TW200302831A - Novel anti-inflammatory androstane derivative - Google Patents
Novel anti-inflammatory androstane derivative Download PDFInfo
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- TW200302831A TW200302831A TW092102383A TW92102383A TW200302831A TW 200302831 A TW200302831 A TW 200302831A TW 092102383 A TW092102383 A TW 092102383A TW 92102383 A TW92102383 A TW 92102383A TW 200302831 A TW200302831 A TW 200302831A
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- compound
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- alkyl
- solvate
- pharmaceutical formulation
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- 150000001440 androstane derivatives Chemical class 0.000 title 1
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Otolaryngology (AREA)
- Organic Chemistry (AREA)
- Emergency Medicine (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
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|---|---|---|---|
| US10/066,836 US6759398B2 (en) | 2000-08-05 | 2002-02-04 | Anti-inflammatory androstane derivative |
Publications (1)
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| TW200302831A true TW200302831A (en) | 2003-08-16 |
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| TW092102383A TW200302831A (en) | 2002-02-04 | 2003-02-06 | Novel anti-inflammatory androstane derivative |
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| JP (2) | JP2005527496A (https=) |
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| MY (1) | MY139577A (https=) |
| TW (1) | TW200302831A (https=) |
| WO (1) | WO2003066036A1 (https=) |
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-
2002
- 2002-02-04 US US10/066,836 patent/US6759398B2/en not_active Expired - Lifetime
-
2003
- 2003-02-04 WO PCT/GB2003/000467 patent/WO2003066036A1/en not_active Ceased
- 2003-02-04 AU AU2003207016A patent/AU2003207016A1/en not_active Abandoned
- 2003-02-04 EP EP10178712A patent/EP2363121A1/en not_active Withdrawn
- 2003-02-04 US US10/503,417 patent/US20050164997A1/en not_active Abandoned
- 2003-02-04 JP JP2003565460A patent/JP2005527496A/ja active Pending
- 2003-02-04 EP EP03704756A patent/EP1471900A1/en not_active Withdrawn
- 2003-02-05 MY MYPI20030385A patent/MY139577A/en unknown
- 2003-02-06 TW TW092102383A patent/TW200302831A/zh unknown
-
2010
- 2010-08-06 JP JP2010177124A patent/JP2010280701A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| MY139577A (en) | 2009-10-30 |
| EP1471900A1 (en) | 2004-11-03 |
| JP2005527496A (ja) | 2005-09-15 |
| US20050164997A1 (en) | 2005-07-28 |
| EP2363121A1 (en) | 2011-09-07 |
| US20020177581A1 (en) | 2002-11-28 |
| WO2003066036A1 (en) | 2003-08-14 |
| AU2003207016A1 (en) | 2003-09-02 |
| US6759398B2 (en) | 2004-07-06 |
| JP2010280701A (ja) | 2010-12-16 |
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