TR199802661T2 - 5-HT-2C Resept�r kar��tlar� olarak faydal� indolin t�revleri. - Google Patents
5-HT-2C Resept�r kar��tlar� olarak faydal� indolin t�revleri.Info
- Publication number
- TR199802661T2 TR199802661T2 TR1998/02661T TR9802661T TR199802661T2 TR 199802661 T2 TR199802661 T2 TR 199802661T2 TR 1998/02661 T TR1998/02661 T TR 1998/02661T TR 9802661 T TR9802661 T TR 9802661T TR 199802661 T2 TR199802661 T2 TR 199802661T2
- Authority
- TR
- Turkey
- Prior art keywords
- receptor antagonists
- derivatives useful
- indoline derivatives
- alkyl
- indoline
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9612883.0A GB9612883D0 (en) | 1996-06-20 | 1996-06-20 | Novel compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR199802661T2 true TR199802661T2 (xx) | 1999-03-22 |
Family
ID=10795575
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR1998/02661T TR199802661T2 (xx) | 1996-06-20 | 1997-06-16 | 5-HT-2C Resept�r kar��tlar� olarak faydal� indolin t�revleri. |
Country Status (33)
| Country | Link |
|---|---|
| US (1) | US6369060B1 (OSRAM) |
| EP (1) | EP0912554B1 (OSRAM) |
| JP (1) | JP2000512306A (OSRAM) |
| KR (1) | KR20000022045A (OSRAM) |
| CN (1) | CN1229408A (OSRAM) |
| AP (2) | AP9801410A0 (OSRAM) |
| AR (1) | AR008243A1 (OSRAM) |
| AT (1) | ATE228514T1 (OSRAM) |
| AU (1) | AU718597B2 (OSRAM) |
| BG (1) | BG103089A (OSRAM) |
| BR (1) | BR9709911A (OSRAM) |
| CA (1) | CA2258240A1 (OSRAM) |
| CO (1) | CO4890847A1 (OSRAM) |
| CZ (1) | CZ420598A3 (OSRAM) |
| DE (1) | DE69717449T2 (OSRAM) |
| DZ (1) | DZ2250A1 (OSRAM) |
| EA (1) | EA001780B1 (OSRAM) |
| ES (1) | ES2187783T3 (OSRAM) |
| GB (1) | GB9612883D0 (OSRAM) |
| HU (1) | HUP9903439A3 (OSRAM) |
| ID (1) | ID19433A (OSRAM) |
| IL (1) | IL127417A0 (OSRAM) |
| MA (1) | MA24214A1 (OSRAM) |
| NO (1) | NO985972D0 (OSRAM) |
| NZ (1) | NZ333229A (OSRAM) |
| OA (1) | OA10944A (OSRAM) |
| PE (1) | PE86698A1 (OSRAM) |
| PL (1) | PL330796A1 (OSRAM) |
| SK (1) | SK282706B6 (OSRAM) |
| TR (1) | TR199802661T2 (OSRAM) |
| TW (1) | TW382015B (OSRAM) |
| WO (1) | WO1997048699A1 (OSRAM) |
| ZA (1) | ZA975415B (OSRAM) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999043650A2 (en) * | 1998-02-25 | 1999-09-02 | Smithkline Beecham Plc | Process(es) for the preparation of 6-trifluoromethyl-indoline derivatives |
| GB0019950D0 (en) * | 2000-08-12 | 2000-09-27 | Smithkline Beecham Plc | Compounds |
| AU2002346507A1 (en) | 2001-11-28 | 2003-06-10 | Pharmacia And Upjohn Company | Benzazepine derivatives and their use as 5-ht ligands |
| CA2475254A1 (en) * | 2002-03-04 | 2003-09-18 | Pharmacia & Upjohn Company | Pyridinyloxy derivatives as 5-ht receptor ligands |
| KR101062376B1 (ko) * | 2008-04-10 | 2011-09-06 | 한국화학연구원 | 신규 인돌 카르복실산 비스피리딜 카르복사마이드 유도체,이의 제조방법 및 이를 유효성분으로 함유하는 조성물 |
| WO2010083044A1 (en) | 2009-01-16 | 2010-07-22 | Massachusetts Institute Of Technology | Diagnosis and treatment of autism spectrum disorders |
| ES2847883T3 (es) | 2010-12-17 | 2021-08-04 | Glaxo Group Ltd | Uso de inhibidores de LP-PLA2 en el tratamiento y prevención de enfermedades oculares |
| WO2014046544A1 (en) | 2012-09-21 | 2014-03-27 | Aapa B.V. | Substituted 3-heteroaryloxy-3-(hetero)aryl-propylamines as serotonin transporter and serotonin ht2c receptor modulators |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1989001333A1 (en) * | 1987-08-07 | 1989-02-23 | The Australian National University | IMIDAZO[1,2-b]PYRIDAZINES |
| NZ254785A (en) | 1992-08-20 | 1995-09-26 | Smithkline Beecham Plc | Heterocyclically-condensed indoles and medicaments |
| GB9313913D0 (en) * | 1993-07-06 | 1993-08-18 | Smithkline Beecham Plc | Novel compounds |
| FI973205L (fi) | 1995-02-02 | 1997-10-01 | Smithkline Beecham Plc | Indolijohdannaisia 5-HT-reseptoriantagonisteina |
| GB9607219D0 (en) * | 1996-04-04 | 1996-06-12 | Smithkline Beecham Plc | Novel compounds |
| GB9615767D0 (en) * | 1996-07-26 | 1996-09-04 | Smithkline Beecham Plc | Novel treatment |
-
1996
- 1996-06-20 GB GBGB9612883.0A patent/GB9612883D0/en active Pending
-
1997
- 1997-06-16 DE DE69717449T patent/DE69717449T2/de not_active Expired - Fee Related
- 1997-06-16 CA CA002258240A patent/CA2258240A1/en not_active Abandoned
- 1997-06-16 WO PCT/EP1997/003156 patent/WO1997048699A1/en not_active Ceased
- 1997-06-16 CN CN97197311A patent/CN1229408A/zh active Pending
- 1997-06-16 EA EA199900043A patent/EA001780B1/ru not_active IP Right Cessation
- 1997-06-16 HU HU9903439A patent/HUP9903439A3/hu unknown
- 1997-06-16 BR BR9709911A patent/BR9709911A/pt unknown
- 1997-06-16 CZ CZ984205A patent/CZ420598A3/cs unknown
- 1997-06-16 JP JP10502259A patent/JP2000512306A/ja active Pending
- 1997-06-16 TR TR1998/02661T patent/TR199802661T2/xx unknown
- 1997-06-16 AT AT97928224T patent/ATE228514T1/de not_active IP Right Cessation
- 1997-06-16 NZ NZ333229A patent/NZ333229A/xx unknown
- 1997-06-16 PL PL97330796A patent/PL330796A1/xx unknown
- 1997-06-16 KR KR1019980710443A patent/KR20000022045A/ko not_active Ceased
- 1997-06-16 ES ES97928224T patent/ES2187783T3/es not_active Expired - Lifetime
- 1997-06-16 AU AU32602/97A patent/AU718597B2/en not_active Ceased
- 1997-06-16 AP APAP/P/1998/001410A patent/AP9801410A0/en unknown
- 1997-06-16 EP EP97928224A patent/EP0912554B1/en not_active Expired - Lifetime
- 1997-06-16 US US09/202,780 patent/US6369060B1/en not_active Expired - Fee Related
- 1997-06-16 SK SK1752-98A patent/SK282706B6/sk unknown
- 1997-06-16 IL IL12741797A patent/IL127417A0/xx unknown
- 1997-06-18 DZ DZ970100A patent/DZ2250A1/fr active
- 1997-06-18 AP APAP/P/1997/001037A patent/AP745A/en active
- 1997-06-18 PE PE1997000510A patent/PE86698A1/es not_active Application Discontinuation
- 1997-06-18 AR ARP970102673A patent/AR008243A1/es unknown
- 1997-06-18 MA MA24666A patent/MA24214A1/fr unknown
- 1997-06-19 TW TW086108551A patent/TW382015B/zh not_active IP Right Cessation
- 1997-06-19 ZA ZA975415A patent/ZA975415B/xx unknown
- 1997-06-20 ID IDP972126A patent/ID19433A/id unknown
- 1997-06-20 CO CO97034431A patent/CO4890847A1/es unknown
-
1998
- 1998-12-18 OA OA9800245A patent/OA10944A/en unknown
- 1998-12-18 NO NO985972A patent/NO985972D0/no unknown
-
1999
- 1999-01-15 BG BG103089A patent/BG103089A/xx unknown
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