TW201119654A - Aminopyridine derivatives - Google Patents

Aminopyridine derivatives Download PDF

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Publication number
TW201119654A
TW201119654A TW099136776A TW99136776A TW201119654A TW 201119654 A TW201119654 A TW 201119654A TW 099136776 A TW099136776 A TW 099136776A TW 99136776 A TW99136776 A TW 99136776A TW 201119654 A TW201119654 A TW 201119654A
Authority
TW
Taiwan
Prior art keywords
phenyl
amino
ethyl
group
ylmethyl
Prior art date
Application number
TW099136776A
Other languages
English (en)
Chinese (zh)
Inventor
David Michael Evans
Christine Elizabeth Allan
Original Assignee
Vantia Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vantia Ltd filed Critical Vantia Ltd
Publication of TW201119654A publication Critical patent/TW201119654A/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
TW099136776A 2009-10-28 2010-10-27 Aminopyridine derivatives TW201119654A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25560609P 2009-10-28 2009-10-28
GBGB0918922.6A GB0918922D0 (en) 2009-10-28 2009-10-28 Aminopyridine derivatives

Publications (1)

Publication Number Publication Date
TW201119654A true TW201119654A (en) 2011-06-16

Family

ID=41434814

Family Applications (1)

Application Number Title Priority Date Filing Date
TW099136776A TW201119654A (en) 2009-10-28 2010-10-27 Aminopyridine derivatives

Country Status (5)

Country Link
AR (1) AR078817A1 (es)
GB (1) GB0918922D0 (es)
TW (1) TW201119654A (es)
UY (1) UY32975A (es)
WO (1) WO2011051671A1 (es)

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* Cited by examiner, † Cited by third party
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EP2665708A4 (en) * 2011-01-20 2014-07-09 Univ Colorado Regents MODULATORS OF THE TLR3 / DSRNA COMPLEX AND APPLICATIONS THEREOF
GB2510407A (en) 2013-02-04 2014-08-06 Kalvista Pharmaceuticals Ltd Aqueous suspensions of kallikrein inhibitors for parenteral administration
JP2016152772A (ja) * 2013-06-27 2016-08-25 味の素株式会社 新規うま味付与剤
WO2020094008A1 (zh) * 2018-11-06 2020-05-14 天津药物研究院有限公司 2-氧代-1，2-二氢喹啉类衍生物、其制备方法及其在医药上的应用
WO2021028645A1 (en) 2019-08-09 2021-02-18 Kalvista Pharmaceuticals Limited Plasma kallikrein inhibitors

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Also Published As

Publication number Publication date
WO2011051671A1 (en) 2011-05-05
AR078817A1 (es) 2011-12-07
GB0918922D0 (en) 2009-12-16
UY32975A (es) 2011-05-31

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