HRP20190231T1 - Stabilna formulacija za parenteralnu primjenu tapentadola - Google Patents

Stabilna formulacija za parenteralnu primjenu tapentadola

Info

Publication number
HRP20190231T1
HRP20190231T1 HRP20190231TT HRP20190231T HRP20190231T1 HR P20190231 T1 HRP20190231 T1 HR P20190231T1 HR P20190231T T HRP20190231T T HR P20190231TT HR P20190231 T HRP20190231 T HR P20190231T HR P20190231 T1 HRP20190231 T1 HR P20190231T1
Authority
HR
Croatia
Prior art keywords
tapentadol
parenteral administration
stable formulation
formulation
stable
Prior art date
Application number
HRP20190231TT
Other languages
English (en)
Inventor
Marc Schiller
Carlos Van Hemelrijck
Stefanie Straub
Eva Cornelia WULSTEN
Ulrike Bertram
Ulrich Reinhold
Original Assignee
Grünenthal GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=55661386&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20190231(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Grünenthal GmbH filed Critical Grünenthal GmbH
Publication of HRP20190231T1 publication Critical patent/HRP20190231T1/hr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/12—Carboxylic acids; Salts or anhydrides thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/08—Solutions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
HRP20190231TT 2015-03-27 2019-02-05 Stabilna formulacija za parenteralnu primjenu tapentadola HRP20190231T1 (hr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP15161487 2015-03-27
EP15169730 2015-05-28
EP16714327.0A EP3273953B1 (en) 2015-03-27 2016-03-23 Stable formulation for parenteral administration of tapentadol
PCT/EP2016/056376 WO2016156147A1 (en) 2015-03-27 2016-03-23 Stable formulation for parenteral administration of tapentadol

Publications (1)

Publication Number Publication Date
HRP20190231T1 true HRP20190231T1 (hr) 2019-04-05

Family

ID=55661386

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20190231TT HRP20190231T1 (hr) 2015-03-27 2019-02-05 Stabilna formulacija za parenteralnu primjenu tapentadola

Country Status (28)

Country Link
US (2) US20160279078A1 (hr)
EP (2) EP3273953B1 (hr)
JP (1) JP6923447B2 (hr)
KR (1) KR20170132282A (hr)
CN (1) CN107847471A (hr)
AU (1) AU2016239772B2 (hr)
BR (1) BR112017018569A2 (hr)
CA (1) CA2979034A1 (hr)
CL (1) CL2017002306A1 (hr)
CO (1) CO2017009400A2 (hr)
CY (1) CY1121371T1 (hr)
DK (1) DK3273953T3 (hr)
EA (1) EA036258B1 (hr)
EC (1) ECSP17064188A (hr)
ES (2) ES2822113T3 (hr)
HK (1) HK1252705A1 (hr)
HR (1) HRP20190231T1 (hr)
HU (1) HUE042612T2 (hr)
IL (1) IL254136A0 (hr)
LT (1) LT3273953T (hr)
MX (1) MX2017012312A (hr)
PE (1) PE20171651A1 (hr)
PL (1) PL3273953T3 (hr)
PT (2) PT3479823T (hr)
RS (1) RS58301B1 (hr)
SI (1) SI3273953T1 (hr)
TW (1) TW201642843A (hr)
WO (1) WO2016156147A1 (hr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT2680832T (pt) 2011-03-04 2019-10-28 Gruenenthal Gmbh Formulação farmacêutica aquosa de tapentadol para administração oral
PT3479823T (pt) 2015-03-27 2020-09-29 Gruenenthal Gmbh Formulação estável para administração parentérica de tapentadol
MX2019003257A (es) 2016-09-23 2019-06-10 Gruenenthal Gmbh Formulacion estable para la administracion parenteral de tapentadol.
EP3585370A1 (en) 2017-02-23 2020-01-01 Grünenthal GmbH Tapentadol as local anesthetic

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Also Published As

Publication number Publication date
BR112017018569A2 (pt) 2018-04-24
SI3273953T1 (sl) 2019-03-29
ES2710299T3 (es) 2019-04-24
PT3273953T (pt) 2019-04-01
CL2017002306A1 (es) 2018-03-23
DK3273953T3 (en) 2019-03-11
LT3273953T (lt) 2019-02-25
EA201792144A1 (ru) 2018-03-30
PE20171651A1 (es) 2017-11-13
AU2016239772B2 (en) 2021-05-13
EP3273953B1 (en) 2019-01-02
ECSP17064188A (es) 2018-03-31
KR20170132282A (ko) 2017-12-01
EA036258B1 (ru) 2020-10-20
AU2016239772A1 (en) 2017-09-14
EP3479823B1 (en) 2020-09-09
JP6923447B2 (ja) 2021-08-18
CY1121371T1 (el) 2020-05-29
US11013701B2 (en) 2021-05-25
ES2822113T3 (es) 2021-04-29
EP3273953A1 (en) 2018-01-31
WO2016156147A1 (en) 2016-10-06
MX2017012312A (es) 2018-01-18
RS58301B1 (sr) 2019-03-29
EP3479823A1 (en) 2019-05-08
PL3273953T3 (pl) 2019-07-31
HUE042612T2 (hu) 2019-07-29
JP2018509462A (ja) 2018-04-05
CA2979034A1 (en) 2016-10-06
US20160279078A1 (en) 2016-09-29
IL254136A0 (en) 2017-10-31
PT3479823T (pt) 2020-09-29
CO2017009400A2 (es) 2018-01-05
HK1252705A1 (zh) 2019-05-31
TW201642843A (zh) 2016-12-16
CN107847471A (zh) 2018-03-27
US20180125800A1 (en) 2018-05-10

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