ZA200807459B - Pyrrolotriazine aniline prodrugs compounds useful as kinase inhibitors - Google Patents

Pyrrolotriazine aniline prodrugs compounds useful as kinase inhibitors

Info

Publication number
ZA200807459B
ZA200807459B ZA200807459A ZA200807459A ZA200807459B ZA 200807459 B ZA200807459 B ZA 200807459B ZA 200807459 A ZA200807459 A ZA 200807459A ZA 200807459 A ZA200807459 A ZA 200807459A ZA 200807459 B ZA200807459 B ZA 200807459B
Authority
ZA
South Africa
Prior art keywords
kinase inhibitors
compounds useful
prodrugs compounds
pyrrolotriazine
aniline
Prior art date
Application number
ZA200807459A
Other languages
English (en)
Inventor
Liu Chunjian
Leftheris Katerina
Vivekananda M Vrudkhula
Lin James
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ZA200807459B publication Critical patent/ZA200807459B/xx

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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ZA200807459A 2006-03-07 2008-08-29 Pyrrolotriazine aniline prodrugs compounds useful as kinase inhibitors ZA200807459B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US77985106P 2006-03-07 2006-03-07

Publications (1)

Publication Number Publication Date
ZA200807459B true ZA200807459B (en) 2009-11-25

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ID=38475749

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ZA200807459A ZA200807459B (en) 2006-03-07 2008-08-29 Pyrrolotriazine aniline prodrugs compounds useful as kinase inhibitors

Country Status (17)

Country Link
US (2) US7572795B2 (xx)
EP (1) EP2001886A2 (xx)
JP (1) JP2009535295A (xx)
KR (1) KR20080107408A (xx)
CN (1) CN101395158A (xx)
AR (1) AR059778A1 (xx)
AU (1) AU2007223342A1 (xx)
BR (1) BRPI0708644A2 (xx)
CA (1) CA2645031A1 (xx)
EA (1) EA200801945A1 (xx)
IL (1) IL193653A0 (xx)
MX (1) MX2008011136A (xx)
NO (1) NO20083717L (xx)
PE (1) PE20080139A1 (xx)
TW (1) TW200804390A (xx)
WO (1) WO2007103839A2 (xx)
ZA (1) ZA200807459B (xx)

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