TW301655B - - Google Patents
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- Publication number
- TW301655B TW301655B TW083104367A TW83104367A TW301655B TW 301655 B TW301655 B TW 301655B TW 083104367 A TW083104367 A TW 083104367A TW 83104367 A TW83104367 A TW 83104367A TW 301655 B TW301655 B TW 301655B
- Authority
- TW
- Taiwan
- Prior art keywords
- group
- compound
- page
- cns
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/54—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring
- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB939310091A GB9310091D0 (en) | 1993-05-17 | 1993-05-17 | New polypeptide compound and a process for preparation thereof |
GB939325269A GB9325269D0 (en) | 1993-12-10 | 1993-12-10 | New polypeptide compound and a process for preparation thereof |
Publications (1)
Publication Number | Publication Date |
---|---|
TW301655B true TW301655B (pt) | 1997-04-01 |
Family
ID=26302903
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW083104367A TW301655B (pt) | 1993-05-17 | 1994-05-14 |
Country Status (18)
Country | Link |
---|---|
US (2) | US5569646A (pt) |
EP (1) | EP0644199B1 (pt) |
JP (1) | JP3551469B2 (pt) |
KR (1) | KR100346489B1 (pt) |
CN (1) | CN1057306C (pt) |
AT (1) | ATE194846T1 (pt) |
AU (1) | AU681119B2 (pt) |
CA (1) | CA2123921A1 (pt) |
DE (1) | DE69425304T2 (pt) |
DK (1) | DK0644199T3 (pt) |
ES (1) | ES2148254T3 (pt) |
GR (1) | GR3034366T3 (pt) |
HU (1) | HUT68385A (pt) |
IL (1) | IL109615A (pt) |
PH (1) | PH30811A (pt) |
PT (1) | PT644199E (pt) |
RU (1) | RU2164230C2 (pt) |
TW (1) | TW301655B (pt) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5874403A (en) * | 1992-10-15 | 1999-02-23 | Merck & Co., Inc. | Amino acid conjugates of cyclohexapeptidyl amines |
US5948753A (en) * | 1993-05-04 | 1999-09-07 | Merck & Co., Inc. | Cyclohexapeptidyl propanolamine compounds |
US5854276A (en) * | 1995-06-29 | 1998-12-29 | Fujisawa Pharmaceutical Co., Ltd. | Substance WF16616, process for production thereof, and use thereof |
WO1997017365A1 (en) * | 1995-11-09 | 1997-05-15 | Merck & Co., Inc. | Cyclohexapeptidyl bisamine compound, compositions containing said compound and methods of use |
US6117641A (en) | 1996-04-11 | 2000-09-12 | Mitotix, Inc. | Assays and reagents for identifying anti-fungal agents and uses related thereto |
KR20000005397A (ko) | 1996-04-11 | 2000-01-25 | 맨수리 무잠밀 엠 | 항-진균제를확인하기위한검정방법및시약,및이의용도 |
US6727082B1 (en) | 1996-04-11 | 2004-04-27 | Gpc Biotech Inc. | Assays and reagents for identifying anti-fungal agents, and uses related thereto |
US5854212A (en) * | 1996-10-23 | 1998-12-29 | Merck & Co., Inc. | Cyclohexapeptidyl bisamine compound, compositions containing said compound and methods of use |
AUPO381496A0 (en) * | 1996-11-25 | 1996-12-19 | Fujisawa Pharmaceutical Co., Ltd. | New compound |
CN1240713C (zh) * | 1998-02-09 | 2006-02-08 | 藤泽药品工业株式会社 | 化合物 |
WO1999047551A1 (en) * | 1998-03-16 | 1999-09-23 | Fujisawa Pharmaceutical Co., Ltd. | Wf14573 or its salt, production thereof and use thereof |
DE69934683T2 (de) | 1998-04-23 | 2007-10-18 | Aventis Pharma Deutschland Gmbh | Verfahren zur reduzierung von echinocandin-peptiden zu deren c4-monodeoxyhomotyrosin analoga |
AU6408499A (en) * | 1998-10-05 | 2000-04-26 | Abbott Laboratories | Cyclic peptides as antifungal agents |
AUPP999799A0 (en) | 1999-04-27 | 1999-05-20 | Fujisawa Pharmaceutical Co., Ltd. | New compound |
FR2794747B1 (fr) * | 1999-06-09 | 2004-04-16 | Hoechst Marion Roussel Inc | Nouveaux derives de l'echinocandine, leur procede de preparation et leur application comme anti-fongiques |
TWI233805B (en) * | 1999-07-01 | 2005-06-11 | Fujisawa Pharmaceutical Co | Stabilized pharmaceutical composition in lyophilized form as antifungal agent |
AUPR362001A0 (en) * | 2001-03-08 | 2001-04-05 | Fujisawa Pharmaceutical Co., Ltd. | New compound |
CN101861330A (zh) * | 2007-10-29 | 2010-10-13 | 安斯泰来制药有限公司 | 多肽化合物 |
ES2634431T3 (es) * | 2009-03-16 | 2017-09-27 | The Governing Council Of The University Of Toronto | Moléculas de aminoácidos cíclicos y procedimientos de preparación de las mismas |
US8927801B2 (en) * | 2009-04-13 | 2015-01-06 | The Procter & Gamble Company | Absorbent articles comprising wetness indicators |
JP2014088326A (ja) * | 2011-02-22 | 2014-05-15 | Astellas Pharma Inc | ポリペプチド化合物 |
CN102512379B (zh) * | 2011-12-16 | 2017-03-08 | 深圳市健元医药科技有限公司 | 一种新型棘白菌素类抗真菌药物组合物及其制备方法 |
CN102627689B (zh) * | 2012-03-30 | 2014-08-06 | 上海天伟生物制药有限公司 | 一种环肽类化合物的水合物及其制备方法和用途 |
CN102786591B (zh) * | 2012-08-31 | 2014-03-12 | 哈尔滨工业大学 | 定向诱导合成金属硫蛋白的工艺 |
WO2017079820A1 (en) | 2015-11-11 | 2017-05-18 | Encycle Therapeutics, Inc. | CYCLIC PEPTIDES TARGETING α4β7 INTEGRIN |
JP7035044B2 (ja) | 2016-11-11 | 2022-03-14 | ジーランド ファーマ エー/エス | α4β7インテグリンを標的とする環状ペプチド多量体 |
CA3062385A1 (en) | 2017-05-10 | 2018-11-15 | Encycle Therapeutics, Inc. | Homodetic cyclic peptides targeting a4s7 1ntegrin |
CN112759627B (zh) * | 2021-03-12 | 2021-10-01 | 河南科技大学 | 一种抗白色念珠菌多肽及其应用 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5166135A (en) * | 1988-09-12 | 1992-11-24 | Merck & Company, Inc. | Method for the control of pneumocystis carinii |
GB8925593D0 (en) * | 1989-11-13 | 1990-01-04 | Fujisawa Pharmaceutical Co | Fr901379 substance and preparation thereof |
US5386009A (en) * | 1990-03-19 | 1995-01-31 | Merck & Co. Inc. | Lipopeptide derivatives |
US5330973A (en) * | 1990-03-19 | 1994-07-19 | Merck & Co., Inc. | Lipopeptide derivatives |
US5159059A (en) * | 1990-05-29 | 1992-10-27 | Merck & Co., Inc. | Process for reduction of certain cyclohexapeptide compounds |
FI912873A (fi) * | 1990-06-18 | 1991-12-19 | Fujisawa Pharmaceutical Co | Ny polypeptidfoerening och foerfarande foer dess framstaellning. |
WO1994009033A1 (en) * | 1992-10-16 | 1994-04-28 | Merck & Co., Inc. | An improved process for cyclohexapeptidyl bisamine compounds |
-
1994
- 1994-05-10 AU AU61994/94A patent/AU681119B2/en not_active Ceased
- 1994-05-10 IL IL10961594A patent/IL109615A/xx not_active IP Right Cessation
- 1994-05-12 DE DE69425304T patent/DE69425304T2/de not_active Expired - Fee Related
- 1994-05-12 PH PH48267A patent/PH30811A/en unknown
- 1994-05-12 EP EP94107406A patent/EP0644199B1/en not_active Expired - Lifetime
- 1994-05-12 DK DK94107406T patent/DK0644199T3/da active
- 1994-05-12 AT AT94107406T patent/ATE194846T1/de not_active IP Right Cessation
- 1994-05-12 PT PT94107406T patent/PT644199E/pt unknown
- 1994-05-12 ES ES94107406T patent/ES2148254T3/es not_active Expired - Lifetime
- 1994-05-14 TW TW083104367A patent/TW301655B/zh active
- 1994-05-16 HU HU9401515A patent/HUT68385A/hu not_active Application Discontinuation
- 1994-05-16 CN CN94105193A patent/CN1057306C/zh not_active Expired - Fee Related
- 1994-05-16 KR KR1019940010607A patent/KR100346489B1/ko not_active IP Right Cessation
- 1994-05-16 RU RU94016354/04A patent/RU2164230C2/ru not_active IP Right Cessation
- 1994-05-16 US US08/242,854 patent/US5569646A/en not_active Expired - Fee Related
- 1994-05-17 JP JP12697794A patent/JP3551469B2/ja not_active Expired - Fee Related
- 1994-05-17 CA CA002123921A patent/CA2123921A1/en not_active Abandoned
-
1996
- 1996-07-03 US US08/675,212 patent/US5693750A/en not_active Expired - Fee Related
-
2000
- 2000-09-08 GR GR20000402052T patent/GR3034366T3/el not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
KR100346489B1 (ko) | 2002-11-18 |
US5569646A (en) | 1996-10-29 |
DK0644199T3 (da) | 2000-09-18 |
ES2148254T3 (es) | 2000-10-16 |
EP0644199B1 (en) | 2000-07-19 |
AU6199494A (en) | 1994-11-24 |
CN1100104A (zh) | 1995-03-15 |
CN1057306C (zh) | 2000-10-11 |
US5693750A (en) | 1997-12-02 |
PH30811A (en) | 1997-10-17 |
IL109615A (en) | 2000-12-06 |
GR3034366T3 (en) | 2000-12-29 |
HUT68385A (en) | 1995-06-28 |
DE69425304D1 (de) | 2000-08-24 |
JPH06340693A (ja) | 1994-12-13 |
ATE194846T1 (de) | 2000-08-15 |
AU681119B2 (en) | 1997-08-21 |
DE69425304T2 (de) | 2000-12-21 |
CA2123921A1 (en) | 1994-11-18 |
PT644199E (pt) | 2001-01-31 |
JP3551469B2 (ja) | 2004-08-04 |
IL109615A0 (en) | 1994-08-26 |
RU2164230C2 (ru) | 2001-03-20 |
EP0644199A1 (en) | 1995-03-22 |
HU9401515D0 (en) | 1994-08-29 |
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