA202105103A UA129890C2 (uk) 2019-02-13 2020-02-10 ТІЄНО[3,2-b]ПІРИДИН-7-АМІНОВІ СПОЛУКИ ДЛЯ ЛІКУВАННЯ СІМЕЙНОЇ ДИЗАВТОНОМІЇ

Country Status (17)

Country Link
US (1) US12384797B2 (enExample)
EP (1) EP3924049B1 (enExample)
JP (1) JP7587511B2 (enExample)
KR (1) KR102907028B1 (enExample)
CN (1) CN113795304A (enExample)
AU (1) AU2020222881C1 (enExample)
BR (1) BR112021015853A2 (enExample)
CA (1) CA3129067A1 (enExample)
CL (1) CL2021002137A1 (enExample)
CO (1) CO2021010598A2 (enExample)
EA (1) EA202192170A1 (enExample)
IL (1) IL285399B2 (enExample)
MX (1) MX2021009667A (enExample)
PE (1) PE20220139A1 (enExample)
SG (1) SG11202108519TA (enExample)
UA (1) UA129890C2 (enExample)
WO (1) WO2020167628A1 (enExample)

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Also Published As

Publication number Publication date
US20220135586A1 (en) 2022-05-05
AU2020222881B2 (en) 2025-07-10
EA202192170A1 (ru) 2021-11-15
PE20220139A1 (es) 2022-01-27
EP3924049B1 (en) 2026-08-12
BR112021015853A2 (pt) 2021-10-05
CA3129067A1 (en) 2020-08-20
CN113795304A (zh) 2021-12-14
US12384797B2 (en) 2025-08-12
AU2020222881C1 (en) 2026-01-22
IL285399B2 (en) 2025-06-01
MX2021009667A (es) 2021-12-10
AU2020222881A1 (en) 2021-09-09
WO2020167628A1 (en) 2020-08-20
KR20210137040A (ko) 2021-11-17
JP2022520822A (ja) 2022-04-01
CL2021002137A1 (es) 2022-02-25
IL285399A (en) 2021-09-30
KR102907028B1 (ko) 2026-01-05
SG11202108519TA (en) 2021-09-29
CO2021010598A2 (es) 2021-08-30
JP7587511B2 (ja) 2024-11-20
IL285399B1 (en) 2025-02-01
EP3924049A1 (en) 2021-12-22

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