TW201919618A - 用於治療肉瘤的化合物 - Google Patents

用於治療肉瘤的化合物 Download PDF

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Publication number
TW201919618A
TW201919618A TW107120396A TW107120396A TW201919618A TW 201919618 A TW201919618 A TW 201919618A TW 107120396 A TW107120396 A TW 107120396A TW 107120396 A TW107120396 A TW 107120396A TW 201919618 A TW201919618 A TW 201919618A
Authority
TW
Taiwan
Prior art keywords
pharmaceutically acceptable
sarcoma
acceptable salt
patient
tinostamostatin
Prior art date
Application number
TW107120396A
Other languages
English (en)
Chinese (zh)
Inventor
湯瑪士 約爾格 梅林
Original Assignee
盧森堡商歐陸斯迪公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 盧森堡商歐陸斯迪公司 filed Critical 盧森堡商歐陸斯迪公司
Publication of TW201919618A publication Critical patent/TW201919618A/zh

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61NELECTROTHERAPY; MAGNETOTHERAPY; RADIATION THERAPY; ULTRASOUND THERAPY
    • A61N5/00Radiation therapy
    • A61N5/10X-ray therapy; Gamma-ray therapy; Particle-irradiation therapy
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Pathology (AREA)
  • Radiology & Medical Imaging (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
TW107120396A 2017-06-13 2018-06-13 用於治療肉瘤的化合物 TW201919618A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1709403.8A GB201709403D0 (en) 2017-06-13 2017-06-13 Compounds for treating sarcoma
??1709403.8 2017-06-13

Publications (1)

Publication Number Publication Date
TW201919618A true TW201919618A (zh) 2019-06-01

Family

ID=59358374

Family Applications (1)

Application Number Title Priority Date Filing Date
TW107120396A TW201919618A (zh) 2017-06-13 2018-06-13 用於治療肉瘤的化合物

Country Status (14)

Country Link
US (3) US11576899B2 (enExample)
EP (1) EP3638232B1 (enExample)
JP (1) JP2020523355A (enExample)
KR (1) KR20200014791A (enExample)
AR (1) AR112144A1 (enExample)
AU (1) AU2018285822B2 (enExample)
BR (1) BR112019026463A2 (enExample)
CA (1) CA3067065A1 (enExample)
ES (1) ES2970224T3 (enExample)
GB (1) GB201709403D0 (enExample)
IL (1) IL271020A (enExample)
MX (1) MX2019015212A (enExample)
TW (1) TW201919618A (enExample)
WO (1) WO2018229133A1 (enExample)

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GB201709406D0 (en) 2017-06-13 2017-07-26 Euro-Cletique S A Compounds for treating TNBC
WO2020128913A1 (en) 2018-12-18 2020-06-25 Mundipharma International Corporation Limited Compounds for treating multiple myeloma

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Also Published As

Publication number Publication date
US11576899B2 (en) 2023-02-14
WO2018229133A1 (en) 2018-12-20
AR112144A1 (es) 2019-09-25
AU2018285822B2 (en) 2024-01-04
MX2019015212A (es) 2020-08-17
JP2020523355A (ja) 2020-08-06
CA3067065A1 (en) 2018-12-20
AU2018285822A1 (en) 2019-12-19
US20200113870A1 (en) 2020-04-16
BR112019026463A2 (pt) 2020-07-14
US20230277507A1 (en) 2023-09-07
IL271020A (en) 2020-01-30
GB201709403D0 (en) 2017-07-26
ES2970224T3 (es) 2024-05-27
US20250375424A1 (en) 2025-12-11
KR20200014791A (ko) 2020-02-11
EP3638232B1 (en) 2023-12-13
EP3638232A1 (en) 2020-04-22
US12257237B2 (en) 2025-03-25
EP3638232C0 (en) 2023-12-13

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