TWI731837B - 醫藥組合、包含該組合之醫藥組成物和套組以及該組合之用途 - Google Patents

醫藥組合、包含該組合之醫藥組成物和套組以及該組合之用途 Download PDF

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TWI731837B
TWI731837B TW104116781A TW104116781A TWI731837B TW I731837 B TWI731837 B TW I731837B TW 104116781 A TW104116781 A TW 104116781A TW 104116781 A TW104116781 A TW 104116781A TW I731837 B TWI731837 B TW I731837B
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combination
cancer
compound
formula
pharmaceutically acceptable
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TW104116781A
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Chinese (zh)
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TW201613577A (en
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湯瑪士 約爾格 梅林
恩里克 瑪麗亞 奧西奧
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盧森堡商歐陸斯迪公司
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
TW104116781A 2014-05-28 2015-05-26 醫藥組合、包含該組合之醫藥組成物和套組以及該組合之用途 TWI731837B (zh)

Applications Claiming Priority (2)

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GBGB1409485.8A GB201409485D0 (en) 2014-05-28 2014-05-28 Pharmaceutical composition
GB1409485.8 2014-05-28

Publications (2)

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TW201613577A TW201613577A (en) 2016-04-16
TWI731837B true TWI731837B (zh) 2021-07-01

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US (4) US10744120B2 (cg-RX-API-DMAC7.html)
EP (1) EP3148584B1 (cg-RX-API-DMAC7.html)
JP (2) JP2017518292A (cg-RX-API-DMAC7.html)
KR (1) KR20170008846A (cg-RX-API-DMAC7.html)
CN (1) CN106488776B (cg-RX-API-DMAC7.html)
AU (1) AU2015266053B2 (cg-RX-API-DMAC7.html)
BR (1) BR112016027043B1 (cg-RX-API-DMAC7.html)
CA (1) CA2950340C (cg-RX-API-DMAC7.html)
DK (1) DK3148584T3 (cg-RX-API-DMAC7.html)
EA (1) EA038323B1 (cg-RX-API-DMAC7.html)
ES (1) ES2885429T3 (cg-RX-API-DMAC7.html)
GB (1) GB201409485D0 (cg-RX-API-DMAC7.html)
IL (1) IL249230A0 (cg-RX-API-DMAC7.html)
MX (1) MX383254B (cg-RX-API-DMAC7.html)
PH (1) PH12016502352A1 (cg-RX-API-DMAC7.html)
SG (2) SG10201810404XA (cg-RX-API-DMAC7.html)
TW (1) TWI731837B (cg-RX-API-DMAC7.html)
UA (1) UA121392C2 (cg-RX-API-DMAC7.html)
WO (1) WO2015181157A1 (cg-RX-API-DMAC7.html)

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TWI573792B (zh) 2012-02-01 2017-03-11 歐陸斯迪公司 新穎治療劑
GB201409488D0 (en) 2014-05-28 2014-07-09 Euro Celtique Sa Pharmaceutical composition
GB201409485D0 (en) * 2014-05-28 2014-07-09 Euro Celtique Sa Pharmaceutical composition
GB201409471D0 (en) 2014-05-28 2014-07-09 Euro Celtique Sa Pharmaceutical composition
US11266631B2 (en) 2016-10-11 2022-03-08 Purdue Pharmaceutical Products L.P. Hodgkin lymphoma therapy
GB201709402D0 (en) 2017-06-13 2017-07-26 Euro Celtique Sa Compounds for treating t-pll
GB201709405D0 (en) 2017-06-13 2017-07-26 Euro Celtique Sa Compounds for treating ovarian cancer
GB201709406D0 (en) 2017-06-13 2017-07-26 Euro-Cletique S A Compounds for treating TNBC
GB201709403D0 (en) 2017-06-13 2017-07-26 Euro Celtique Sa Compounds for treating sarcoma
KR20210105380A (ko) * 2018-12-18 2021-08-26 먼디파머 인터내셔널 코포레이션 리미티드 다발성 골수종을 치료하기 위한 화합물

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Also Published As

Publication number Publication date
US10744120B2 (en) 2020-08-18
ES2885429T3 (es) 2021-12-13
IL249230A0 (en) 2017-02-28
GB201409485D0 (en) 2014-07-09
CA2950340A1 (en) 2015-12-03
US11541038B2 (en) 2023-01-03
SG11201609362YA (en) 2016-12-29
MX2016015437A (es) 2017-06-23
BR112016027043B1 (pt) 2023-01-31
US20230285363A1 (en) 2023-09-14
AU2015266053B2 (en) 2020-07-02
EA201692481A1 (ru) 2017-04-28
CN106488776A (zh) 2017-03-08
US20170296513A1 (en) 2017-10-19
WO2015181157A1 (en) 2015-12-03
CN106488776B (zh) 2021-01-22
PH12016502352A1 (en) 2017-02-13
EA038323B1 (ru) 2021-08-10
US20210059989A1 (en) 2021-03-04
CA2950340C (en) 2023-10-17
JP2017518292A (ja) 2017-07-06
MX383254B (es) 2025-03-13
AU2015266053A1 (en) 2016-11-17
UA121392C2 (uk) 2020-05-25
BR112016027043A2 (pt) 2017-08-15
US12064417B2 (en) 2024-08-20
TW201613577A (en) 2016-04-16
EP3148584B1 (en) 2021-05-26
BR112016027043A8 (pt) 2021-07-20
KR20170008846A (ko) 2017-01-24
SG10201810404XA (en) 2018-12-28
US20250049762A1 (en) 2025-02-13
JP2021046446A (ja) 2021-03-25
DK3148584T3 (da) 2021-08-30
EP3148584A1 (en) 2017-04-05

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