TW201642843A - 他噴他多腸胃外給藥的穩定製劑 - Google Patents

他噴他多腸胃外給藥的穩定製劑 Download PDF

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Publication number
TW201642843A
TW201642843A TW105108920A TW105108920A TW201642843A TW 201642843 A TW201642843 A TW 201642843A TW 105108920 A TW105108920 A TW 105108920A TW 105108920 A TW105108920 A TW 105108920A TW 201642843 A TW201642843 A TW 201642843A
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TW
Taiwan
Prior art keywords
composition
tapentadol
composition according
conjugate
container
Prior art date
Application number
TW105108920A
Other languages
English (en)
Chinese (zh)
Inventor
馬克 席勒
黑梅瑞克 卡洛斯 梵
斯特凡妮 施特勞布
艾娃 沃爾斯特
烏爾力克 伯特蘭
烏爾里希 萊因霍爾德
Original Assignee
歌林達有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=55661386&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TW201642843(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 歌林達有限公司 filed Critical 歌林達有限公司
Publication of TW201642843A publication Critical patent/TW201642843A/zh

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
TW105108920A 2015-03-27 2016-03-23 他噴他多腸胃外給藥的穩定製劑 TW201642843A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP15161487 2015-03-27
EP15169730 2015-05-28

Publications (1)

Publication Number Publication Date
TW201642843A true TW201642843A (zh) 2016-12-16

Family

ID=55661386

Family Applications (1)

Application Number Title Priority Date Filing Date
TW105108920A TW201642843A (zh) 2015-03-27 2016-03-23 他噴他多腸胃外給藥的穩定製劑

Country Status (28)

Country Link
US (2) US20160279078A1 (de)
EP (2) EP3273953B1 (de)
JP (1) JP6923447B2 (de)
KR (1) KR20170132282A (de)
CN (1) CN107847471A (de)
AU (1) AU2016239772B2 (de)
BR (1) BR112017018569A2 (de)
CA (1) CA2979034A1 (de)
CL (1) CL2017002306A1 (de)
CO (1) CO2017009400A2 (de)
CY (1) CY1121371T1 (de)
DK (1) DK3273953T3 (de)
EA (1) EA036258B1 (de)
EC (1) ECSP17064188A (de)
ES (2) ES2822113T3 (de)
HK (1) HK1252705A1 (de)
HR (1) HRP20190231T1 (de)
HU (1) HUE042612T2 (de)
IL (1) IL254136A0 (de)
LT (1) LT3273953T (de)
MX (1) MX2017012312A (de)
PE (1) PE20171651A1 (de)
PL (1) PL3273953T3 (de)
PT (2) PT3479823T (de)
RS (1) RS58301B1 (de)
SI (1) SI3273953T1 (de)
TW (1) TW201642843A (de)
WO (1) WO2016156147A1 (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
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PT3479823T (pt) 2015-03-27 2020-09-29 Gruenenthal Gmbh Formulação estável para administração parentérica de tapentadol
MX2019003257A (es) 2016-09-23 2019-06-10 Gruenenthal Gmbh Formulacion estable para la administracion parenteral de tapentadol.
EP3585370A1 (de) 2017-02-23 2020-01-01 Grünenthal GmbH Tapentadol als lokalanästhetikum

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Also Published As

Publication number Publication date
BR112017018569A2 (pt) 2018-04-24
SI3273953T1 (sl) 2019-03-29
ES2710299T3 (es) 2019-04-24
PT3273953T (pt) 2019-04-01
CL2017002306A1 (es) 2018-03-23
DK3273953T3 (en) 2019-03-11
LT3273953T (lt) 2019-02-25
EA201792144A1 (ru) 2018-03-30
PE20171651A1 (es) 2017-11-13
AU2016239772B2 (en) 2021-05-13
EP3273953B1 (de) 2019-01-02
ECSP17064188A (es) 2018-03-31
KR20170132282A (ko) 2017-12-01
EA036258B1 (ru) 2020-10-20
AU2016239772A1 (en) 2017-09-14
EP3479823B1 (de) 2020-09-09
JP6923447B2 (ja) 2021-08-18
CY1121371T1 (el) 2020-05-29
US11013701B2 (en) 2021-05-25
ES2822113T3 (es) 2021-04-29
EP3273953A1 (de) 2018-01-31
WO2016156147A1 (en) 2016-10-06
MX2017012312A (es) 2018-01-18
RS58301B1 (sr) 2019-03-29
EP3479823A1 (de) 2019-05-08
PL3273953T3 (pl) 2019-07-31
HUE042612T2 (hu) 2019-07-29
JP2018509462A (ja) 2018-04-05
CA2979034A1 (en) 2016-10-06
US20160279078A1 (en) 2016-09-29
IL254136A0 (en) 2017-10-31
PT3479823T (pt) 2020-09-29
CO2017009400A2 (es) 2018-01-05
HK1252705A1 (zh) 2019-05-31
HRP20190231T1 (hr) 2019-04-05
CN107847471A (zh) 2018-03-27
US20180125800A1 (en) 2018-05-10

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