TW200813017A - Factor XA inhibitors - Google Patents
Factor XA inhibitors Download PDFInfo
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- TW200813017A TW200813017A TW096115906A TW96115906A TW200813017A TW 200813017 A TW200813017 A TW 200813017A TW 096115906 A TW096115906 A TW 096115906A TW 96115906 A TW96115906 A TW 96115906A TW 200813017 A TW200813017 A TW 200813017A
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
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| AU2008239659B2 (en) | 2007-04-13 | 2013-09-05 | Millennium Pharmaceuticals, Inc. | Combination anticoagulant therapy with a compound that acts as a factor Xa inhibitor |
| EP2586439A1 (en) | 2007-05-02 | 2013-05-01 | Portola Pharmaceuticals, Inc. | Combination therapy with a compound acting as a platelet ADP receptor inhibitor |
| SI2915564T1 (sl) | 2007-09-28 | 2021-03-31 | Alexion Pharmaceuticals, Inc. | Antidoti za zaviralce dejavnika Ksa in postopki njihove uporabe |
| US8455439B2 (en) | 2008-11-14 | 2013-06-04 | Portola Pharmaceuticals, Inc. | Antidotes for factor Xa inhibitors and methods of using the same in combination with blood coagulating agents |
| FI3604510T3 (fi) | 2009-03-30 | 2025-06-26 | Alexion Pharma Inc | Vastalääkkeitä tekijä xa:n estäjille ja menetelmiä niiden käyttämiseksi |
| PT2453910T (pt) | 2009-07-15 | 2016-12-07 | Portola Pharm Inc | Formulação de dose unitária de antídoto contra inibidores de fator xa para uso na prevenção de sangramento |
-
2007
- 2007-05-04 TW TW096115906A patent/TW200813017A/zh unknown
- 2007-05-04 AU AU2007247928A patent/AU2007247928B2/en not_active Ceased
- 2007-05-04 NZ NZ572418A patent/NZ572418A/en not_active IP Right Cessation
- 2007-05-04 US US11/744,735 patent/US7763608B2/en not_active Expired - Fee Related
- 2007-05-04 BR BRPI0711296-3A patent/BRPI0711296A2/pt not_active Application Discontinuation
- 2007-05-04 CN CN200780015911XA patent/CN101490036B/zh not_active Expired - Fee Related
- 2007-05-04 EA EA200802288A patent/EA015942B1/ru not_active IP Right Cessation
- 2007-05-04 AR ARP070101952A patent/AR060768A1/es unknown
- 2007-05-04 JP JP2009510100A patent/JP5227311B2/ja not_active Expired - Fee Related
- 2007-05-04 WO PCT/US2007/068262 patent/WO2007131179A1/en not_active Ceased
- 2007-05-04 MX MX2008014193A patent/MX2008014193A/es active IP Right Grant
- 2007-05-04 KR KR1020087029729A patent/KR20090010098A/ko not_active Ceased
- 2007-05-04 CA CA002651303A patent/CA2651303A1/en not_active Abandoned
- 2007-05-04 EP EP07761905.4A patent/EP2016072B1/en active Active
-
2008
- 2008-07-02 US US12/166,944 patent/US7767697B2/en not_active Expired - Fee Related
- 2008-10-23 IL IL194891A patent/IL194891A/en active IP Right Grant
- 2008-10-31 ZA ZA2008/09362A patent/ZA200809362B/en unknown
-
2010
- 2010-05-11 US US12/777,956 patent/US8063077B2/en not_active Expired - Fee Related
- 2010-10-05 ZA ZA2010/07095A patent/ZA201007095B/en unknown
-
2011
- 2011-10-10 US US13/270,170 patent/US8349873B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US8349873B2 (en) | 2013-01-08 |
| IL194891A0 (en) | 2009-08-03 |
| US20110118244A2 (en) | 2011-05-19 |
| US20070259924A1 (en) | 2007-11-08 |
| CN101490036B (zh) | 2013-07-17 |
| EA015942B1 (ru) | 2011-12-30 |
| US20120088795A1 (en) | 2012-04-12 |
| US7763608B2 (en) | 2010-07-27 |
| IL194891A (en) | 2014-06-30 |
| EP2016072B1 (en) | 2014-07-16 |
| US8063077B2 (en) | 2011-11-22 |
| US7767697B2 (en) | 2010-08-03 |
| WO2007131179A1 (en) | 2007-11-15 |
| US20100249117A1 (en) | 2010-09-30 |
| CA2651303A1 (en) | 2007-11-15 |
| JP2009536218A (ja) | 2009-10-08 |
| JP5227311B2 (ja) | 2013-07-03 |
| NZ572418A (en) | 2011-08-26 |
| CN101490036A (zh) | 2009-07-22 |
| BRPI0711296A2 (pt) | 2011-08-23 |
| ZA201007095B (en) | 2011-06-29 |
| ZA200809362B (en) | 2012-01-25 |
| MX2008014193A (es) | 2009-03-31 |
| AU2007247928B2 (en) | 2013-06-13 |
| HK1126490A1 (en) | 2009-09-04 |
| US20090030045A1 (en) | 2009-01-29 |
| AR060768A1 (es) | 2008-07-10 |
| KR20090010098A (ko) | 2009-01-28 |
| AU2007247928A1 (en) | 2007-11-15 |
| EP2016072A1 (en) | 2009-01-21 |
| EA200802288A1 (ru) | 2009-04-28 |
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