TWI599575B - 表現gip受體活性之胰高血糖素類似物 - Google Patents

表現gip受體活性之胰高血糖素類似物 Download PDF

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Publication number
TWI599575B
TWI599575B TW102121606A TW102121606A TWI599575B TW I599575 B TWI599575 B TW I599575B TW 102121606 A TW102121606 A TW 102121606A TW 102121606 A TW102121606 A TW 102121606A TW I599575 B TWI599575 B TW I599575B
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amino acid
peptide
acid
seq
group
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TW102121606A
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TW201402598A (zh
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理查D 迪瑪奇
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印第安納大學科技研究公司
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Zoology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Toxicology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
TW102121606A 2012-06-21 2013-06-18 表現gip受體活性之胰高血糖素類似物 TWI599575B (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261662868P 2012-06-21 2012-06-21
US201261716878P 2012-10-22 2012-10-22

Publications (2)

Publication Number Publication Date
TW201402598A TW201402598A (zh) 2014-01-16
TWI599575B true TWI599575B (zh) 2017-09-21

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TW102121606A TWI599575B (zh) 2012-06-21 2013-06-18 表現gip受體活性之胰高血糖素類似物

Country Status (13)

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US (1) US9340600B2 (cg-RX-API-DMAC10.html)
EP (1) EP2864351B1 (cg-RX-API-DMAC10.html)
JP (1) JP6311708B2 (cg-RX-API-DMAC10.html)
KR (1) KR20150023013A (cg-RX-API-DMAC10.html)
CN (1) CN104583232B (cg-RX-API-DMAC10.html)
AR (1) AR091477A1 (cg-RX-API-DMAC10.html)
CA (1) CA2877358A1 (cg-RX-API-DMAC10.html)
ES (1) ES2602486T3 (cg-RX-API-DMAC10.html)
HK (1) HK1209764A1 (cg-RX-API-DMAC10.html)
MX (1) MX2014015558A (cg-RX-API-DMAC10.html)
RU (1) RU2015101697A (cg-RX-API-DMAC10.html)
TW (1) TWI599575B (cg-RX-API-DMAC10.html)
WO (1) WO2013192129A1 (cg-RX-API-DMAC10.html)

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US20140011738A1 (en) 2014-01-09
US9340600B2 (en) 2016-05-17
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CA2877358A1 (en) 2013-12-27
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