UA127897C2 - Інгібітори аргінази - Google Patents

Інгібітори аргінази Download PDF

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Publication number
UA127897C2
UA127897C2 UAA202006325A UAA202006325A UA127897C2 UA 127897 C2 UA127897 C2 UA 127897C2 UA A202006325 A UAA202006325 A UA A202006325A UA A202006325 A UAA202006325 A UA A202006325A UA 127897 C2 UA127897 C2 UA 127897C2
Authority
UA
Ukraine
Prior art keywords
cancer
group
disease
pharmaceutically acceptable
agent
Prior art date
Application number
UAA202006325A
Other languages
English (en)
Ukrainian (uk)
Inventor
Корін Ніколь Фолі
Корин Николь Фоли
Ребекка Луїс Ґрейндж
Ребекка Луис Грейндж
Тезджан Ґуней
Тезджан Гуней
Ярослав Калісіак
Ярослав Калисиак
Ерік Томас Ньюкомб
Эрик Томас Ньюкомб
Анх Тху Тран
Original Assignee
Аркус Байосайєнсіз, Інк.
Аркус Байосайенсиз, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Аркус Байосайєнсіз, Інк., Аркус Байосайенсиз, Инк. filed Critical Аркус Байосайєнсіз, Інк.
Publication of UA127897C2 publication Critical patent/UA127897C2/uk

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/69—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/555—Heterocyclic compounds containing heavy metals, e.g. hemin, hematin, melarsoprol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00—Medicinal preparations containing inorganic active ingredients
    • A61K33/24—Heavy metals; Compounds thereof
    • A61K33/243—Platinum; Compounds thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
UAA202006325A 2018-03-05 2019-03-04 Інгібітори аргінази UA127897C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862638412P 2018-03-05 2018-03-05
PCT/US2019/020507 WO2019173188A1 (en) 2018-03-05 2019-03-04 Arginase inhibitors

Publications (1)

Publication Number Publication Date
UA127897C2 true UA127897C2 (uk) 2024-02-07

Family

ID=67847429

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA202006325A UA127897C2 (uk) 2018-03-05 2019-03-04 Інгібітори аргінази

Country Status (21)

Country Link
US (1) US12054500B2 (enExample)
EP (1) EP3761992A4 (enExample)
JP (1) JP7402167B2 (enExample)
KR (1) KR102656571B1 (enExample)
CN (1) CN111818928A (enExample)
AU (1) AU2019229978B2 (enExample)
BR (1) BR112020017604A2 (enExample)
CA (1) CA3091805A1 (enExample)
CL (1) CL2020002271A1 (enExample)
CO (1) CO2020012060A2 (enExample)
CR (1) CR20200445A (enExample)
EA (1) EA202092086A1 (enExample)
IL (1) IL276813B2 (enExample)
MX (1) MX2020009290A (enExample)
MY (1) MY205512A (enExample)
PE (1) PE20210452A1 (enExample)
PH (1) PH12020551352A1 (enExample)
SG (1) SG11202008113RA (enExample)
UA (1) UA127897C2 (enExample)
WO (1) WO2019173188A1 (enExample)
ZA (1) ZA202006006B (enExample)

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TW202325279A (zh) 2021-10-29 2023-07-01 美商阿克思生物科學有限公司 HIF-2α抑制劑及其使用方法
CN119156228A (zh) 2022-05-02 2024-12-17 艾库斯生物科学有限公司 抗tigit抗体及其用途
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Also Published As

Publication number Publication date
IL276813B2 (en) 2024-09-01
ZA202006006B (en) 2025-02-26
CO2020012060A2 (es) 2021-01-18
PE20210452A1 (es) 2021-03-08
CA3091805A1 (en) 2019-09-12
CL2020002271A1 (es) 2021-04-09
EP3761992A1 (en) 2021-01-13
JP2021516237A (ja) 2021-07-01
KR20200128117A (ko) 2020-11-11
AU2019229978A1 (en) 2020-10-15
MX2020009290A (es) 2020-09-28
CR20200445A (es) 2021-04-27
KR102656571B1 (ko) 2024-04-11
US12054500B2 (en) 2024-08-06
AU2019229978B2 (en) 2024-05-30
US20210002306A1 (en) 2021-01-07
MY205512A (en) 2024-10-24
CN111818928A (zh) 2020-10-23
WO2019173188A1 (en) 2019-09-12
JP7402167B2 (ja) 2023-12-20
IL276813A (en) 2020-10-29
EA202092086A1 (ru) 2021-02-09
SG11202008113RA (en) 2020-09-29
BR112020017604A2 (pt) 2020-12-22
IL276813B1 (en) 2024-05-01
PH12020551352A1 (en) 2021-06-21
EP3761992A4 (en) 2021-11-24

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