TR199901484T2 - 2-Amino-2-imidazolin, guanidin ve 2-amino-3,4,5,6-tetrahidropirimidin türevleri hazirlama islemi. - Google Patents

2-Amino-2-imidazolin, guanidin ve 2-amino-3,4,5,6-tetrahidropirimidin türevleri hazirlama islemi.

Info

Publication number
TR199901484T2
TR199901484T2 TR1999/01484T TR9901484T TR199901484T2 TR 199901484 T2 TR199901484 T2 TR 199901484T2 TR 1999/01484 T TR1999/01484 T TR 1999/01484T TR 9901484 T TR9901484 T TR 9901484T TR 199901484 T2 TR199901484 T2 TR 199901484T2
Authority
TR
Turkey
Prior art keywords
amino
tetrahidropirimidin
rlama
revleri
lemi
Prior art date
Application number
TR1999/01484T
Other languages
English (en)
Inventor
Godlewski Michael
Rees Klopfenstein Sean
Reddy Mundla Screenivasa
Lee Seibel William
Original Assignee
The Procter & Gamble Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by The Procter & Gamble Company filed Critical The Procter & Gamble Company
Publication of TR199901484T2 publication Critical patent/TR199901484T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44—Nitrogen atoms not forming part of a nitro radical
    • C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

(Formül(B), Formül(1)); Bu bulus istemlerde açiklandigi gibi B yapisini haiz bir bilesik veya totomerlerini hazirlamak için bir islem sunmaktadir. Bu islem (1) genel yapisina sahip bir ara madde hazirlama adimindan olusur; burada R metil, etil ve benzil arasindan seçilir; R3 ise -O-R5 veya -R6'dir.
TR1999/01484T 1996-11-25 1997-11-25 2-Amino-2-imidazolin, guanidin ve 2-amino-3,4,5,6-tetrahidropirimidin türevleri hazirlama islemi. TR199901484T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US3431896P 1996-11-25 1996-11-25

Publications (1)

Publication Number Publication Date
TR199901484T2 true TR199901484T2 (tr) 1999-09-21

Family

ID=21875679

Family Applications (1)

Application Number Title Priority Date Filing Date
TR1999/01484T TR199901484T2 (tr) 1996-11-25 1997-11-25 2-Amino-2-imidazolin, guanidin ve 2-amino-3,4,5,6-tetrahidropirimidin türevleri hazirlama islemi.

Country Status (21)

Country Link
EP (1) EP0944603B1 (tr)
JP (1) JP2001506605A (tr)
KR (1) KR20000069132A (tr)
AR (1) AR008920A1 (tr)
AT (1) ATE232851T1 (tr)
AU (1) AU732056B2 (tr)
BR (1) BR9713296A (tr)
CA (1) CA2272690C (tr)
CO (1) CO4910165A1 (tr)
CZ (1) CZ183599A3 (tr)
DE (1) DE69719210T2 (tr)
DK (1) DK0944603T3 (tr)
ID (1) ID22896A (tr)
IL (1) IL130095A0 (tr)
NO (1) NO312721B1 (tr)
PE (1) PE28099A1 (tr)
SK (1) SK69899A3 (tr)
TR (1) TR199901484T2 (tr)
TW (1) TW472043B (tr)
WO (1) WO1998023595A1 (tr)
ZA (1) ZA9710581B (tr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996004270A1 (en) 1994-08-04 1996-02-15 Synaptic Pharmaceutical Corporation Novel benzimidazole derivatives
US6495583B1 (en) 1997-03-25 2002-12-17 Synaptic Pharmaceutical Corporation Benzimidazole derivatives
US20040167194A1 (en) 2003-02-20 2004-08-26 Randall Jared Lynn Methods of making 6-[(4,5-Dihydro-1H-imidazol-2-yl)amino-]-7-methyl-1H-benzimidazole-4-carbonitrile and its preferred salt form
US11077053B2 (en) 2018-08-21 2021-08-03 Allergan, Inc. Alpha-2-adrenergic receptor agonists for treatment of presbyopia, visual glare, visual starbursts, visual halos and night myopia

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670807A1 (de) * 1967-02-17 1971-03-11 Bayer Ag Verfahren zur Herstellung von cyclischen Guanidinen
DE2854659A1 (de) * 1978-12-18 1980-07-10 Boehringer Sohn Ingelheim Neue 3,4-disubstituierte 2-phenylimino-imidazolidine, deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zu deren herstellung

Also Published As

Publication number Publication date
CZ183599A3 (cs) 1999-10-13
JP2001506605A (ja) 2001-05-22
EP0944603A1 (en) 1999-09-29
PE28099A1 (es) 1999-03-31
ID22896A (id) 1999-12-16
DK0944603T3 (da) 2003-06-16
BR9713296A (pt) 1999-10-26
KR20000069132A (ko) 2000-11-25
CO4910165A1 (es) 2000-04-24
IL130095A0 (en) 2000-02-29
NO992501D0 (no) 1999-05-25
DE69719210D1 (de) 2003-03-27
AU7402198A (en) 1998-06-22
AU732056B2 (en) 2001-04-12
ATE232851T1 (de) 2003-03-15
EP0944603B1 (en) 2003-02-19
NO992501L (no) 1999-07-22
ZA9710581B (en) 1998-06-12
AR008920A1 (es) 2000-02-23
DE69719210T2 (de) 2004-02-12
NO312721B1 (no) 2002-06-24
TW472043B (en) 2002-01-11
WO1998023595A1 (en) 1998-06-04
CA2272690C (en) 2004-07-13
SK69899A3 (en) 2000-01-18
CA2272690A1 (en) 1998-06-04

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