TW201105666A - Substituted 2-carboxamide cycloamino ureas - Google Patents
Substituted 2-carboxamide cycloamino ureas Download PDFInfo
- Publication number
- TW201105666A TW201105666A TW099121705A TW99121705A TW201105666A TW 201105666 A TW201105666 A TW 201105666A TW 099121705 A TW099121705 A TW 099121705A TW 99121705 A TW99121705 A TW 99121705A TW 201105666 A TW201105666 A TW 201105666A
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- Taiwan
- Prior art keywords
- leu
- group
- glu
- alkyl
- lys
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Classifications
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P3/06—Antihyperlipidemics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Epidemiology (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
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| US27002909P | 2009-07-02 | 2009-07-02 |
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| EP (1) | EP2448935B1 (OSRAM) |
| JP (1) | JP2012531456A (OSRAM) |
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| CN (1) | CN102471332A (OSRAM) |
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| MX (1) | MX2012000177A (OSRAM) |
| TW (1) | TW201105666A (OSRAM) |
| UY (1) | UY32747A (OSRAM) |
| WO (1) | WO2011000905A1 (OSRAM) |
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- 2010-06-30 UY UY0001032747A patent/UY32747A/es not_active Application Discontinuation
- 2010-07-01 JP JP2012518092A patent/JP2012531456A/ja active Pending
- 2010-07-01 AU AU2010268019A patent/AU2010268019A1/en not_active Abandoned
- 2010-07-01 WO PCT/EP2010/059352 patent/WO2011000905A1/en not_active Ceased
- 2010-07-01 BR BRPI1015909A patent/BRPI1015909A2/pt not_active IP Right Cessation
- 2010-07-01 KR KR1020127002827A patent/KR20120092552A/ko not_active Withdrawn
- 2010-07-01 AR ARP100102354A patent/AR077367A1/es unknown
- 2010-07-01 TW TW099121705A patent/TW201105666A/zh unknown
- 2010-07-01 MX MX2012000177A patent/MX2012000177A/es not_active Application Discontinuation
- 2010-07-01 CA CA2766855A patent/CA2766855A1/en not_active Abandoned
- 2010-07-01 EP EP10730435.4A patent/EP2448935B1/en not_active Not-in-force
- 2010-07-01 EA EA201200086A patent/EA201200086A1/ru unknown
- 2010-07-01 CN CN2010800300379A patent/CN102471332A/zh active Pending
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| WO2011000905A1 (en) | 2011-01-06 |
| CA2766855A1 (en) | 2011-01-06 |
| KR20120092552A (ko) | 2012-08-21 |
| EP2448935B1 (en) | 2015-06-24 |
| AU2010268019A1 (en) | 2012-01-19 |
| EA201200086A1 (ru) | 2012-07-30 |
| US20110003818A1 (en) | 2011-01-06 |
| UY32747A (es) | 2011-01-31 |
| BRPI1015909A2 (pt) | 2019-09-24 |
| AR077367A1 (es) | 2011-08-24 |
| US8293753B2 (en) | 2012-10-23 |
| MX2012000177A (es) | 2012-02-28 |
| CN102471332A (zh) | 2012-05-23 |
| JP2012531456A (ja) | 2012-12-10 |
| EP2448935A1 (en) | 2012-05-09 |
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