TW200804390A - Pyrrolotriazine aniline prodrug compounds useful as kinase inhibitors - Google Patents
Pyrrolotriazine aniline prodrug compounds useful as kinase inhibitors Download PDFInfo
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- TW200804390A TW200804390A TW096107889A TW96107889A TW200804390A TW 200804390 A TW200804390 A TW 200804390A TW 096107889 A TW096107889 A TW 096107889A TW 96107889 A TW96107889 A TW 96107889A TW 200804390 A TW200804390 A TW 200804390A
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| HRP20040988A2 (en) * | 2002-04-23 | 2005-06-30 | Bristol-Myers Squibb Company A Delaware (Usa) Corp | Pyrrolo-triazine aniline compounds useful as kinas |
| EA200801945A1 (ru) * | 2006-03-07 | 2009-02-27 | Бристол-Маерс Сквибб Компани | Пирролотриазинанилиновые пролекарственные соединения, полезные в качестве ингибиторов киназы |
| WO2009158446A2 (en) * | 2008-06-25 | 2009-12-30 | Bristol-Myers Squibb Company | Crystalline forms of ((((4-((5-(cyclopropylcarbamoyl)-2-methylphenyl)amino)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl)carbonyl)(propyl)carbamoyl)oxy)methyl (4-(phosphonooxy)phenyl)acetate, method of preparation and use thereof |
| WO2009158450A1 (en) * | 2008-06-25 | 2009-12-30 | Bristol-Myers Squibb Company | Crystalline forms of ((((4-((5-(cyclopropylcarbamoyl)-2-methylphenyl)amino)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl)carbonyl)(propyl)carbamoyl)oxy)methyl (4-(phosphonooxy)phenyl)acetate, preparation and use thereof |
| RU2554347C2 (ru) | 2008-08-19 | 2015-06-27 | Ксенопорт, Инк. | Пролекарства метилгидрофумарата, фармацевтические композиции с ними и способы применения |
| TW201035100A (en) | 2008-12-19 | 2010-10-01 | Cephalon Inc | Pyrrolotriazines as ALK and JAK2 inhibitors |
| CN102596921B (zh) * | 2009-09-29 | 2015-04-29 | 葛兰素集团有限公司 | 新化合物 |
| JP5752691B2 (ja) | 2009-09-29 | 2015-07-22 | グラクソ グループ リミテッドGlaxo Group Limited | 新規化合物 |
| CN102918045A (zh) | 2010-03-31 | 2013-02-06 | 百时美施贵宝公司 | 作为蛋白激酶抑制剂的取代的吡咯并三嗪 |
| WO2012031057A1 (en) | 2010-09-01 | 2012-03-08 | Bristol-Myers Squibb Company | Bms- 582949 for the treatment of resistant rheumatic disease |
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- 2007-03-05 WO PCT/US2007/063250 patent/WO2007103839A2/en not_active Ceased
- 2007-03-05 CN CNA2007800079168A patent/CN101395158A/zh active Pending
- 2007-03-05 EP EP07757860A patent/EP2001886A2/en not_active Withdrawn
- 2007-03-05 JP JP2008558486A patent/JP2009535295A/ja active Pending
- 2007-03-05 CA CA002645031A patent/CA2645031A1/en not_active Abandoned
- 2007-03-05 KR KR1020087021851A patent/KR20080107408A/ko not_active Withdrawn
- 2007-03-05 AU AU2007223342A patent/AU2007223342A1/en not_active Abandoned
- 2007-03-05 MX MX2008011136A patent/MX2008011136A/es not_active Application Discontinuation
- 2007-03-05 BR BRPI0708644-0A patent/BRPI0708644A2/pt not_active IP Right Cessation
- 2007-03-06 US US11/682,331 patent/US7572795B2/en active Active
- 2007-03-06 PE PE2007000242A patent/PE20080139A1/es not_active Application Discontinuation
- 2007-03-07 AR ARP070100944A patent/AR059778A1/es unknown
- 2007-03-07 TW TW096107889A patent/TW200804390A/zh unknown
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- 2008-08-29 NO NO20083717A patent/NO20083717L/no not_active Application Discontinuation
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2009
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI483935B (zh) * | 2009-06-25 | 2015-05-11 | Alkermes Pharma Ireland Ltd | Nh-酸性化合物之前驅藥 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20090156555A1 (en) | 2009-06-18 |
| BRPI0708644A2 (pt) | 2011-06-07 |
| CN101395158A (zh) | 2009-03-25 |
| EP2001886A2 (en) | 2008-12-17 |
| WO2007103839A2 (en) | 2007-09-13 |
| PE20080139A1 (es) | 2008-03-10 |
| US7572795B2 (en) | 2009-08-11 |
| US20070213300A1 (en) | 2007-09-13 |
| AU2007223342A1 (en) | 2007-09-13 |
| IL193653A0 (en) | 2009-08-03 |
| CA2645031A1 (en) | 2007-09-13 |
| MX2008011136A (es) | 2008-09-08 |
| WO2007103839A3 (en) | 2008-06-05 |
| AR059778A1 (es) | 2008-04-30 |
| JP2009535295A (ja) | 2009-10-01 |
| EA200801945A1 (ru) | 2009-02-27 |
| ZA200807459B (en) | 2009-11-25 |
| NO20083717L (no) | 2008-10-06 |
| KR20080107408A (ko) | 2008-12-10 |
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